BR9904283A - Complexos estáveis de compostos fracamente solúveis - Google Patents

Complexos estáveis de compostos fracamente solúveis

Info

Publication number
BR9904283A
BR9904283A BR9904283-5A BR9904283A BR9904283A BR 9904283 A BR9904283 A BR 9904283A BR 9904283 A BR9904283 A BR 9904283A BR 9904283 A BR9904283 A BR 9904283A
Authority
BR
Brazil
Prior art keywords
soluble compounds
poorly soluble
complexes
ionic polymers
insoluble
Prior art date
Application number
BR9904283-5A
Other languages
English (en)
Portuguese (pt)
Inventor
Antonio A Albano
Wantanee Phuapradit
Harpreet K Sandhu
Navnit Hargovindas Shah
Original Assignee
Hoffmann La Roche
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Family has litigation
First worldwide family litigation filed litigation Critical https://patents.darts-ip.com/?family=26798138&utm_source=google_patent&utm_medium=platform_link&utm_campaign=public_patent_search&patent=BR9904283(A) "Global patent litigation dataset” by Darts-ip is licensed under a Creative Commons Attribution 4.0 International License.
Application filed by Hoffmann La Roche filed Critical Hoffmann La Roche
Publication of BR9904283A publication Critical patent/BR9904283A/pt

Links

Classifications

    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00—Medicinal preparations characterised by special physical form
    • A61K9/14—Particulate form, e.g. powders, Processes for size reducing of pure drugs or the resulting products, Pure drug nanoparticles
    • A61K9/141—Intimate drug-carrier mixtures characterised by the carrier, e.g. ordered mixtures, adsorbates, solid solutions, eutectica, co-dried, co-solubilised, co-kneaded, co-milled, co-ground products, co-precipitates, co-evaporates, co-extrudates, co-melts; Drug nanoparticles with adsorbed surface modifiers
    • A61K9/146—Intimate drug-carrier mixtures characterised by the carrier, e.g. ordered mixtures, adsorbates, solid solutions, eutectica, co-dried, co-solubilised, co-kneaded, co-milled, co-ground products, co-precipitates, co-evaporates, co-extrudates, co-melts; Drug nanoparticles with adsorbed surface modifiers with organic macromolecular compounds
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K47/00—Medicinal preparations characterised by the non-active ingredients used, e.g. carriers or inert additives; Targeting or modifying agents chemically bound to the active ingredient
    • A61K47/50—Medicinal preparations characterised by the non-active ingredients used, e.g. carriers or inert additives; Targeting or modifying agents chemically bound to the active ingredient the non-active ingredient being chemically bound to the active ingredient, e.g. polymer-drug conjugates
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K47/00—Medicinal preparations characterised by the non-active ingredients used, e.g. carriers or inert additives; Targeting or modifying agents chemically bound to the active ingredient
    • A61K47/50—Medicinal preparations characterised by the non-active ingredients used, e.g. carriers or inert additives; Targeting or modifying agents chemically bound to the active ingredient the non-active ingredient being chemically bound to the active ingredient, e.g. polymer-drug conjugates
    • A61K47/51—Medicinal preparations characterised by the non-active ingredients used, e.g. carriers or inert additives; Targeting or modifying agents chemically bound to the active ingredient the non-active ingredient being chemically bound to the active ingredient, e.g. polymer-drug conjugates the non-active ingredient being a modifying agent
    • A61K47/56—Medicinal preparations characterised by the non-active ingredients used, e.g. carriers or inert additives; Targeting or modifying agents chemically bound to the active ingredient the non-active ingredient being chemically bound to the active ingredient, e.g. polymer-drug conjugates the non-active ingredient being a modifying agent the modifying agent being an organic macromolecular compound, e.g. an oligomeric, polymeric or dendrimeric molecule
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P17/00—Drugs for dermatological disorders
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • A61P31/12—Antivirals
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P7/00—Drugs for disorders of the blood or the extracellular fluid
    • A61P7/02—Antithrombotic agents; Anticoagulants; Platelet aggregation inhibitors

Landscapes

  • Health & Medical Sciences (AREA)
  • Engineering & Computer Science (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Animal Behavior & Ethology (AREA)
  • General Health & Medical Sciences (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • Epidemiology (AREA)
  • General Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Hematology (AREA)
  • Virology (AREA)
  • Communicable Diseases (AREA)
  • Oncology (AREA)
  • Diabetes (AREA)
  • Dermatology (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Medicinal Preparation (AREA)
  • Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
  • Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
  • Nitrogen Condensed Heterocyclic Rings (AREA)
  • Plural Heterocyclic Compounds (AREA)
  • Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
BR9904283-5A 1998-09-22 1999-09-21 Complexos estáveis de compostos fracamente solúveis BR9904283A (pt)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
US10133698P 1998-09-22 1998-09-22
US13653199P 1999-05-28 1999-05-28

