AP558A - New erythromycin derivatives, their preparation process and their use as medicaments. - Google Patents

New erythromycin derivatives, their preparation process and their use as medicaments. Download PDF

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Publication number
AP558A
AP558A APAP/P/1995/000744A AP9500744A AP558A AP 558 A AP558 A AP 558A AP 9500744 A AP9500744 A AP 9500744A AP 558 A AP558 A AP 558A
Authority
AP
ARIPO
Prior art keywords
butanamine
methyl
dideoxy
oxy
formula
Prior art date
Application number
APAP/P/1995/000744A
Other languages
English (en)
Other versions
AP9500744A0 (en
Inventor
Constantin Agouridas
Jean-Francis Chantot (Deceased)
Alexis Denis
Solange Gouin D'ambrieres
Martret Odile Le
Original Assignee
Aventis Pharma Sa
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Aventis Pharma Sa filed Critical Aventis Pharma Sa
Publication of AP9500744A0 publication Critical patent/AP9500744A0/xx
Application granted granted Critical
Publication of AP558A publication Critical patent/AP558A/en

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Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07H—SUGARS; DERIVATIVES THEREOF; NUCLEOSIDES; NUCLEOTIDES; NUCLEIC ACIDS
    • C07H17/00—Compounds containing heterocyclic radicals directly attached to hetero atoms of saccharide radicals
    • C07H17/04—Heterocyclic radicals containing only oxygen as ring hetero atoms
    • C07H17/08—Hetero rings containing eight or more ring members, e.g. erythromycins
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P17/00—Drugs for dermatological disorders
    • A61P17/10—Anti-acne agents
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P27/00—Drugs for disorders of the senses
    • A61P27/16—Otologicals
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • A61P31/04—Antibacterial agents
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • A61P31/12—Antivirals
    • A61P31/14—Antivirals for RNA viruses
    • A61P31/16—Antivirals for RNA viruses for influenza or rhinoviruses
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P33/00—Antiparasitic agents
    • A61P33/02—Antiprotozoals, e.g. for leishmaniasis, trichomoniasis, toxoplasmosis
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07H—SUGARS; DERIVATIVES THEREOF; NUCLEOSIDES; NUCLEOTIDES; NUCLEIC ACIDS
    • C07H17/00—Compounds containing heterocyclic radicals directly attached to hetero atoms of saccharide radicals

Landscapes

  • Health & Medical Sciences (AREA)
  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • General Health & Medical Sciences (AREA)
  • Veterinary Medicine (AREA)
  • Medicinal Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • General Chemical & Material Sciences (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Animal Behavior & Ethology (AREA)
  • Engineering & Computer Science (AREA)
  • Public Health (AREA)
  • Molecular Biology (AREA)
  • Biochemistry (AREA)
  • Biotechnology (AREA)
  • Genetics & Genomics (AREA)
  • Virology (AREA)
  • Communicable Diseases (AREA)
  • Oncology (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Pulmonology (AREA)
  • Tropical Medicine & Parasitology (AREA)
  • Dermatology (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Saccharide Compounds (AREA)
  • Nitrogen Condensed Heterocyclic Rings (AREA)
  • Quinoline Compounds (AREA)
  • Plural Heterocyclic Compounds (AREA)
  • Heterocyclic Carbon Compounds Containing A Hetero Ring Having Oxygen Or Sulfur (AREA)
  • Indole Compounds (AREA)
  • Pyrrole Compounds (AREA)
  • Thiazole And Isothizaole Compounds (AREA)
  • Other In-Based Heterocyclic Compounds (AREA)
APAP/P/1995/000744A 1994-05-03 1995-05-02 New erythromycin derivatives, their preparation process and their use as medicaments. AP558A (en)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
FR9405368A FR2719587B1 (fr) 1994-05-03 1994-05-03 Nouveaux dérivés de l'érythromycine, leur procédé de préparation et leur application comme médicaments.

Publications (2)

Publication Number Publication Date
AP9500744A0 AP9500744A0 (en) 1995-07-31
AP558A true AP558A (en) 1996-11-07

Family

ID=9462785

Family Applications (1)

Application Number Title Priority Date Filing Date
APAP/P/1995/000744A AP558A (en) 1994-05-03 1995-05-02 New erythromycin derivatives, their preparation process and their use as medicaments.

Country Status (43)

Country Link
US (2) US5635485A (fi)
EP (1) EP0680967B1 (fi)
JP (4) JP2992540B2 (fi)
KR (1) KR100312267B1 (fi)
CN (2) CN1052984C (fi)
AP (1) AP558A (fi)
AT (1) ATE172203T1 (fi)
AU (1) AU684027B2 (fi)
BG (1) BG63087B1 (fi)
BR (1) BR9507700A (fi)
CA (1) CA2189271C (fi)
CZ (1) CZ293455B6 (fi)
DE (2) DE69505296T2 (fi)
DK (1) DK0680967T3 (fi)
DZ (1) DZ1878A1 (fi)
EE (1) EE03263B1 (fi)
ES (1) ES2122472T3 (fi)
FI (1) FI111263B (fi)
FR (1) FR2719587B1 (fi)
GE (1) GEP19991538B (fi)
HK (1) HK1010732A1 (fi)
HU (2) HU227493B1 (fi)
IL (1) IL113245A (fi)
LU (1) LU90872I2 (fi)
LV (1) LV11739B (fi)
MA (1) MA23534A1 (fi)
MD (1) MD1233C2 (fi)
NL (1) NL300077I1 (fi)
NO (2) NO308853B1 (fi)
NZ (1) NZ285416A (fi)
OA (1) OA10319A (fi)
PL (1) PL182034B1 (fi)
RO (1) RO113350B1 (fi)
RU (1) RU2144036C1 (fi)
SI (1) SI0680967T1 (fi)
SK (1) SK281707B6 (fi)
TJ (1) TJ313B (fi)
TN (1) TNSN95049A1 (fi)
TW (1) TW341573B (fi)
UA (1) UA51618C2 (fi)
WO (1) WO1995029929A1 (fi)
YU (1) YU49235B (fi)
ZA (1) ZA953501B (fi)

