IL140040A0 - N-linked sulfonamides of n-heterocyclic carboxylic acids or carboxylic acid isosteres - Google Patents

N-linked sulfonamides of n-heterocyclic carboxylic acids or carboxylic acid isosteres

Info

Publication number
IL140040A0
IL140040A0 IL14004098A IL14004098A IL140040A0 IL 140040 A0 IL140040 A0 IL 140040A0 IL 14004098 A IL14004098 A IL 14004098A IL 14004098 A IL14004098 A IL 14004098A IL 140040 A0 IL140040 A0 IL 140040A0
Authority
IL
Israel
Prior art keywords
carboxylic acid
acid isosteres
heterocyclic
carboxylic acids
linked sulfonamides
Prior art date
Application number
IL14004098A
Other languages
English (en)
Original Assignee
Guilford Pharm Inc
Amgen Inc
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Guilford Pharm Inc, Amgen Inc filed Critical Guilford Pharm Inc
Publication of IL140040A0 publication Critical patent/IL140040A0/xx

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D207/00—Heterocyclic compounds containing five-membered rings not condensed with other rings, with one nitrogen atom as the only ring hetero atom
    • C07D207/02—Heterocyclic compounds containing five-membered rings not condensed with other rings, with one nitrogen atom as the only ring hetero atom with only hydrogen or carbon atoms directly attached to the ring nitrogen atom
    • C07D207/04—Heterocyclic compounds containing five-membered rings not condensed with other rings, with one nitrogen atom as the only ring hetero atom with only hydrogen or carbon atoms directly attached to the ring nitrogen atom having no double bonds between ring members or between ring members and non-ring members
    • C07D207/08—Heterocyclic compounds containing five-membered rings not condensed with other rings, with one nitrogen atom as the only ring hetero atom with only hydrogen or carbon atoms directly attached to the ring nitrogen atom having no double bonds between ring members or between ring members and non-ring members with hydrocarbon radicals, substituted by hetero atoms, attached to ring carbon atoms
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K8/00—Cosmetics or similar toiletry preparations
    • A61K8/18—Cosmetics or similar toiletry preparations characterised by the composition
    • A61K8/30—Cosmetics or similar toiletry preparations characterised by the composition containing organic compounds
    • A61K8/49—Cosmetics or similar toiletry preparations characterised by the composition containing organic compounds containing heterocyclic compounds
    • A61K8/4906—Cosmetics or similar toiletry preparations characterised by the composition containing organic compounds containing heterocyclic compounds with one nitrogen as the only hetero atom
    • A61K8/4913—Cosmetics or similar toiletry preparations characterised by the composition containing organic compounds containing heterocyclic compounds with one nitrogen as the only hetero atom having five membered rings, e.g. pyrrolidone carboxylic acid
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P17/00—Drugs for dermatological disorders
    • A61P17/14—Drugs for dermatological disorders for baldness or alopecia
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61Q—SPECIFIC USE OF COSMETICS OR SIMILAR TOILETRY PREPARATIONS
    • A61Q7/00—Preparations for affecting hair growth
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D207/00—Heterocyclic compounds containing five-membered rings not condensed with other rings, with one nitrogen atom as the only ring hetero atom
    • C07D207/02—Heterocyclic compounds containing five-membered rings not condensed with other rings, with one nitrogen atom as the only ring hetero atom with only hydrogen or carbon atoms directly attached to the ring nitrogen atom
    • C07D207/04—Heterocyclic compounds containing five-membered rings not condensed with other rings, with one nitrogen atom as the only ring hetero atom with only hydrogen or carbon atoms directly attached to the ring nitrogen atom having no double bonds between ring members or between ring members and non-ring members
    • C07D207/10—Heterocyclic compounds containing five-membered rings not condensed with other rings, with one nitrogen atom as the only ring hetero atom with only hydrogen or carbon atoms directly attached to the ring nitrogen atom having no double bonds between ring members or between ring members and non-ring members with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
    • C07D207/16—Carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D403/00—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, not provided for by group C07D401/00
    • C07D403/02—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, not provided for by group C07D401/00 containing two hetero rings
    • C07D403/04—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, not provided for by group C07D401/00 containing two hetero rings directly linked by a ring-member-to-ring-member bond
IL14004098A 1998-06-03 1998-12-03 N-linked sulfonamides of n-heterocyclic carboxylic acids or carboxylic acid isosteres IL140040A0 (en)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
US8784298P 1998-06-03 1998-06-03
PCT/US1998/025572 WO1999062880A1 (en) 1998-06-03 1998-12-03 N-linked sulfonamides of n-heterocyclic carboxylic acids or carboxylic acid isosteres

Publications (1)

Publication Number Publication Date
IL140040A0 true IL140040A0 (en) 2002-02-10

Family

ID=22207576

Family Applications (1)

Application Number Title Priority Date Filing Date
IL14004098A IL140040A0 (en) 1998-06-03 1998-12-03 N-linked sulfonamides of n-heterocyclic carboxylic acids or carboxylic acid isosteres

Country Status (17)

Country Link
US (3) US7459473B2 (ru)
EP (1) EP1084106A1 (ru)
JP (1) JP2002516904A (ru)
KR (1) KR20010052503A (ru)
CN (1) CN1295561A (ru)
AU (1) AU1708099A (ru)
BG (1) BG105012A (ru)
BR (1) BR9815882A (ru)
CA (1) CA2334002A1 (ru)
EA (1) EA200001247A1 (ru)
HU (1) HUP0102935A3 (ru)
IL (1) IL140040A0 (ru)
NO (1) NO20006078L (ru)
PL (1) PL348661A1 (ru)
SK (1) SK18302000A3 (ru)
WO (1) WO1999062880A1 (ru)
ZA (1) ZA9811060B (ru)

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SE0202539D0 (sv) 2002-08-27 2002-08-27 Astrazeneca Ab Compounds
SE0401762D0 (sv) 2004-07-05 2004-07-05 Astrazeneca Ab Novel compounds
US7648992B2 (en) 2004-07-05 2010-01-19 Astrazeneca Ab Hydantoin derivatives for the treatment of obstructive airway diseases
SE0401763D0 (sv) * 2004-07-05 2004-07-05 Astrazeneca Ab Compounds
SE0403086D0 (sv) 2004-12-17 2004-12-17 Astrazeneca Ab Compounds
SE0403085D0 (sv) 2004-12-17 2004-12-17 Astrazeneca Ab Novel componds
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EA027986B9 (ru) 2012-12-20 2018-01-31 Инсепшн 2, Инк. Соединения триазолона и их применение
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Also Published As

Publication number Publication date
HUP0102935A2 (en) 2001-12-28
CA2334002A1 (en) 1999-12-09
US20040082622A1 (en) 2004-04-29
SK18302000A3 (sk) 2001-06-11
NO20006078L (no) 2001-02-05
US7078424B2 (en) 2006-07-18
US20020052514A1 (en) 2002-05-02
WO1999062880A1 (en) 1999-12-09
KR20010052503A (ko) 2001-06-25
AU1708099A (en) 1999-12-20
NO20006078D0 (no) 2000-11-30
HUP0102935A3 (en) 2002-01-28
BR9815882A (pt) 2002-09-17
US7459473B2 (en) 2008-12-02
EA200001247A1 (ru) 2001-08-27
ZA9811060B (en) 1999-12-03
CN1295561A (zh) 2001-05-16
EP1084106A1 (en) 2001-03-21
US20020052510A1 (en) 2002-05-02
PL348661A1 (en) 2002-06-03
JP2002516904A (ja) 2002-06-11
BG105012A (en) 2001-08-31

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