Publications (1)

Publication Number Publication Date
BR9904283A true BR9904283A (pt) 2000-09-26

Family

ID=26798138

Family Applications (1)

Application Number Title Priority Date Filing Date
BR9904283-5A BR9904283A (pt) 1998-09-22 1999-09-21 Complexos estáveis de compostos fracamente solúveis

Country Status (32)

Country Link
US (1) US6350786B1 (cg-RX-API-DMAC10.html)
EP (1) EP0988863B2 (cg-RX-API-DMAC10.html)
JP (5) JP2000095708A (cg-RX-API-DMAC10.html)
KR (1) KR100362019B1 (cg-RX-API-DMAC10.html)
CN (1) CN1201821C (cg-RX-API-DMAC10.html)
AR (2) AR022096A1 (cg-RX-API-DMAC10.html)
AT (1) ATE265232T1 (cg-RX-API-DMAC10.html)
AU (1) AU770745B2 (cg-RX-API-DMAC10.html)
BR (1) BR9904283A (cg-RX-API-DMAC10.html)
CA (1) CA2282906C (cg-RX-API-DMAC10.html)
CO (1) CO5140077A1 (cg-RX-API-DMAC10.html)
CZ (1) CZ300215B6 (cg-RX-API-DMAC10.html)
DE (1) DE69916733T3 (cg-RX-API-DMAC10.html)
DK (1) DK0988863T4 (cg-RX-API-DMAC10.html)
ES (1) ES2218918T5 (cg-RX-API-DMAC10.html)
HR (1) HRP990287B1 (cg-RX-API-DMAC10.html)
HU (1) HU228341B1 (cg-RX-API-DMAC10.html)
ID (1) ID24034A (cg-RX-API-DMAC10.html)
IL (1) IL131957A (cg-RX-API-DMAC10.html)
MA (1) MA26692A1 (cg-RX-API-DMAC10.html)
MY (1) MY124377A (cg-RX-API-DMAC10.html)
NO (1) NO326928B1 (cg-RX-API-DMAC10.html)
NZ (1) NZ337884A (cg-RX-API-DMAC10.html)
PE (1) PE20001049A1 (cg-RX-API-DMAC10.html)
PL (1) PL202757B1 (cg-RX-API-DMAC10.html)
PT (1) PT988863E (cg-RX-API-DMAC10.html)
RS (1) RS50193B (cg-RX-API-DMAC10.html)
RU (1) RU2240827C2 (cg-RX-API-DMAC10.html)
SG (1) SG97131A1 (cg-RX-API-DMAC10.html)
SI (1) SI0988863T2 (cg-RX-API-DMAC10.html)
TR (1) TR199902324A2 (cg-RX-API-DMAC10.html)
TW (1) TWI234465B (cg-RX-API-DMAC10.html)

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PE20001049A1 (es) 2000-10-17
RU2240827C2 (ru) 2004-11-27
JP2016196515A (ja) 2016-11-24
PT988863E (pt) 2004-07-30
JP2015187170A (ja) 2015-10-29
HRP990287B1 (en) 2004-12-31
ID24034A (id) 2000-07-06
CZ330499A3 (cs) 2000-04-12
SI0988863T2 (sl) 2009-08-31
MA26692A1 (fr) 2004-12-20
EP0988863B2 (en) 2009-03-18
NZ337884A (en) 2001-02-23
JP2013035875A (ja) 2013-02-21
CA2282906C (en) 2010-07-20
SI0988863T1 (en) 2004-08-31
CO5140077A1 (es) 2002-03-22
RS50193B (sr) 2009-05-06
DE69916733D1 (de) 2004-06-03
DE69916733T3 (de) 2009-09-24
YU47399A (cg-RX-API-DMAC10.html) 2002-08-12
IL131957A (en) 2005-06-19
TWI234465B (en) 2005-06-21
JP2007224048A (ja) 2007-09-06
DK0988863T4 (da) 2009-06-08
EP0988863A3 (en) 2000-08-09
HUP9903189A3 (en) 2009-07-28
CN1251312A (zh) 2000-04-26
HRP990287A2 (en) 2000-06-30
HUP9903189A2 (hu) 2000-06-28
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