EA200001247A1 - N-связанные сульфонамиды n-гетероциклических карбоновых кислот или изостеры карбоновых кислот - Google Patents

N-связанные сульфонамиды n-гетероциклических карбоновых кислот или изостеры карбоновых кислот

Info

Publication number
EA200001247A1
EA200001247A1 EA200001247A EA200001247A EA200001247A1 EA 200001247 A1 EA200001247 A1 EA 200001247A1 EA 200001247 A EA200001247 A EA 200001247A EA 200001247 A EA200001247 A EA 200001247A EA 200001247 A1 EA200001247 A1 EA 200001247A1
Authority
EA
Eurasian Patent Office
Prior art keywords
carbonic acids
heterocyclic
isateres
sulphonamides
bonded
Prior art date
Application number
EA200001247A
Other languages
English (en)
Inventor
Грегори С. Гамильтон
Марк Х. Норман
Йонг-Квиан Ву
Original Assignee
Джи Пи Ай Нил Холдингс, Инк.
Эмджен, Инк.
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Джи Пи Ай Нил Холдингс, Инк., Эмджен, Инк. filed Critical Джи Пи Ай Нил Холдингс, Инк.
Publication of EA200001247A1 publication Critical patent/EA200001247A1/ru

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D207/00—Heterocyclic compounds containing five-membered rings not condensed with other rings, with one nitrogen atom as the only ring hetero atom
    • C07D207/02—Heterocyclic compounds containing five-membered rings not condensed with other rings, with one nitrogen atom as the only ring hetero atom with only hydrogen or carbon atoms directly attached to the ring nitrogen atom
    • C07D207/04—Heterocyclic compounds containing five-membered rings not condensed with other rings, with one nitrogen atom as the only ring hetero atom with only hydrogen or carbon atoms directly attached to the ring nitrogen atom having no double bonds between ring members or between ring members and non-ring members
    • C07D207/08—Heterocyclic compounds containing five-membered rings not condensed with other rings, with one nitrogen atom as the only ring hetero atom with only hydrogen or carbon atoms directly attached to the ring nitrogen atom having no double bonds between ring members or between ring members and non-ring members with hydrocarbon radicals, substituted by hetero atoms, attached to ring carbon atoms
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K8/00—Cosmetics or similar toiletry preparations
    • A61K8/18—Cosmetics or similar toiletry preparations characterised by the composition
    • A61K8/30—Cosmetics or similar toiletry preparations characterised by the composition containing organic compounds
    • A61K8/49—Cosmetics or similar toiletry preparations characterised by the composition containing organic compounds containing heterocyclic compounds
    • A61K8/4906—Cosmetics or similar toiletry preparations characterised by the composition containing organic compounds containing heterocyclic compounds with one nitrogen as the only hetero atom
    • A61K8/4913—Cosmetics or similar toiletry preparations characterised by the composition containing organic compounds containing heterocyclic compounds with one nitrogen as the only hetero atom having five membered rings, e.g. pyrrolidone carboxylic acid
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P17/00—Drugs for dermatological disorders
    • A61P17/14—Drugs for dermatological disorders for baldness or alopecia
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61Q—SPECIFIC USE OF COSMETICS OR SIMILAR TOILETRY PREPARATIONS
    • A61Q7/00—Preparations for affecting hair growth
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D207/00—Heterocyclic compounds containing five-membered rings not condensed with other rings, with one nitrogen atom as the only ring hetero atom
    • C07D207/02—Heterocyclic compounds containing five-membered rings not condensed with other rings, with one nitrogen atom as the only ring hetero atom with only hydrogen or carbon atoms directly attached to the ring nitrogen atom
    • C07D207/04—Heterocyclic compounds containing five-membered rings not condensed with other rings, with one nitrogen atom as the only ring hetero atom with only hydrogen or carbon atoms directly attached to the ring nitrogen atom having no double bonds between ring members or between ring members and non-ring members
    • C07D207/10—Heterocyclic compounds containing five-membered rings not condensed with other rings, with one nitrogen atom as the only ring hetero atom with only hydrogen or carbon atoms directly attached to the ring nitrogen atom having no double bonds between ring members or between ring members and non-ring members with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
    • C07D207/16—Carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D403/00—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, not provided for by group C07D401/00
    • C07D403/02—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, not provided for by group C07D401/00 containing two hetero rings
    • C07D403/04—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, not provided for by group C07D401/00 containing two hetero rings directly linked by a ring-member-to-ring-member bond

Abstract

Это изобретение относится к новым N-связанным сульфонамидам N-гетероциклических карбоновых кислот и изостерам карбоновых кислот, их получению и использованию для лечения неврологических нарушений, в том числе физически поврежденных нервов, и нейродегенеративных заболеваний и для лечения алопеции и активации роста волос.Международная заявка была опубликована вместе с отчетом о международном поиске.
EA200001247A 1998-06-03 1998-12-03 N-связанные сульфонамиды n-гетероциклических карбоновых кислот или изостеры карбоновых кислот EA200001247A1 (ru)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
US8784298P 1998-06-03 1998-06-03
PCT/US1998/025572 WO1999062880A1 (en) 1998-06-03 1998-12-03 N-linked sulfonamides of n-heterocyclic carboxylic acids or carboxylic acid isosteres

Publications (1)

Publication Number Publication Date
EA200001247A1 true EA200001247A1 (ru) 2001-08-27

Family

ID=22207576

Family Applications (1)

Application Number Title Priority Date Filing Date
EA200001247A EA200001247A1 (ru) 1998-06-03 1998-12-03 N-связанные сульфонамиды n-гетероциклических карбоновых кислот или изостеры карбоновых кислот

Country Status (17)

Country Link
US (3) US7459473B2 (ru)
EP (1) EP1084106A1 (ru)
JP (1) JP2002516904A (ru)
KR (1) KR20010052503A (ru)
CN (1) CN1295561A (ru)
AU (1) AU1708099A (ru)
BG (1) BG105012A (ru)
BR (1) BR9815882A (ru)
CA (1) CA2334002A1 (ru)
EA (1) EA200001247A1 (ru)
HU (1) HUP0102935A3 (ru)
IL (1) IL140040A0 (ru)
NO (1) NO20006078L (ru)
PL (1) PL348661A1 (ru)
SK (1) SK18302000A3 (ru)
WO (1) WO1999062880A1 (ru)
ZA (1) ZA9811060B (ru)

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US9776976B2 (en) 2013-09-06 2017-10-03 Inception 2, Inc. Triazolone compounds and uses thereof
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US20020052514A1 (en) 2002-05-02
BG105012A (en) 2001-08-31
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HUP0102935A2 (en) 2001-12-28
US20040082622A1 (en) 2004-04-29
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HUP0102935A3 (en) 2002-01-28
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