UA78273C2 - Bilayer pharmaceutical tablet containing telmisartan and hydrochlorothiazide and method for producing thereof - Google Patents
Bilayer pharmaceutical tablet containing telmisartan and hydrochlorothiazide and method for producing thereof Download PDFInfo
- Publication number
- UA78273C2 UA78273C2 UA20040806794A UA20040806794A UA78273C2 UA 78273 C2 UA78273 C2 UA 78273C2 UA 20040806794 A UA20040806794 A UA 20040806794A UA 20040806794 A UA20040806794 A UA 20040806794A UA 78273 C2 UA78273 C2 UA 78273C2
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- Prior art keywords
- tablet
- layer
- telmisartan
- composition
- tablets
- Prior art date
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- 238000004519 manufacturing process Methods 0.000 title description 8
- OZCVMXDGSSXWFT-UHFFFAOYSA-N 6-chloro-1,1-dioxo-3,4-dihydro-2h-1$l^{6},2,4-benzothiadiazine-7-sulfonamide;2-[4-[[4-methyl-6-(1-methylbenzimidazol-2-yl)-2-propylbenzimidazol-1-yl]methyl]phenyl]benzoic acid Chemical compound C1=C(Cl)C(S(=O)(=O)N)=CC2=C1NCNS2(=O)=O.CCCC1=NC2=C(C)C=C(C=3N(C4=CC=CC=C4N=3)C)C=C2N1CC(C=C1)=CC=C1C1=CC=CC=C1C(O)=O OZCVMXDGSSXWFT-UHFFFAOYSA-N 0.000 title 1
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- A61K9/2072—Pills, tablets, discs, rods characterised by shape, structure or size; Tablets with holes, special break lines or identification marks; Partially coated tablets; Disintegrating flat shaped forms
- A61K9/2086—Layered tablets, e.g. bilayer tablets; Tablets of the type inert core-active coat
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Landscapes
- Health & Medical Sciences (AREA)
- Life Sciences & Earth Sciences (AREA)
- Veterinary Medicine (AREA)
- Chemical & Material Sciences (AREA)
- Public Health (AREA)
- Medicinal Chemistry (AREA)
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- Heart & Thoracic Surgery (AREA)
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- Urology & Nephrology (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Medicinal Preparation (AREA)
- Analysing Materials By The Use Of Radiation (AREA)
- Inorganic Insulating Materials (AREA)
- Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
- Lubricants (AREA)
- Separation Using Semi-Permeable Membranes (AREA)
- Medicines Containing Material From Animals Or Micro-Organisms (AREA)
- Treatment Of Liquids With Adsorbents In General (AREA)
- Solid-Sorbent Or Filter-Aiding Compositions (AREA)
Applications Claiming Priority (1)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| PCT/EP2002/000395 WO2003059327A1 (en) | 2002-01-16 | 2002-01-16 | Bilayer pharmaceutical tablet comprising telmisartan and a diuretic and preparation thereof |
Publications (1)
| Publication Number | Publication Date |
|---|---|
| UA78273C2 true UA78273C2 (en) | 2007-03-15 |
Family
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Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
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| UA20040806794A UA78273C2 (en) | 2002-01-16 | 2002-01-16 | Bilayer pharmaceutical tablet containing telmisartan and hydrochlorothiazide and method for producing thereof |
Country Status (30)
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| US (3) | US20050089575A1 (bg) |
| EP (3) | EP2260833B1 (bg) |
| JP (2) | JP4181503B2 (bg) |
| KR (2) | KR100851770B1 (bg) |
| CN (2) | CN101352421A (bg) |
| AT (1) | ATE380547T1 (bg) |
| AU (2) | AU2002242676B2 (bg) |
| BG (3) | BG66524B1 (bg) |
| BR (1) | BR0215514A (bg) |
| CA (2) | CA2651604C (bg) |
| CY (3) | CY1107226T1 (bg) |
