CA1307003C - Phenyl carbamate - Google Patents

Phenyl carbamate

Info

Publication number
CA1307003C
CA1307003C CA000560457A CA560457A CA1307003C CA 1307003 C CA1307003 C CA 1307003C CA 000560457 A CA000560457 A CA 000560457A CA 560457 A CA560457 A CA 560457A CA 1307003 C CA1307003 C CA 1307003C
Authority
CA
Canada
Prior art keywords
compound
ethyl
free base
formula
pharmaceutically acceptable
Prior art date
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
Expired - Lifetime
Application number
CA000560457A
Other languages
English (en)
French (fr)
Inventor
Albert Enz
Current Assignee (The listed assignees may be inaccurate. Google has not performed a legal analysis and makes no representation or warranty as to the accuracy of the list.)
Novartis AG
Original Assignee
Sandoz AG
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Family has litigation
First worldwide family litigation filed litigation Critical https://patents.darts-ip.com/?family=6322236&utm_source=google_patent&utm_medium=platform_link&utm_campaign=public_patent_search&patent=CA1307003(C) "Global patent litigation dataset” by Darts-ip is licensed under a Creative Commons Attribution 4.0 International License.
Application filed by Sandoz AG filed Critical Sandoz AG
Application granted granted Critical
Publication of CA1307003C publication Critical patent/CA1307003C/en
Anticipated expiration legal-status Critical
Expired - Lifetime legal-status Critical Current

Links

Classifications

    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00—Medicinal preparations containing organic active ingredients
    • A61K31/325—Carbamic acids; Thiocarbamic acids; Anhydrides or salts thereof
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07C—ACYCLIC OR CARBOCYCLIC COMPOUNDS
    • C07C271/00—Derivatives of carbamic acids, i.e. compounds containing any of the groups, the nitrogen atom not being part of nitro or nitroso groups
    • C07C271/06—Esters of carbamic acids
    • C07C271/40—Esters of carbamic acids having oxygen atoms of carbamate groups bound to carbon atoms of six-membered aromatic rings
    • C07C271/42—Esters of carbamic acids having oxygen atoms of carbamate groups bound to carbon atoms of six-membered aromatic rings with the nitrogen atoms of the carbamate groups bound to hydrogen atoms or to acyclic carbon atoms
    • C07C271/44—Esters of carbamic acids having oxygen atoms of carbamate groups bound to carbon atoms of six-membered aromatic rings with the nitrogen atoms of the carbamate groups bound to hydrogen atoms or to acyclic carbon atoms to hydrogen atoms or to carbon atoms of unsubstituted hydrocarbon radicals
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00—Medicinal preparations containing organic active ingredients
    • A61K31/21—Esters, e.g. nitroglycerine, selenocyanates
    • A61K31/27—Esters, e.g. nitroglycerine, selenocyanates of carbamic or thiocarbamic acids, meprobamate, carbachol, neostigmine
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P17/00—Drugs for dermatological disorders
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00—Drugs for disorders of the nervous system
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00—Drugs for disorders of the nervous system
    • A61P25/02—Drugs for disorders of the nervous system for peripheral neuropathies
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00—Drugs for disorders of the nervous system
    • A61P25/24—Antidepressants
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00—Drugs for disorders of the nervous system
    • A61P25/26—Psychostimulants, e.g. nicotine, cocaine
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00—Drugs for disorders of the nervous system
    • A61P25/28—Drugs for disorders of the nervous system for treating neurodegenerative disorders of the central nervous system, e.g. nootropic agents, cognition enhancers, drugs for treating Alzheimer's disease or other forms of dementia
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P43/00—Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00

Landscapes

  • Health & Medical Sciences (AREA)
  • Chemical & Material Sciences (AREA)
  • General Health & Medical Sciences (AREA)
  • Veterinary Medicine (AREA)
  • Public Health (AREA)
  • Medicinal Chemistry (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • Organic Chemistry (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Engineering & Computer Science (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • General Chemical & Material Sciences (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Biomedical Technology (AREA)
  • Neurology (AREA)
  • Neurosurgery (AREA)
  • Epidemiology (AREA)
  • Psychiatry (AREA)
  • Emergency Medicine (AREA)
  • Dermatology (AREA)
  • Pain & Pain Management (AREA)
  • Hospice & Palliative Care (AREA)
  • Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
  • Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Medicinal Preparation (AREA)
CA000560457A 1987-03-04 1988-03-03 Phenyl carbamate Expired - Lifetime CA1307003C (en)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
DE3706914 1987-03-04
DEP3706914.4 1987-03-04

Publications (1)

Publication Number Publication Date
CA1307003C true CA1307003C (en) 1992-09-01

Family

ID=6322236

Family Applications (1)

Application Number Title Priority Date Filing Date
CA000560457A Expired - Lifetime CA1307003C (en) 1987-03-04 1988-03-03 Phenyl carbamate

Country Status (29)

