AP2007004234A0 - Dipeptidyl peptidase-IV inhibitors - Google Patents

Dipeptidyl peptidase-IV inhibitors

Info

Publication number
AP2007004234A0
AP2007004234A0 AP2007004234A AP2007004234A AP2007004234A0 AP 2007004234 A0 AP2007004234 A0 AP 2007004234A0 AP 2007004234 A AP2007004234 A AP 2007004234A AP 2007004234 A AP2007004234 A AP 2007004234A AP 2007004234 A0 AP2007004234 A0 AP 2007004234A0
Authority
AP
ARIPO
Prior art keywords
inhibitors
dipeptidyl peptidase
dipeptidyl
peptidase
Prior art date
Application number
AP2007004234A
Other languages
English (en)
Inventor
Heiko Kroth
Tim Feuerstein
Frank Richter
Original Assignee
Alantos Pharm Holding
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Family has litigation
First worldwide family litigation filed litigation Critical https://patents.darts-ip.com/?family=36694223&utm_source=google_patent&utm_medium=platform_link&utm_campaign=public_patent_search&patent=AP2007004234(A0) "Global patent litigation dataset” by Darts-ip is licensed under a Creative Commons Attribution 4.0 International License.
Application filed by Alantos Pharm Holding filed Critical Alantos Pharm Holding
Publication of AP2007004234A0 publication Critical patent/AP2007004234A0/xx

Links

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    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
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    • C07D207/02—Heterocyclic compounds containing five-membered rings not condensed with other rings, with one nitrogen atom as the only ring hetero atom with only hydrogen or carbon atoms directly attached to the ring nitrogen atom
    • C07D207/04—Heterocyclic compounds containing five-membered rings not condensed with other rings, with one nitrogen atom as the only ring hetero atom with only hydrogen or carbon atoms directly attached to the ring nitrogen atom having no double bonds between ring members or between ring members and non-ring members
    • C07D207/10—Heterocyclic compounds containing five-membered rings not condensed with other rings, with one nitrogen atom as the only ring hetero atom with only hydrogen or carbon atoms directly attached to the ring nitrogen atom having no double bonds between ring members or between ring members and non-ring members with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
    • C07D207/16—Carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals
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    • A61K31/33—Heterocyclic compounds
    • A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/41—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having five-membered rings with two or more ring hetero atoms, at least one of which being nitrogen, e.g. tetrazole
    • A61K31/415—1,2-Diazoles
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    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D209/00—Heterocyclic compounds containing five-membered rings, condensed with other rings, with one nitrogen atom as the only ring hetero atom
    • C07D209/02—Heterocyclic compounds containing five-membered rings, condensed with other rings, with one nitrogen atom as the only ring hetero atom condensed with one carbocyclic ring
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    • C07D209/00—Heterocyclic compounds containing five-membered rings, condensed with other rings, with one nitrogen atom as the only ring hetero atom
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    • C07D401/00—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom
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    • C07D401/12—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings linked by a chain containing hetero atoms as chain links
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    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D403/00—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, not provided for by group C07D401/00
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    • C07D403/12—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, not provided for by group C07D401/00 containing two hetero rings linked by a chain containing hetero atoms as chain links
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    • C07D413/02—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms containing two hetero rings
    • C07D413/12—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms containing two hetero rings linked by a chain containing hetero atoms as chain links
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    • C07D487/02—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00 in which the condensed system contains two hetero rings
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    • C07D495/02—Heterocyclic compounds containing in the condensed system at least one hetero ring having sulfur atoms as the only ring hetero atoms in which the condensed system contains two hetero rings
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  • Neurology (AREA)
  • Biomedical Technology (AREA)
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  • Addiction (AREA)
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  • Endocrinology (AREA)
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  • Physical Education & Sports Medicine (AREA)
  • Urology & Nephrology (AREA)
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AP2007004234A 2005-04-22 2006-04-21 Dipeptidyl peptidase-IV inhibitors AP2007004234A0 (en)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
US67415105P 2005-04-22 2005-04-22
PCT/US2006/015200 WO2006116157A2 (en) 2005-04-22 2006-04-21 Dipeptidyl peptidase-iv inhibitors