| CZ (1) | CZ303145B6 (bg) |
| DE (1) | DE60224096T3 (bg) |
| DK (3) | DK2260833T3 (bg) |
| EA (2) | EA007614B1 (bg) |
| ES (3) | ES2400138T3 (bg) |
| HK (1) | HK1073785A1 (bg) |
| HR (1) | HRP20040649B1 (bg) |
| HU (1) | HU229941B1 (bg) |
| IL (4) | IL162754A0 (bg) |
| ME (1) | ME02761B (bg) |
| MX (1) | MXPA04006997A (bg) |
| NO (3) | NO345891B1 (bg) |
| NZ (1) | NZ534502A (bg) |
| PT (3) | PT2260833E (bg) |
| RS (1) | RS52012B (bg) |
| SI (1) | SI1467712T2 (bg) |
| SK (1) | SK288439B6 (bg) |
| UA (1) | UA78273C2 (bg) |
| WO (1) | WO2003059327A1 (bg) |
Families Citing this family (108)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| EP2260833B1 (en) * | 2002-01-16 | 2012-11-21 | Boehringer Ingelheim Pharma GmbH & Co. KG | Bilayer pharmaceutical tablet comprising telmisartan and a diuretic |
| US7407955B2 (en) | 2002-08-21 | 2008-08-05 | Boehringer Ingelheim Pharma Gmbh & Co., Kg | 8-[3-amino-piperidin-1-yl]-xanthines, the preparation thereof and their use as pharmaceutical compositions |
| US8980870B2 (en) | 2002-09-24 | 2015-03-17 | Boehringer Ingelheim International Gmbh | Solid telmisartan pharmaceutical formulations |
| DE10244681A1 (de) * | 2002-09-24 | 2004-04-08 | Boehringer Ingelheim International Gmbh | Neue feste Telmisartan enthaltende pharmazeutische Formulierungen und deren Herstellung |
| US20040224917A1 (en) | 2003-01-14 | 2004-11-11 | Gilead Sciences, Inc. | Compositions and methods for combination antiviral therapy |
| DE10319450A1 (de) * | 2003-04-30 | 2004-11-18 | Boehringer Ingelheim Pharma Gmbh & Co. Kg | Pharmazeutische Formulierung des Telmisartan Natriumsalzes |
| US9029363B2 (en) | 2003-04-30 | 2015-05-12 | Boehringer Ingelheim International Gmbh | Telmisartan sodium salt pharmaceutical formulation |
| CA2532450C (en) * | 2003-07-16 | 2012-09-11 | Boehringer Ingelheim International Gmbh | Chlorthalidone combinations |
| WO2005082329A2 (en) * | 2004-02-19 | 2005-09-09 | Ranbaxy Laboratories Limited | Process for the preparation of solid dosage forms of valsartan and hydrochlorthiazide |
| US20060078615A1 (en) * | 2004-10-12 | 2006-04-13 | Boehringer Ingelheim International Gmbh | Bilayer tablet of telmisartan and simvastatin |
| MX2007004426A (es) | 2004-10-15 | 2007-06-14 | Teva Pharma | Procesos para preparar telmisartan. |
| US20060293377A1 (en) * | 2004-11-03 | 2006-12-28 | Shlomit Wizel | Amorphous and polymorphic forms of telmisartan sodium |
| DE102004054054A1 (de) | 2004-11-05 | 2006-05-11 | Boehringer Ingelheim Pharma Gmbh & Co. Kg | Verfahren zur Herstellung chiraler 8-(3-Amino-piperidin-1-yl)-xanthine |
| UA89065C2 (ru) * | 2004-11-05 | 2009-12-25 | Бёрингэр Ингэльхайм Интэрнациональ Гмбх | Двухслойная таблетка, которая содержит телмисартан и амлодипин |
| CN101080225A (zh) * | 2004-12-17 | 2007-11-28 | 贝林格尔·英格海姆国际有限公司 | 包含替米沙坦及氢氯噻嗪的组合治疗 |
| CN100370984C (zh) * | 2005-03-11 | 2008-02-27 | 浙江泰利森药业有限公司 | 替米沙坦分散片及其制备方法 |
| TWI471145B (zh) | 2005-06-13 | 2015-02-01 | Bristol Myers Squibb & Gilead Sciences Llc | 單一式藥學劑量型 |
| TWI375560B (en) | 2005-06-13 | 2012-11-01 | Gilead Sciences Inc | Composition comprising dry granulated emtricitabine and tenofovir df and method for making the same |
| TWI388345B (zh) * | 2005-06-27 | 2013-03-11 | Sankyo Co | 用於高血壓之預防或治療之包含血管緊張素ⅱ受體拮抗劑及鈣通道阻斷劑之固體劑型 |
| GT200600371A (es) * | 2005-08-17 | 2007-03-21 | Formas de dosis sólidas de valsartan y amlodipina y método para hacer las mismas | |
| CA2623018A1 (en) * | 2005-11-22 | 2007-05-31 | Teva Pharmaceutical Industries Ltd. | Pharmaceutical compositions of telmisartan |
