ZA200708179B - Dipeptidyl peptidase-IV inhibitors - Google Patents

Dipeptidyl peptidase-IV inhibitors

Info

Publication number
ZA200708179B
ZA200708179B ZA200708179A ZA200708179A ZA200708179B ZA 200708179 B ZA200708179 B ZA 200708179B ZA 200708179 A ZA200708179 A ZA 200708179A ZA 200708179 A ZA200708179 A ZA 200708179A ZA 200708179 B ZA200708179 B ZA 200708179B
Authority
ZA
South Africa
Prior art keywords
inhibitors
dipeptidyl peptidase
dipeptidyl
peptidase
Prior art date
Application number
ZA200708179A
Other languages
English (en)
Inventor
Heiko Kroth
Tim Feuerstein
Frank Richter
Juergen Boer
Michael Essers
Bert Nolte
Matthias Schneider
Matthias Hochguertel
Fritz-Frieder Frickel
Arthur Taveras
Christoph Steeneck
Original Assignee
Alantos Pharmaceuticals Holding Inc
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Family has litigation
First worldwide family litigation filed litigation Critical https://patents.darts-ip.com/?family=36694223&utm_source=google_patent&utm_medium=platform_link&utm_campaign=public_patent_search&patent=ZA200708179(B) "Global patent litigation dataset” by Darts-ip is licensed under a Creative Commons Attribution 4.0 International License.
Application filed by Alantos Pharmaceuticals Holding Inc filed Critical Alantos Pharmaceuticals Holding Inc
Publication of ZA200708179B publication Critical patent/ZA200708179B/xx

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    • C07D207/02—Heterocyclic compounds containing five-membered rings not condensed with other rings, with one nitrogen atom as the only ring hetero atom with only hydrogen or carbon atoms directly attached to the ring nitrogen atom
    • C07D207/04—Heterocyclic compounds containing five-membered rings not condensed with other rings, with one nitrogen atom as the only ring hetero atom with only hydrogen or carbon atoms directly attached to the ring nitrogen atom having no double bonds between ring members or between ring members and non-ring members
    • C07D207/10—Heterocyclic compounds containing five-membered rings not condensed with other rings, with one nitrogen atom as the only ring hetero atom with only hydrogen or carbon atoms directly attached to the ring nitrogen atom having no double bonds between ring members or between ring members and non-ring members with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
    • C07D207/16—Carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals
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    • A61K31/41—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having five-membered rings with two or more ring hetero atoms, at least one of which being nitrogen, e.g. tetrazole
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ZA200708179A 2005-04-22 2006-04-21 Dipeptidyl peptidase-IV inhibitors ZA200708179B (en)

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US67415105P 2005-04-22 2005-04-22

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ZA200708179B true ZA200708179B (en) 2009-12-30

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US (3) US7553861B2 (enExample)
EP (1) EP1888562B1 (enExample)
JP (2) JP4568361B2 (enExample)
KR (1) KR20080000665A (enExample)
CN (1) CN101277949A (enExample)
AP (1) AP2007004234A0 (enExample)
AU (2) AU2006239929B2 (enExample)
BR (1) BRPI0608469A2 (enExample)
CA (1) CA2599419A1 (enExample)
CR (1) CR9462A (enExample)
EA (1) EA200702208A1 (enExample)
ES (1) ES2477868T3 (enExample)
IL (1) IL186607A0 (enExample)
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NO (1) NO20075973L (enExample)
TN (1) TNSN07244A1 (enExample)
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ZA (1) ZA200708179B (enExample)

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DE102004054054A1 (de) 2004-11-05 2006-05-11 Boehringer Ingelheim Pharma Gmbh & Co. Kg Verfahren zur Herstellung chiraler 8-(3-Amino-piperidin-1-yl)-xanthine
MX2007011453A (es) * 2005-04-22 2008-02-12 Alantos Pharmaceuticals Holding Inc Inhibidores de la dipeptidil peptidasa-iv.
EP1942921A4 (en) * 2005-10-25 2011-03-09 Merck Sharp & Dohme COMBINATION OF A DIPEPTIDYL-PEPTIDASE-4 HEMMER AND AN ANTIHYPERTENSIVE AGENT FOR THE TREATMENT OF DIABETES AND HYPERTONIA
WO2007078726A2 (en) * 2005-12-16 2007-07-12 Merck & Co., Inc. Pharmaceutical compositions of combinations of dipeptidyl peptidase-4 inhibitors with metformin
EP1852108A1 (en) 2006-05-04 2007-11-07 Boehringer Ingelheim Pharma GmbH & Co.KG DPP IV inhibitor formulations
PE20080251A1 (es) 2006-05-04 2008-04-25 Boehringer Ingelheim Int Usos de inhibidores de dpp iv
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AU2006239929B2 (en) 2011-11-03
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WO2006116157A3 (en) 2007-04-19
CR9462A (es) 2008-04-16
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MX2007011453A (es) 2008-02-12
US8076330B2 (en) 2011-12-13
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