CL2003002353A1 - Compuestos derivados de diaminotriazoles, inhibidores d ela proteina quinasa; composicion farmaceutica; procedimiento de preparacion; y su uso del compuesto en el tratamiento de enfermedades de desordenes alergicos, proliferacion, autoinmunes, condic - Google Patents
Compuestos derivados de diaminotriazoles, inhibidores d ela proteina quinasa; composicion farmaceutica; procedimiento de preparacion; y su uso del compuesto en el tratamiento de enfermedades de desordenes alergicos, proliferacion, autoinmunes, condicInfo
- Publication number
- CL2003002353A1 CL2003002353A1 CL200302353A CL2003002353A CL2003002353A1 CL 2003002353 A1 CL2003002353 A1 CL 2003002353A1 CL 200302353 A CL200302353 A CL 200302353A CL 2003002353 A CL2003002353 A CL 2003002353A CL 2003002353 A1 CL2003002353 A1 CL 2003002353A1
- Authority
- CL
- Chile
- Prior art keywords
- diaminotriazols
- condic
- autoimmunes
- quinasa
- proteina
- Prior art date
Links
- 150000001875 compounds Chemical class 0.000 title 2
- 208000037265 diseases, disorders, signs and symptoms Diseases 0.000 title 2
- NVKAWKQGWWIWPM-ABEVXSGRSA-N 17-β-hydroxy-5-α-Androstan-3-one Chemical compound C1C(=O)CC[C@]2(C)[C@H]3CC[C@](C)([C@H](CC4)O)[C@@H]4[C@@H]3CC[C@H]21 NVKAWKQGWWIWPM-ABEVXSGRSA-N 0.000 title 1
- 230000000172 allergic effect Effects 0.000 title 1
- 208000010668 atopic eczema Diseases 0.000 title 1
- 201000010099 disease Diseases 0.000 title 1
- 239000003112 inhibitor Substances 0.000 title 1
- 238000000034 method Methods 0.000 title 1
- 239000008194 pharmaceutical composition Substances 0.000 title 1
- 230000035755 proliferation Effects 0.000 title 1
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- C07D401/02—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings
- C07D401/04—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings directly linked by a ring-member-to-ring-member bond
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- C07D487/02—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00 in which the condensed system contains two hetero rings
- C07D487/04—Ortho-condensed systems
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D495/00—Heterocyclic compounds containing in the condensed system at least one hetero ring having sulfur atoms as the only ring hetero atoms
- C07D495/02—Heterocyclic compounds containing in the condensed system at least one hetero ring having sulfur atoms as the only ring hetero atoms in which the condensed system contains two hetero rings
- C07D495/04—Ortho-condensed systems
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| US42668102P | 2002-11-15 | 2002-11-15 | |
| US44770503P | 2003-02-11 | 2003-02-11 |
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| CL200302353A CL2003002353A1 (es) | 2002-11-15 | 2003-11-14 | Compuestos derivados de diaminotriazoles, inhibidores d ela proteina quinasa; composicion farmaceutica; procedimiento de preparacion; y su uso del compuesto en el tratamiento de enfermedades de desordenes alergicos, proliferacion, autoinmunes, condic |
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| DK113716B (da) * | 1960-07-30 | 1969-04-21 | Takeda Chemical Industries Ltd | Fremgangsmåde til fremstilling af 1-[pyrimidinyl-(2)]-guanazolforbindelser eller salte deraf. |
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| CA2309690A1 (en) * | 1997-11-11 | 1999-05-20 | Pfizer Products Inc. | Thienopyrimidine and thienopyridine derivatives useful as anticancer agents |
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| JP2003525201A (ja) | 1998-08-20 | 2003-08-26 | スミスクライン・ビーチャム・コーポレイション | 新規な置換トリアゾール化合物 |
| WO2000025780A1 (en) * | 1998-10-29 | 2000-05-11 | Bristol-Myers Squibb Company | Compounds derived from an amine nucleus that are inhibitors of impdh enzyme |
| US6596747B2 (en) * | 1998-10-29 | 2003-07-22 | Bristol-Myers Squibb Company | Compounds derived from an amine nucleus and pharmaceutical compositions comprising same |
