ZA200407339B - Combination treatments for chemokine-mediated diseases. - Google Patents

Combination treatments for chemokine-mediated diseases. Download PDF

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Publication number
ZA200407339B
ZA200407339B ZA200407339A ZA200407339A ZA200407339B ZA 200407339 B ZA200407339 B ZA 200407339B ZA 200407339 A ZA200407339 A ZA 200407339A ZA 200407339 A ZA200407339 A ZA 200407339A ZA 200407339 B ZA200407339 B ZA 200407339B
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South Africa
Prior art keywords
group
compound
substituted
ohh
solvate
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ZA200407339A
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English (en)
Inventor
Arthur G Taveras
Daniel Lundell
James Jakway
Loretta A Bober
Purakkattle Biju
Matasim Billah
William Kreutner
Jay S Fine
Jianhua Chao
Younong Yu
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Schering Corp
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Publication of ZA200407339B publication Critical patent/ZA200407339B/en

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ZA200407339A 2002-03-18 2004-09-13 Combination treatments for chemokine-mediated diseases. ZA200407339B (en)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
US36531402P 2002-03-18 2002-03-18

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ZA200407339B true ZA200407339B (en) 2005-10-06

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ZA200407339A ZA200407339B (en) 2002-03-18 2004-09-13 Combination treatments for chemokine-mediated diseases.

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US (2) US20040053953A1 (enExample)
EP (1) EP1485089B1 (enExample)
JP (1) JP4733350B2 (enExample)
CN (1) CN100444839C (enExample)
AR (1) AR040400A1 (enExample)
AU (1) AU2003220384B2 (enExample)
BR (1) BR0308739A (enExample)
CA (1) CA2479126C (enExample)
MX (1) MXPA04009127A (enExample)
NO (1) NO20044402L (enExample)
NZ (1) NZ535314A (enExample)
TW (2) TW200808314A (enExample)
WO (1) WO2003080053A1 (enExample)
ZA (1) ZA200407339B (enExample)

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US7718678B2 (en) 2005-06-29 2010-05-18 Schering Corporation Di-substituted oxadiazoles as CXC-chemokine receptor ligands
DE602006017849D1 (de) 2005-06-29 2010-12-09 Schering Corp 5,6-disubstituierte oxadiazolopyrazine und thiadiazolopyrazine als liganden des cxc-chemokinrezeptors
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JP2009539990A (ja) 2006-06-12 2009-11-19 シェーリング コーポレイション Ｃｘｃｒ２またはｃｘｃｒ１とｃｘｃｒ２との両方のいずれかの選択的アンタゴニストの薬学的処方物および組成物ならびに炎症性障害を治療するためにそれらを使用する方法
TW200813033A (en) * 2006-07-07 2008-03-16 Schering Corp 3, 4-di-substituted cyclobutene-1, 2-diones as CXC-chemokine receptor ligands
US8450348B2 (en) * 2007-02-21 2013-05-28 Forma Tm, Llc Derivatives of squaric acid with anti-proliferative activity
BRPI0812222A2 (pt) 2007-06-06 2014-12-16 Novartis Ag Compostos ciclobutenodiona substituídos anti-inflamatórios.
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UA103198C2 (en) 2008-08-04 2013-09-25 Новартис Аг Squaramide derivatives as cxcr2 antagonists
WO2010131146A1 (en) * 2009-05-12 2010-11-18 Pfizer Limited Cyclobutenedione derivatives
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TWI724056B (zh) 2015-11-19 2021-04-11 美商卡默森屈有限公司 Ｃｘｃｒ２抑制劑
TWI734715B (zh) 2015-11-19 2021-08-01 美商卡默森屈有限公司 趨化因子受體調節劑
RU2020106383A (ru) 2017-08-14 2021-09-16 Аллерган, Инк. 3,4-двузамещенные 3-циклобутен-1,2-дионы и их применение
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IL275839B2 (en) 2018-01-08 2024-02-01 Chemocentryx Inc Methods for the treatment of generalized abscess psoriasis using a CCR6 or CXCR2 antagonist
UA128700C2 (uk) 2018-09-21 2024-10-02 Пфайзер Інк. N-заміщені діоксоциклобутеніламіно-3-гідроксипіколінаміди, прийнятні як інгібітори ccr6
CN112851635B (zh) * 2019-11-28 2022-09-16 中国医学科学院药物研究所 环状砜类化合物及其制备方法、用途和药物组合物
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US7960433B2 (en) 2011-06-14
US20070155756A1 (en) 2007-07-05
BR0308739A (pt) 2005-01-11
MXPA04009127A (es) 2005-01-25
EP1485089B1 (en) 2013-04-17
JP4733350B2 (ja) 2011-07-27
WO2003080053A1 (en) 2003-10-02
CN100444839C (zh) 2008-12-24
AR040400A1 (es) 2005-04-06
NZ535314A (en) 2007-08-31
AU2003220384B2 (en) 2007-05-10
TW200304811A (en) 2003-10-16
JP2005533005A (ja) 2005-11-04
CA2479126A1 (en) 2003-10-02
EP1485089A1 (en) 2004-12-15
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CA2479126C (en) 2011-11-15
CN1652779A (zh) 2005-08-10

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