| US20070116759A1 (en) * | 2005-11-22 | 2007-05-24 | Gershon Kolatkar | Pharmaceutical compositions of telmisartan |
| US8637078B2 (en) * | 2005-11-24 | 2014-01-28 | Boehringer Ingelheim International Gmbh | Bilayer tablet comprising telmisartan and diuretic |
| US20070259930A1 (en) * | 2006-04-10 | 2007-11-08 | Knopp Neurosciences, Inc. | Compositions and methods of using r(+) pramipexole |
| US8518926B2 (en) * | 2006-04-10 | 2013-08-27 | Knopp Neurosciences, Inc. | Compositions and methods of using (R)-pramipexole |
| EP1852108A1 (en) | 2006-05-04 | 2007-11-07 | Boehringer Ingelheim Pharma GmbH & Co.KG | DPP IV inhibitor formulations |
| EA030606B1 (ru) | 2006-05-04 | 2018-08-31 | Бёрингер Ингельхайм Интернациональ Гмбх | Способы приготовления лекарственного средства, содержащего полиморфы |
| PE20110235A1 (es) | 2006-05-04 | 2011-04-14 | Boehringer Ingelheim Int | Combinaciones farmaceuticas que comprenden linagliptina y metmorfina |
| KR20090021169A (ko) | 2006-05-16 | 2009-02-27 | 크놉 뉴로사이언시스 인코포레이티드 | Ｒ(+) 및 ｓ(-) 프라미펙솔을 포함하는 조성물 및 이의 사용 방법 |
| EP2465500A1 (en) | 2006-05-16 | 2012-06-20 | Knopp Neurosciences, Inc. | Therapeutically effective amounts of R(+) and S(-) pramipexole for use in the treatment of parkinson's disease |
| NZ573173A (en) | 2006-06-01 | 2012-03-30 | Msd Consumer Care Inc | Phenylephrine pharmaceutical formulation and compositions for colonic absorption |
| CA2654890C (en) | 2006-06-16 | 2015-10-06 | Lek Pharmaceuticals D.D. | Pharmaceutical composition |
| AR061627A1 (es) * | 2006-06-27 | 2008-09-10 | Novartis Ag | Formas de dosificacion solidas de valsartan, amlodipina, e hidroclorotiazida, y metodo para elaborarlas |
| KR100888131B1 (ko) * | 2006-10-10 | 2009-03-11 | 한올제약주식회사 | 시간차 투약 원리를 이용한 심혈관계 질환 치료용 복합제제 |
| EP2079452A4 (en) * | 2006-10-30 | 2010-01-06 | Hanall Pharmaceutical Co Ltd | CONTROLLED RELEASE PHARMACEUTICAL COMPOSITION CONTAINING THIAZIDS AND BLOCKERS OF ANGIOTENSIN II RECEPTORS |
| US8524695B2 (en) * | 2006-12-14 | 2013-09-03 | Knopp Neurosciences, Inc. | Modified release formulations of (6R)-4,5,6,7-tetrahydro-N6-propyl-2,6-benzothiazole-diamine and methods of using the same |
| WO2008113056A2 (en) | 2007-03-14 | 2008-09-18 | Knopp Neurosciences, Inc. | Synthesis of chirally purified substituted benzothiazole diamines |
| EP1970053A1 (en) * | 2007-03-14 | 2008-09-17 | Boehringer Ingelheim Pharma GmbH & Co. KG | Pharmaceutical composition |
| US20080286344A1 (en) * | 2007-05-16 | 2008-11-20 | Olivia Darmuzey | Solid form |
| US20090004248A1 (en) * | 2007-06-29 | 2009-01-01 | Frank Bunick | Dual portion dosage lozenge form |
| US20100247649A1 (en) * | 2007-10-30 | 2010-09-30 | Dr. Reddy's Laboratories Ltd. | Pharmaceutical formulations comprising telmisartan and hydrochlorothiazide |
| CN101842085B (zh) | 2007-10-31 | 2013-01-30 | 麦克内尔-Ppc股份有限公司 | 口腔崩解剂型 |
| PL2252273T3 (pl) * | 2008-03-19 | 2017-07-31 | Ratiopharm Gmbh | Stała kompozycja farmaceutyczna zawierająca niepeptydowy związek antagonistyczny receptora angiotensyny II i środek moczopędny |
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| EP2291177A2 (en) * | 2008-05-05 | 2011-03-09 | Farmaprojects, S.A. | Stable pharmaceutical compositions and their processes for preparation suitable for industrial scale |
| CZ301070B6 (cs) * | 2008-07-31 | 2009-10-29 | Zentiva, A. S. | Telmisartan tablety |
| KR20200118243A (ko) | 2008-08-06 | 2020-10-14 | 베링거 인겔하임 인터내셔날 게엠베하 | 메트포르민 요법이 부적합한 환자에서의 당뇨병 치료 |
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