ATE419849T1 - Diaminotriazole derivate und deren verwendung als protein kinase inhibitoren - Google Patents
Diaminotriazole derivate und deren verwendung als protein kinase inhibitorenInfo
- Publication number
- ATE419849T1 ATE419849T1 AT03789812T AT03789812T ATE419849T1 AT E419849 T1 ATE419849 T1 AT E419849T1 AT 03789812 T AT03789812 T AT 03789812T AT 03789812 T AT03789812 T AT 03789812T AT E419849 T1 ATE419849 T1 AT E419849T1
- Authority
- AT
- Austria
- Prior art keywords
- diaminotriazole
- derivatives
- protein kinase
- kinase inhibitors
- inhibitors
- Prior art date
Links
- DQSBZDLZCZUJCJ-UHFFFAOYSA-N 2h-triazole-4,5-diamine Chemical class NC=1N=NNC=1N DQSBZDLZCZUJCJ-UHFFFAOYSA-N 0.000 title 1
- 229940045988 antineoplastic drug protein kinase inhibitors Drugs 0.000 title 1
- 239000003909 protein kinase inhibitor Substances 0.000 title 1
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- C07D401/04—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings directly linked by a ring-member-to-ring-member bond
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| DK113716B (da) * | 1960-07-30 | 1969-04-21 | Takeda Chemical Industries Ltd | Fremgangsmåde til fremstilling af 1-[pyrimidinyl-(2)]-guanazolforbindelser eller salte deraf. |
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| NZ520093A (en) * | 1997-11-11 | 2004-03-26 | Pfizer Prod Inc | Thienopyrimidine and thienopyridine derivatives useful as anticancer agents |
| JP2002510033A (ja) * | 1998-01-12 | 2002-04-02 | ザ・サルク・インスティチュート | 二重微小dnaを有する細胞を処理するための組成物およびその処理方法 |
| US6599910B1 (en) | 1998-08-20 | 2003-07-29 | Smithkline Beecham Corporation | Substituted triazole compounds |
| AU764479B2 (en) * | 1998-10-29 | 2003-08-21 | Bristol-Myers Squibb Company | Compounds derived from an amine nucleus that are inhibitors of IMPDH enzyme |
| US6596747B2 (en) * | 1998-10-29 | 2003-07-22 | Bristol-Myers Squibb Company | Compounds derived from an amine nucleus and pharmaceutical compositions comprising same |
| WO2001056993A2 (en) * | 2000-02-05 | 2001-08-09 | Vertex Pharmaceuticals Incorporated | Pyrazole compositions useful as inhibitors of erk |
| PT1355889E (pt) * | 2000-12-22 | 2006-09-29 | Ortho Mcneil Pharm Inc | Derivados diamina triazole substituidos como inibidores de cinase |
| DE10123586A1 (de) * | 2001-05-08 | 2002-11-28 | Schering Ag | 3,5-Diamino-1,2,4-triazole als Kinase Inhibitoren |
| TWI335913B (en) * | 2002-11-15 | 2011-01-11 | Vertex Pharma | Diaminotriazoles useful as inhibitors of protein kinases |
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2003
- 2003-11-14 TW TW092132032A patent/TWI335913B/zh not_active IP Right Cessation
- 2003-11-14 AR ARP030104218A patent/AR042052A1/es unknown
- 2003-11-14 CL CL200302353A patent/CL2003002353A1/es unknown
- 2003-11-17 NZ NZ540662A patent/NZ540662A/en unknown
- 2003-11-17 RU RU2005118418/04A patent/RU2350606C2/ru not_active IP Right Cessation
- 2003-11-17 DK DK03789812T patent/DK1562589T3/da active
- 2003-11-17 EP EP03789812A patent/EP1562589B1/de not_active Expired - Lifetime
- 2003-11-17 US US10/715,111 patent/US7279469B2/en not_active Expired - Fee Related
- 2003-11-17 CA CA002505789A patent/CA2505789A1/en not_active Abandoned
- 2003-11-17 AT AT03789812T patent/ATE419849T1/de active
- 2003-11-17 ES ES03789812T patent/ES2318189T3/es not_active Expired - Lifetime
- 2003-11-17 JP JP2004570619A patent/JP4783020B2/ja not_active Expired - Fee Related
- 2003-11-17 PT PT03789812T patent/PT1562589E/pt unknown
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- 2003-11-17 MX MXPA05005223A patent/MXPA05005223A/es unknown
- 2003-11-17 KR KR1020057008795A patent/KR20060013480A/ko not_active Ceased
- 2003-11-17 DE DE60325761T patent/DE60325761D1/de not_active Expired - Lifetime
- 2003-11-17 PL PL377825A patent/PL377825A1/pl not_active Application Discontinuation
- 2003-11-17 SI SI200331537T patent/SI1562589T1/sl unknown
- 2003-11-17 WO PCT/US2003/036849 patent/WO2004046120A2/en not_active Ceased
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|---|---|
| NZ540662A (en) | 2008-04-30 |
| DE60325761D1 (de) | 2009-02-26 |
| ES2318189T3 (es) | 2009-05-01 |
| AU2003294329B2 (en) | 2010-04-29 |
| CL2003002353A1 (es) | 2005-02-04 |
| US20080014189A1 (en) | 2008-01-17 |
| US20040214817A1 (en) | 2004-10-28 |
| NO20052888L (no) | 2005-08-12 |
| TWI335913B (en) | 2011-01-11 |
| CA2505789A1 (en) | 2004-06-03 |
| PT1562589E (pt) | 2009-04-15 |
| DK1562589T3 (da) | 2009-02-16 |
| JP2006515313A (ja) | 2006-05-25 |
| RU2005118418A (ru) | 2006-02-10 |
| NO20052888D0 (no) | 2005-06-10 |
| WO2004046120A2 (en) | 2004-06-03 |
| AR042052A1 (es) | 2005-06-08 |
| WO2004046120A3 (en) | 2004-08-12 |
| AU2003294329A1 (en) | 2004-06-15 |
| US7902239B2 (en) | 2011-03-08 |
| TW200413334A (en) | 2004-08-01 |
| US7279469B2 (en) | 2007-10-09 |
| JP4783020B2 (ja) | 2011-09-28 |
| KR20060013480A (ko) | 2006-02-10 |
| MXPA05005223A (es) | 2010-09-07 |
| PL377825A1 (pl) | 2006-02-20 |
| JP2011132263A (ja) | 2011-07-07 |
| EP1562589B1 (de) | 2009-01-07 |
| SI1562589T1 (sl) | 2009-06-30 |
| RU2350606C2 (ru) | 2009-03-27 |
| EP1562589A2 (de) | 2005-08-17 |
| BR0316350A (pt) | 2005-09-27 |
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