Country Link
US (1) US5602176A (enExample)
JP (3) JP2625478B2 (enExample)
KR (1) KR0133686B1 (enExample)
AT (1) AT394190B (enExample)
AU (1) AU618949B2 (enExample)
BE (1) BE1001467A3 (enExample)
CA (1) CA1307003C (enExample)
CH (1) CH675720A5 (enExample)
CS (1) CS411091A3 (enExample)
CY (1) CY1735A (enExample)
DK (1) DK175762B1 (enExample)
ES (1) ES2010527A6 (enExample)
FI (1) FI89165C (enExample)
FR (1) FR2611707B1 (enExample)
GB (1) GB2203040C (enExample)
GR (1) GR1000023B (enExample)
HK (1) HK110093A (enExample)
HU (1) HU201906B (enExample)
IE (1) IE61714B1 (enExample)
IL (1) IL85609A (enExample)
IT (1) IT1219853B (enExample)
LU (2) LU87150A1 (enExample)
MY (1) MY103225A (enExample)
NL (1) NL195004C (enExample)
NZ (1) NZ223714A (enExample)
PT (1) PT86875B (enExample)
SA (1) SA93140384B1 (enExample)
SE (1) SE8800731A0 (enExample)
ZA (1) ZA881584B (enExample)

Families Citing this family (88)

* Cited by examiner, † Cited by third party
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NL195004C (nl) * 1987-03-04 2003-11-04 Novartis Ag Fenylcarbamaat bevattend farmaceutisch preparaat.
FI964113L (fi) * 1994-04-15 1996-10-14 Iyo Masaomi Lääkekoostumus hoitamaan tardiivia dyskinesiaa ja sen käyttö
AU5620998A (en) * 1996-12-18 1998-07-15 Technion Research & Development Foundation Ltd. Phenylethylamine derivatives
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CA2354035A1 (en) * 1998-12-11 2000-06-15 Bonnie Davis Use of acetylcholinesterase inhibitors on the modulation of the hypothalamic-pituitary-gonadal axis
GB9923045D0 (en) * 1999-09-29 1999-12-01 Novartis Ag New oral formulations
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WO2008037433A1 (en) 2006-09-29 2008-04-03 Synthon B.V. Process for making aminoalkylphenyl carbamates and intermediates therefor
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Family Cites Families (3)

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US4469700A (en) * 1981-06-19 1984-09-04 Lowell M. Somers Benzoylecgonine or benzoylnorecgonine as active agents for the treatment of rheumatoid arthritis
IL74497A (en) * 1985-03-05 1990-02-09 Proterra Ag Pharmaceutical compositions containing phenyl carbamate derivatives and certain phenyl carbamate derivatives
NL195004C (nl) * 1987-03-04 2003-11-04 Novartis Ag Fenylcarbamaat bevattend farmaceutisch preparaat.

Also Published As

Publication number Publication date
DK112588A (da) 1988-09-05
FI880972L (fi) 1988-09-05
ES2010527A6 (es) 1989-11-16
SA93140384B1 (ar) 2006-04-04
US5602176A (en) 1997-02-11
KR880011088A (ko) 1988-10-26
SE8800731D0 (sv) 1988-03-02
FI880972A0 (fi) 1988-03-02
HK110093A (en) 1993-10-29
LU90297I2 (fr) 1998-12-07
IE61714B1 (en) 1994-11-30
HUT49325A (en) 1989-09-28
HU201906B (en) 1991-01-28
LU87150A1 (fr) 1988-11-17
FI89165C (fi) 1993-08-25
KR0133686B1 (ko) 1998-04-21
GB2203040B (en) 1990-10-24
JP2625478B2 (ja) 1997-07-02
PT86875B (pt) 1992-05-29
JPS63238054A (ja) 1988-10-04
AU618949B2 (en) 1992-01-16
ATA55188A (de) 1991-08-15
NL195004C (nl) 2003-11-04
JPH09118617A (ja) 1997-05-06
GB2203040A (en) 1988-10-12
NL8800436A (nl) 1988-10-03
JPH09165362A (ja) 1997-06-24
NZ223714A (en) 1994-05-26
IL85609A (en) 1992-07-15
SE8800731L (sv) 1988-09-05
BE1001467A3 (fr) 1989-11-07
GR880100125A (en) 1989-01-31
GR1000023B (el) 1990-01-31
GB8804888D0 (en) 1988-03-30
IT1219853B (it) 1990-05-24
SE8800731A0 (sv) 1988-09-05
IT8847693A0 (it) 1988-03-04
FR2611707B1 (fr) 1990-04-20
IL85609A0 (en) 1988-08-31
ZA881584B (en) 1989-11-29
DK175762B1 (da) 2005-02-14
MY103225A (en) 1993-05-29
JP2859225B2 (ja) 1999-02-17
GB2203040C (en) 2014-07-30
CH675720A5 (enExample) 1990-10-31
IE880583L (en) 1988-09-04
PT86875A (pt) 1988-04-01
AU1255488A (en) 1988-09-08
AT394190B (de) 1992-02-10
FI89165B (fi) 1993-05-14
FR2611707A1 (fr) 1988-09-09
CY1735A (en) 1994-06-03
NL195004B (nl) 2003-07-01
DK112588D0 (da) 1988-03-02
CS411091A3 (en) 1992-12-16

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