CL2004000610A1 - Compuestos heterociclicos, inhibidores de la proteina tirosina quinasa, utiles para preparar un medicamento para tratar artritis reumatoide, esclerosis multiple, enfermedad inflamatoria del intestino, lupus, cancer y otras. - Google Patents

Compuestos heterociclicos, inhibidores de la proteina tirosina quinasa, utiles para preparar un medicamento para tratar artritis reumatoide, esclerosis multiple, enfermedad inflamatoria del intestino, lupus, cancer y otras.

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Publication number
CL2004000610A1
CL2004000610A1 CL200400610A CL2004000610A CL2004000610A1 CL 2004000610 A1 CL2004000610 A1 CL 2004000610A1 CL 200400610 A CL200400610 A CL 200400610A CL 2004000610 A CL2004000610 A CL 2004000610A CL 2004000610 A1 CL2004000610 A1 CL 2004000610A1
Authority
CL
Chile
Prior art keywords
lupus
intestine
inhibitors
cancer
treat
Prior art date
Application number
CL200400610A
Other languages
English (en)
Inventor
Jagabandhu Padmanabha Rame Das
Original Assignee
Bristol Myers Squibb Co
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Family has litigation
First worldwide family litigation filed litigation Critical https://patents.darts-ip.com/?family=33096777&utm_source=google_patent&utm_medium=platform_link&utm_campaign=public_patent_search&patent=CL2004000610(A1) "Global patent litigation dataset” by Darts-ip is licensed under a Creative Commons Attribution 4.0 International License.
Application filed by Bristol Myers Squibb Co filed Critical Bristol Myers Squibb Co
Publication of CL2004000610A1 publication Critical patent/CL2004000610A1/es

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    • A—HUMAN NECESSITIES
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    • A61K31/33—Heterocyclic compounds
    • A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/41—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having five-membered rings with two or more ring hetero atoms, at least one of which being nitrogen, e.g. tetrazole
    • A61K31/425—Thiazoles
    • A61K31/427—Thiazoles not condensed and containing further heterocyclic rings
    • A—HUMAN NECESSITIES
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    • A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/495—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with two or more nitrogen atoms as the only ring heteroatoms, e.g. piperazine or tetrazines
    • A61K31/505—Pyrimidines; Hydrogenated pyrimidines, e.g. trimethoprim
    • A61K31/506—Pyrimidines; Hydrogenated pyrimidines, e.g. trimethoprim not condensed and containing further heterocyclic rings
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    • C07—ORGANIC CHEMISTRY
    • C07C—ACYCLIC OR CARBOCYCLIC COMPOUNDS
    • C07C237/00—Carboxylic acid amides, the carbon skeleton of the acid part being further substituted by amino groups
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    • C07D213/04—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members having three double bonds between ring members or between ring members and non-ring members having no bond between the ring nitrogen atom and a non-ring member or having only hydrogen or carbon atoms directly attached to the ring nitrogen atom
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    • C—CHEMISTRY; METALLURGY
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    • C07D231/10—Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings not condensed with other rings having two or three double bonds between ring members or between ring members and non-ring members
    • C07D231/14—Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings not condensed with other rings having two or three double bonds between ring members or between ring members and non-ring members with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
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    • C07D233/54—Heterocyclic compounds containing 1,3-diazole or hydrogenated 1,3-diazole rings, not condensed with other rings having two double bonds between ring members or between ring members and non-ring members
    • C07D233/66—Heterocyclic compounds containing 1,3-diazole or hydrogenated 1,3-diazole rings, not condensed with other rings having two double bonds between ring members or between ring members and non-ring members with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
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    • C07D239/24—Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings not condensed with other rings having three or more double bonds between ring members or between ring members and non-ring members
    • C07D239/28—Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings not condensed with other rings having three or more double bonds between ring members or between ring members and non-ring members with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, directly attached to ring carbon atoms
    • C07D239/32—One oxygen, sulfur or nitrogen atom
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    • C07D263/34—Heterocyclic compounds containing 1,3-oxazole or hydrogenated 1,3-oxazole rings not condensed with other rings having two or three double bonds between ring members or between ring members and non-ring members with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
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CL200400610A 2003-03-24 2004-03-23 Compuestos heterociclicos, inhibidores de la proteina tirosina quinasa, utiles para preparar un medicamento para tratar artritis reumatoide, esclerosis multiple, enfermedad inflamatoria del intestino, lupus, cancer y otras. CL2004000610A1 (es)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
US10/395,503 US7125875B2 (en) 1999-04-15 2003-03-24 Cyclic protein tyrosine kinase inhibitors

Publications (1)

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CL2004000610A1 true CL2004000610A1 (es) 2005-05-06

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CL200400610A CL2004000610A1 (es) 2003-03-24 2004-03-23 Compuestos heterociclicos, inhibidores de la proteina tirosina quinasa, utiles para preparar un medicamento para tratar artritis reumatoide, esclerosis multiple, enfermedad inflamatoria del intestino, lupus, cancer y otras.

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US (1) US7125875B2 (es)
EP (1) EP1610780B2 (es)
JP (1) JP2006523216A (es)
KR (1) KR101070101B1 (es)
CN (2) CN1764454A (es)
AR (1) AR044506A1 (es)
AT (1) ATE464898T1 (es)
AU (1) AU2004223828B2 (es)
BR (1) BRPI0408782A (es)
CA (1) CA2519898C (es)
CL (1) CL2004000610A1 (es)
CY (1) CY1110225T1 (es)
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