| CA2369076A1 (en) * | 2000-02-05 | 2001-08-09 | Vertex Pharmaceuticals Incorporated | Pyrazole compositions useful as inhibitors of erk |
| DE60120494T2 (de) * | 2000-12-22 | 2006-12-21 | Ortho-Mcneil Pharmaceutical, Inc. | Substituieten triazoldiamin derivaten und ihre verwendung als kinase inhibitoren |
| DE10123586A1 (de) * | 2001-05-08 | 2002-11-28 | Schering Ag | 3,5-Diamino-1,2,4-triazole als Kinase Inhibitoren |
| CL2003002353A1 (es) * | 2002-11-15 | 2005-02-04 | Vertex Pharma | Compuestos derivados de diaminotriazoles, inhibidores d ela proteina quinasa; composicion farmaceutica; procedimiento de preparacion; y su uso del compuesto en el tratamiento de enfermedades de desordenes alergicos, proliferacion, autoinmunes, condic |
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2003
- 2003-11-14 CL CL200302353A patent/CL2003002353A1/es unknown
- 2003-11-14 AR ARP030104218A patent/AR042052A1/es unknown
- 2003-11-14 TW TW092132032A patent/TWI335913B/zh not_active IP Right Cessation
- 2003-11-17 ES ES03789812T patent/ES2318189T3/es not_active Expired - Lifetime
- 2003-11-17 US US10/715,111 patent/US7279469B2/en not_active Expired - Fee Related
- 2003-11-17 SI SI200331537T patent/SI1562589T1/sl unknown
- 2003-11-17 NZ NZ540662A patent/NZ540662A/en unknown
- 2003-11-17 CA CA002505789A patent/CA2505789A1/en not_active Abandoned
- 2003-11-17 AT AT03789812T patent/ATE419849T1/de active
- 2003-11-17 MX MXPA05005223A patent/MXPA05005223A/es unknown
- 2003-11-17 DK DK03789812T patent/DK1562589T3/da active
- 2003-11-17 JP JP2004570619A patent/JP4783020B2/ja not_active Expired - Fee Related
- 2003-11-17 EP EP03789812A patent/EP1562589B1/en not_active Expired - Lifetime
- 2003-11-17 DE DE60325761T patent/DE60325761D1/de not_active Expired - Lifetime
- 2003-11-17 RU RU2005118418/04A patent/RU2350606C2/ru not_active IP Right Cessation
- 2003-11-17 BR BR0316350-4A patent/BR0316350A/pt not_active IP Right Cessation
- 2003-11-17 AU AU2003294329A patent/AU2003294329B2/en not_active Ceased
- 2003-11-17 PT PT03789812T patent/PT1562589E/pt unknown
- 2003-11-17 KR KR1020057008795A patent/KR20060013480A/ko not_active Ceased
- 2003-11-17 PL PL377825A patent/PL377825A1/pl not_active Application Discontinuation
- 2003-11-17 WO PCT/US2003/036849 patent/WO2004046120A2/en not_active Ceased
-
2005
- 2005-06-10 NO NO20052888A patent/NO20052888L/no not_active Application Discontinuation
-
2007
- 2007-07-09 US US11/774,702 patent/US7902239B2/en not_active Expired - Fee Related
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2011
- 2011-04-05 JP JP2011084103A patent/JP2011132263A/ja not_active Withdrawn
Also Published As
| Publication number | Publication date |
|---|---|
| JP2006515313A (ja) | 2006-05-25 |
| WO2004046120A2 (en) | 2004-06-03 |
| MXPA05005223A (es) | 2010-09-07 |
| AU2003294329A1 (en) | 2004-06-15 |
| KR20060013480A (ko) | 2006-02-10 |
| NO20052888L (no) | 2005-08-12 |
| AR042052A1 (es) | 2005-06-08 |
| TWI335913B (en) | 2011-01-11 |
| DE60325761D1 (de) | 2009-02-26 |
| WO2004046120A3 (en) | 2004-08-12 |
| JP4783020B2 (ja) | 2011-09-28 |
| US20080014189A1 (en) | 2008-01-17 |
| EP1562589B1 (en) | 2009-01-07 |
| EP1562589A2 (en) | 2005-08-17 |
| ATE419849T1 (de) | 2009-01-15 |
| PT1562589E (pt) | 2009-04-15 |
| JP2011132263A (ja) | 2011-07-07 |
| PL377825A1 (pl) | 2006-02-20 |
| DK1562589T3 (da) | 2009-02-16 |
| US20040214817A1 (en) | 2004-10-28 |
| CA2505789A1 (en) | 2004-06-03 |
| TW200413334A (en) | 2004-08-01 |
| RU2350606C2 (ru) | 2009-03-27 |
| RU2005118418A (ru) | 2006-02-10 |
| SI1562589T1 (sl) | 2009-06-30 |
| BR0316350A (pt) | 2005-09-27 |
| NO20052888D0 (no) | 2005-06-10 |
| NZ540662A (en) | 2008-04-30 |
| US7902239B2 (en) | 2011-03-08 |
| AU2003294329B2 (en) | 2010-04-29 |
| ES2318189T3 (es) | 2009-05-01 |
| US7279469B2 (en) | 2007-10-09 |
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