BRPI0507787A - métodos, composições e instrumentos para a formação de compostos macrocìclicos - Google Patents

métodos, composições e instrumentos para a formação de compostos macrocìclicos

Info

Publication number
BRPI0507787A
BRPI0507787A BRPI0507787-7A BRPI0507787A BRPI0507787A BR PI0507787 A BRPI0507787 A BR PI0507787A BR PI0507787 A BRPI0507787 A BR PI0507787A BR PI0507787 A BRPI0507787 A BR PI0507787A
Authority
BR
Brazil
Prior art keywords
reaction medium
instruments
compositions
formation
methods
Prior art date
Application number
BRPI0507787-7A
Other languages
English (en)
Inventor
Thomas E Johnson
Billy T Fowler
Original Assignee
Thomas E Johnson
Billy T Fowler
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Thomas E Johnson, Billy T Fowler filed Critical Thomas E Johnson
Publication of BRPI0507787A publication Critical patent/BRPI0507787A/pt

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D291/00Heterocyclic compounds containing rings having nitrogen, oxygen and sulfur atoms as the only ring hetero atoms
    • C07D291/08Heterocyclic compounds containing rings having nitrogen, oxygen and sulfur atoms as the only ring hetero atoms condensed with carbocyclic rings or ring systems
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D491/00Heterocyclic compounds containing in the condensed ring system both one or more rings having oxygen atoms as the only ring hetero atoms and one or more rings having nitrogen atoms as the only ring hetero atoms, not provided for by groups C07D451/00 - C07D459/00, C07D463/00, C07D477/00 or C07D489/00
    • C07D491/02Heterocyclic compounds containing in the condensed ring system both one or more rings having oxygen atoms as the only ring hetero atoms and one or more rings having nitrogen atoms as the only ring hetero atoms, not provided for by groups C07D451/00 - C07D459/00, C07D463/00, C07D477/00 or C07D489/00 in which the condensed system contains two hetero rings
    • C07D491/08Bridged systems
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D313/00Heterocyclic compounds containing rings of more than six members having one oxygen atom as the only ring hetero atom
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D323/00Heterocyclic compounds containing more than two oxygen atoms as the only ring hetero atoms
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07FACYCLIC, CARBOCYCLIC OR HETEROCYCLIC COMPOUNDS CONTAINING ELEMENTS OTHER THAN CARBON, HYDROGEN, HALOGEN, OXYGEN, NITROGEN, SULFUR, SELENIUM OR TELLURIUM
    • C07F5/00Compounds containing elements of Groups 3 or 13 of the Periodic System
    • C07F5/02Boron compounds
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07FACYCLIC, CARBOCYCLIC OR HETEROCYCLIC COMPOUNDS CONTAINING ELEMENTS OTHER THAN CARBON, HYDROGEN, HALOGEN, OXYGEN, NITROGEN, SULFUR, SELENIUM OR TELLURIUM
    • C07F9/00Compounds containing elements of Groups 5 or 15 of the Periodic System
    • C07F9/02Phosphorus compounds
    • C07F9/547Heterocyclic compounds, e.g. containing phosphorus as a ring hetero atom

Abstract

MéTODOS,COMPOSIçõES E INSTRUMENTOS PARA A FORMAçãO DE COMPOSTOS MACROCìCLICOS Esta invenção se relaciona aos métodos, composições,e instrumento para a produção de compostos macrocíclicos. Primeiro, são fornecidos um ou mais reagentes em um meio de reação,que são capazes de formar o composto macrocíclico atavés de uma via de reação desejada que inclui pelo menos ciclização, e que são adiconalmente capazes de formção de oligómeros indesejáveis de uma via de reação indesejáda que inclui. A oligomerização de tais reações no meio de reação é modulada para reduzir a formação de olgómero indesejáveis e/ou para reduzir a separação dos olgómeros indesejáveis do meio de reação,em relação a uma reação de oligomerização não modulada correspondente maximizando, dessa forma,os rendimentos do composto macrocíclico.o compostos macrocíclico assim formado é então recuperado do meio de reação Preferivelmente, o composto macrocíclico se separa espontameamente do meio de reação por meio de separação de fases. Mais prferivelmente, o composto macrocíclico se precipita espontaneamente do meio de reação e pode, portanto, ser facilmente recuperado por filtração simpes.
BRPI0507787-7A 2004-02-17 2005-02-17 métodos, composições e instrumentos para a formação de compostos macrocìclicos BRPI0507787A (pt)

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
US54513104P 2004-02-17 2004-02-17
US11/059,796 US7709632B2 (en) 2004-02-17 2005-02-17 Methods, compositions, and apparatuses for forming macrocyclic compounds
PCT/US2005/005028 WO2006025859A2 (en) 2004-02-17 2005-02-17 Methods, compositions, and apparatuses for forming macrocyclic compounds

Publications (1)

Publication Number Publication Date
BRPI0507787A true BRPI0507787A (pt) 2007-07-17

Family

ID=36000462

Family Applications (1)

Application Number Title Priority Date Filing Date
BRPI0507787-7A BRPI0507787A (pt) 2004-02-17 2005-02-17 métodos, composições e instrumentos para a formação de compostos macrocìclicos

Country Status (15)

Country Link
US (3) US7709632B2 (pt)
EP (1) EP1716153B1 (pt)
JP (1) JP2008504225A (pt)
KR (1) KR20070009574A (pt)
CN (1) CN1946656B (pt)
AU (1) AU2005280639A1 (pt)
BR (1) BRPI0507787A (pt)
CA (1) CA2557582A1 (pt)
HK (1) HK1102694A1 (pt)
IL (2) IL177500A (pt)
MX (1) MXPA06009440A (pt)
NO (1) NO20063745L (pt)
NZ (1) NZ587400A (pt)
RU (2) RU2428422C2 (pt)
WO (1) WO2006025859A2 (pt)

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Also Published As

Publication number Publication date
CN1946656A (zh) 2007-04-11
NO20063745L (no) 2006-11-17
IL207967A0 (en) 2011-08-01
NZ587400A (en) 2012-03-30
KR20070009574A (ko) 2007-01-18
EP1716153A2 (en) 2006-11-02
IL177500A (en) 2011-05-31
RU2428422C2 (ru) 2011-09-10
HK1102694A1 (en) 2007-11-30
AU2005280639A1 (en) 2006-03-09
JP2008504225A (ja) 2008-02-14
RU2006133296A (ru) 2008-03-27
WO2006025859A2 (en) 2006-03-09
US20120157658A1 (en) 2012-06-21
MXPA06009440A (es) 2007-03-15
EP1716153B1 (en) 2013-10-09
US7709632B2 (en) 2010-05-04
IL177500A0 (en) 2006-12-10
CN1946656B (zh) 2011-08-24
WO2006025859A3 (en) 2006-11-23
CA2557582A1 (en) 2006-03-09
US8053571B2 (en) 2011-11-08
RU2010145604A (ru) 2012-05-20
EP1716153A4 (en) 2008-12-17
US20100216970A1 (en) 2010-08-26
US20070217965A1 (en) 2007-09-20

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