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ATE296308T1 (de) * 1996-09-04 2005-06-15 Abbott Lab 6-o-substituierte ketoliden mit antibakteriellen wirkung
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FR2757168B1 (fr) * 1996-12-12 1999-06-11 Hoechst Marion Roussel Inc Nouveaux derives de l'erythromycine, leur procede de preparation et leur application comme medicaments
FR2760017B1 (fr) * 1997-02-27 1999-04-30 Hoechst Marion Roussel Inc Nouveaux derives de l'erytromycine, leur procede de preparation et leur application comme medicaments
US5780605A (en) * 1997-09-08 1998-07-14 Abbott Laboratories 6,9-bridged erythromycin derivatives
FR2771008B1 (fr) * 1997-11-17 2000-04-28 Hoechst Marion Roussel Inc Utilisation des ketolides pour la preparation de compositions pharmaceutiques destinees a prevenir les complications thrombotiques arterielles liees a l'atherosclerose
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Citations (2)

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Publication number Priority date Publication date Assignee Title
EP0487411A1 (fr) * 1990-11-21 1992-05-27 Roussel Uclaf Nouveaux dérivés de l'érythromycine, leur procédé de préparation, les nouveaux intermédiaires obtenus et leur application comme médicaments
FR2692579A1 (fr) * 1992-06-19 1993-12-24 Roussel Uclaf Nouveaux dérivés de la picromycine, leur procédé de préparation et leur application comme médicaments.

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FR2692579A1 (fr) * 1992-06-19 1993-12-24 Roussel Uclaf Nouveaux dérivés de la picromycine, leur procédé de préparation et leur application comme médicaments.

Also Published As

Publication number Publication date
BG63087B1 (bg) 2001-03-30
JP2007269810A (ja) 2007-10-18
LV11739A (lv) 1997-04-20
NO308853B1 (no) 2000-11-06
FI111263B (fi) 2003-06-30
JP2007045847A (ja) 2007-02-22
NO964654D0 (no) 1996-11-04
ATE172203T1 (de) 1998-10-15
WO1995029929A1 (fr) 1995-11-09
SK281707B6 (sk) 2001-07-10
JPH11152296A (ja) 1999-06-08
TJ313B (en) 2001-08-06
EP0680967B1 (fr) 1998-10-14
CN1088709C (zh) 2002-08-07
FI964395A (fi) 1996-10-31
KR100312267B1 (ko) 2002-06-22
YU27095A (sh) 1998-05-15
OA10319A (fr) 1997-10-07
CN1151746A (zh) 1997-06-11
PL182034B1 (pl) 2001-10-31
EE03263B1 (et) 2000-04-17
SI0680967T1 (en) 1999-02-28
AU2449995A (en) 1995-11-29
DE69505296D1 (de) 1998-11-19
NO2001027I1 (no) 2002-01-28
BR9507700A (pt) 1997-08-19
MD1233B1 (en) 1999-05-31
LV11739B (en) 1997-08-20
MA23534A1 (fr) 1995-12-31
HU219599B (hu) 2001-05-28
HK1010732A1 (en) 1999-06-25
TNSN95049A1 (fr) 1996-02-06
HU9904687D0 (en) 2000-03-28
MX9605208A (es) 1997-09-30
JP4658902B2 (ja) 2011-03-23
DK0680967T3 (da) 1999-06-23
CN1052984C (zh) 2000-05-31
DE10299001I1 (de) 2012-07-05
SK140296A3 (en) 1998-04-08
JP2992540B2 (ja) 1999-12-20
FI964395A0 (fi) 1996-10-31
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JP4750755B2 (ja) 2011-08-17
DE10299001I2 (de) 2012-07-05
BG100951A (en) 1997-08-29
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FR2719587A1 (fr) 1995-11-10
IL113245A (en) 1999-11-30
US5635485A (en) 1997-06-03
HU227493B1 (en) 2011-07-28
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RU2144036C1 (ru) 2000-01-10
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HUT75698A (en) 1997-05-28
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JP3998828B2 (ja) 2007-10-31
UA51618C2 (uk) 2002-12-16
JPH0853489A (ja) 1996-02-27
US6100404A (en) 2000-08-08
IL113245A0 (en) 1995-07-31
FR2719587B1 (fr) 1996-07-12
CN1229082A (zh) 1999-09-22
DZ1878A1 (fr) 2002-02-17
ZA953501B (en) 1996-05-02
GEP19991538B (en) 1999-03-05
DE69505296T2 (de) 1999-04-22
TW341573B (en) 1998-10-01
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CZ293455B6 (cs) 2004-05-12
CA2189271C (fr) 2005-12-27
YU49235B (sh) 2004-12-31
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NL300077I1 (nl) 2002-03-01

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