DK1562589T3 - Diaminotriazoler der er nyttige som inhibitorer af proteinkinaser - Google Patents
Diaminotriazoler der er nyttige som inhibitorer af proteinkinaserInfo
- Publication number
- DK1562589T3 DK1562589T3 DK03789812T DK03789812T DK1562589T3 DK 1562589 T3 DK1562589 T3 DK 1562589T3 DK 03789812 T DK03789812 T DK 03789812T DK 03789812 T DK03789812 T DK 03789812T DK 1562589 T3 DK1562589 T3 DK 1562589T3
- Authority
- DK
- Denmark
- Prior art keywords
- inhibitors
- protein kinases
- diaminotriazoles
- useful
- diaminotriazoles useful
- Prior art date
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- C07D401/04—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings directly linked by a ring-member-to-ring-member bond
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PCT/US2003/036849 WO2004046120A2 (en) | 2002-11-15 | 2003-11-17 | Diaminotriazoles useful as inhibitors of protein kinases |
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US20230399331A1 (en) | 2022-06-14 | 2023-12-14 | Incyte Corporation | Solid forms of jak inhibitor and process of preparing the same |
TW202413359A (zh) | 2022-06-22 | 2024-04-01 | 美商英塞特公司 | 雙環胺cdk12抑制劑 |
US20240101557A1 (en) | 2022-07-11 | 2024-03-28 | Incyte Corporation | Fused tricyclic compounds as inhibitors of kras g12v mutants |
US20240058343A1 (en) | 2022-08-05 | 2024-02-22 | Incyte Corporation | Treatment of urticaria using jak inhibitors |
WO2024051667A1 (zh) * | 2022-09-05 | 2024-03-14 | 南京正大天晴制药有限公司 | 具有axl抑制活性的取代三唑化合物 |
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DK113716B (da) * | 1960-07-30 | 1969-04-21 | Takeda Chemical Industries Ltd | Fremgangsmåde til fremstilling af 1-[pyrimidinyl-(2)]-guanazolforbindelser eller salte deraf. |
ID23978A (id) * | 1997-11-11 | 2000-06-14 | Pfizer Prod Inc | Turunan-turunan tienopirimidin dan tienopiridin yang berguna sebagai zat-zat anti kangker |
EP1070140A1 (en) * | 1998-01-12 | 2001-01-24 | Newbiotics Inc. | Compositions and methods for treating cells having double minute dna |
WO2000010563A1 (en) * | 1998-08-20 | 2000-03-02 | Smithkline Beecham Corporation | Novel substituted triazole compounds |
US6596747B2 (en) * | 1998-10-29 | 2003-07-22 | Bristol-Myers Squibb Company | Compounds derived from an amine nucleus and pharmaceutical compositions comprising same |
CA2348234A1 (en) * | 1998-10-29 | 2000-05-11 | Chunjian Liu | Compounds derived from an amine nucleus that are inhibitors of impdh enzyme |
AU782878B2 (en) * | 2000-02-05 | 2005-09-08 | Vertex Pharmaceuticals Incorporated | Pyrazole compositions useful as inhibitors of erk |
CN100357278C (zh) * | 2000-12-22 | 2007-12-26 | 奥索-麦克尼尔药品公司 | 作为激酶抑制剂的取代的三唑二胺衍生物 |
DE10123586A1 (de) | 2001-05-08 | 2002-11-28 | Schering Ag | 3,5-Diamino-1,2,4-triazole als Kinase Inhibitoren |
TWI335913B (en) * | 2002-11-15 | 2011-01-11 | Vertex Pharma | Diaminotriazoles useful as inhibitors of protein kinases |
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2003
- 2003-11-14 TW TW092132032A patent/TWI335913B/zh not_active IP Right Cessation
- 2003-11-14 CL CL200302353A patent/CL2003002353A1/es unknown
- 2003-11-14 AR ARP030104218A patent/AR042052A1/es unknown
- 2003-11-17 KR KR1020057008795A patent/KR20060013480A/ko not_active Application Discontinuation
- 2003-11-17 SI SI200331537T patent/SI1562589T1/sl unknown
- 2003-11-17 MX MXPA05005223A patent/MXPA05005223A/es unknown
- 2003-11-17 AU AU2003294329A patent/AU2003294329B2/en not_active Ceased
- 2003-11-17 PL PL377825A patent/PL377825A1/pl not_active Application Discontinuation
- 2003-11-17 BR BR0316350-4A patent/BR0316350A/pt not_active IP Right Cessation
- 2003-11-17 DK DK03789812T patent/DK1562589T3/da active
- 2003-11-17 AT AT03789812T patent/ATE419849T1/de active
- 2003-11-17 PT PT03789812T patent/PT1562589E/pt unknown
- 2003-11-17 RU RU2005118418/04A patent/RU2350606C2/ru not_active IP Right Cessation
- 2003-11-17 US US10/715,111 patent/US7279469B2/en not_active Expired - Fee Related
- 2003-11-17 DE DE60325761T patent/DE60325761D1/de not_active Expired - Lifetime
- 2003-11-17 NZ NZ540662A patent/NZ540662A/en unknown
- 2003-11-17 JP JP2004570619A patent/JP4783020B2/ja not_active Expired - Fee Related
- 2003-11-17 EP EP03789812A patent/EP1562589B1/en not_active Expired - Lifetime
- 2003-11-17 WO PCT/US2003/036849 patent/WO2004046120A2/en active Application Filing
- 2003-11-17 ES ES03789812T patent/ES2318189T3/es not_active Expired - Lifetime
- 2003-11-17 CA CA002505789A patent/CA2505789A1/en not_active Abandoned
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2005
- 2005-06-10 NO NO20052888A patent/NO20052888L/no not_active Application Discontinuation
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2007
- 2007-07-09 US US11/774,702 patent/US7902239B2/en not_active Expired - Fee Related
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Also Published As
Publication number | Publication date |
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PT1562589E (pt) | 2009-04-15 |
EP1562589B1 (en) | 2009-01-07 |
WO2004046120A2 (en) | 2004-06-03 |
TWI335913B (en) | 2011-01-11 |
AU2003294329A1 (en) | 2004-06-15 |
BR0316350A (pt) | 2005-09-27 |
JP4783020B2 (ja) | 2011-09-28 |
NZ540662A (en) | 2008-04-30 |
NO20052888L (no) | 2005-08-12 |
US7279469B2 (en) | 2007-10-09 |
US7902239B2 (en) | 2011-03-08 |
CL2003002353A1 (es) | 2005-02-04 |
PL377825A1 (pl) | 2006-02-20 |
MXPA05005223A (es) | 2010-09-07 |
DE60325761D1 (de) | 2009-02-26 |
JP2011132263A (ja) | 2011-07-07 |
WO2004046120A3 (en) | 2004-08-12 |
AR042052A1 (es) | 2005-06-08 |
RU2350606C2 (ru) | 2009-03-27 |
CA2505789A1 (en) | 2004-06-03 |
US20080014189A1 (en) | 2008-01-17 |
AU2003294329B2 (en) | 2010-04-29 |
ATE419849T1 (de) | 2009-01-15 |
NO20052888D0 (no) | 2005-06-10 |
US20040214817A1 (en) | 2004-10-28 |
RU2005118418A (ru) | 2006-02-10 |
JP2006515313A (ja) | 2006-05-25 |
KR20060013480A (ko) | 2006-02-10 |
SI1562589T1 (sl) | 2009-06-30 |
TW200413334A (en) | 2004-08-01 |
ES2318189T3 (es) | 2009-05-01 |
EP1562589A2 (en) | 2005-08-17 |
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