Publications (1)

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AP2007004234A0 true AP2007004234A0 (en) 2007-12-31

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AP2007004234A AP2007004234A0 (en) 2005-04-22 2006-04-21 Dipeptidyl peptidase-IV inhibitors

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US (3) US7553861B2 (enExample)
EP (1) EP1888562B1 (enExample)
JP (2) JP4568361B2 (enExample)
KR (1) KR20080000665A (enExample)
CN (1) CN101277949A (enExample)
AP (1) AP2007004234A0 (enExample)
AU (2) AU2006239929B2 (enExample)
BR (1) BRPI0608469A2 (enExample)
CA (1) CA2599419A1 (enExample)
CR (1) CR9462A (enExample)
EA (1) EA200702208A1 (enExample)
ES (1) ES2477868T3 (enExample)
IL (1) IL186607A0 (enExample)
MA (1) MA29387B1 (enExample)
MX (1) MX2007011453A (enExample)
NO (1) NO20075973L (enExample)
TN (1) TNSN07244A1 (enExample)
WO (1) WO2006116157A2 (enExample)
ZA (1) ZA200708179B (enExample)

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US7407955B2 (en) 2002-08-21 2008-08-05 Boehringer Ingelheim Pharma Gmbh & Co., Kg 8-[3-amino-piperidin-1-yl]-xanthines, the preparation thereof and their use as pharmaceutical compositions
DE102004054054A1 (de) 2004-11-05 2006-05-11 Boehringer Ingelheim Pharma Gmbh & Co. Kg Verfahren zur Herstellung chiraler 8-(3-Amino-piperidin-1-yl)-xanthine
KR20080000665A (ko) * 2005-04-22 2008-01-02 알란토스 파마슈티컬즈 홀딩, 인코포레이티드 디펩티딜 펩티다아제-ⅳ 억제제
WO2007050485A2 (en) * 2005-10-25 2007-05-03 Merck & Co., Inc. Combination of a dipeptidyl peptidase-4 inhibitor and an anti-hypertensive agent for the treatment of diabetes and hypertension
US8414921B2 (en) * 2005-12-16 2013-04-09 Merck Sharp & Dohme Corp. Pharmaceutical compositions of combinations of dipeptidyl peptidase-4 inhibitors with metformin
PE20080251A1 (es) 2006-05-04 2008-04-25 Boehringer Ingelheim Int Usos de inhibidores de dpp iv
BRPI0711558A2 (pt) 2006-05-04 2011-11-08 Boeringer Ingelheim Internat Gmbh polimorfos
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CA2599419A1 (en) 2006-11-02
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JP2010150273A (ja) 2010-07-08
BRPI0608469A2 (pt) 2010-01-05
AU2006239929A1 (en) 2006-11-02
ZA200708179B (en) 2009-12-30
US20060270701A1 (en) 2006-11-30
TNSN07244A1 (en) 2008-11-21
AU2010201511A1 (en) 2010-05-06
AU2006239929B2 (en) 2011-11-03
EP1888562B1 (en) 2014-06-18
MA29387B1 (fr) 2008-04-01
JP4568361B2 (ja) 2010-10-27
JP5198494B2 (ja) 2013-05-15
WO2006116157A2 (en) 2006-11-02
WO2006116157A9 (en) 2007-03-01
EA200702208A1 (ru) 2008-04-28
CR9462A (es) 2008-04-16
WO2006116157A3 (en) 2007-04-19
US7553861B2 (en) 2009-06-30
KR20080000665A (ko) 2008-01-02
MX2007011453A (es) 2008-02-12
US8076330B2 (en) 2011-12-13

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