TWI618537B - 糖尿病治療 - Google Patents

糖尿病治療 Download PDF

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Publication number
TWI618537B
TWI618537B TW100122087A TW100122087A TWI618537B TW I618537 B TWI618537 B TW I618537B TW 100122087 A TW100122087 A TW 100122087A TW 100122087 A TW100122087 A TW 100122087A TW I618537 B TWI618537 B TW I618537B
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TW
Taiwan
Prior art keywords
dpp
insulin
inhibitor
diabetes
long
Prior art date
Application number
TW100122087A
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English (en)
Chinese (zh)
Other versions
TW201212919A (en
Inventor
湯瑪斯 克林
麥可 馬克
里歐 湯瑪斯
Original Assignee
百靈佳殷格翰國際股份有限公司
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Family has litigation
First worldwide family litigation filed litigation Critical https://patents.darts-ip.com/?family=44509854&utm_source=google_patent&utm_medium=platform_link&utm_campaign=public_patent_search&patent=TWI618537(B) "Global patent litigation dataset” by Darts-ip is licensed under a Creative Commons Attribution 4.0 International License.
Application filed by 百靈佳殷格翰國際股份有限公司 filed Critical 百靈佳殷格翰國際股份有限公司
Publication of TW201212919A publication Critical patent/TW201212919A/zh
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    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/33Heterocyclic compounds
    • A61K31/395Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/495Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with two or more nitrogen atoms as the only ring heteroatoms, e.g. piperazine or tetrazines
    • A61K31/505Pyrimidines; Hydrogenated pyrimidines, e.g. trimethoprim
    • A61K31/519Pyrimidines; Hydrogenated pyrimidines, e.g. trimethoprim ortho- or peri-condensed with heterocyclic rings
    • A61K31/52Purines, e.g. adenine
    • A61K31/522Purines, e.g. adenine having oxo groups directly attached to the heterocyclic ring, e.g. hypoxanthine, guanine, acyclovir
    • AHUMAN NECESSITIES
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    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/13Amines
    • A61K31/155Amidines (), e.g. guanidine (H2N—C(=NH)—NH2), isourea (N=C(OH)—NH2), isothiourea (—N=C(SH)—NH2)
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/33Heterocyclic compounds
    • A61K31/395Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/435Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom
    • A61K31/44Non condensed pyridines; Hydrogenated derivatives thereof
    • A61K31/4427Non condensed pyridines; Hydrogenated derivatives thereof containing further heterocyclic ring systems
    • A61K31/4439Non condensed pyridines; Hydrogenated derivatives thereof containing further heterocyclic ring systems containing a five-membered ring with nitrogen as a ring hetero atom, e.g. omeprazole
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    • A61K38/16Peptides having more than 20 amino acids; Gastrins; Somatostatins; Melanotropins; Derivatives thereof
    • A61K38/17Peptides having more than 20 amino acids; Gastrins; Somatostatins; Melanotropins; Derivatives thereof from animals; from humans
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    • A61P3/04Anorexiants; Antiobesity agents
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    • A61P3/06Antihyperlipidemics
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
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    • A61P3/08Drugs for disorders of the metabolism for glucose homeostasis
    • AHUMAN NECESSITIES
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    • A61P3/10Drugs for disorders of the metabolism for glucose homeostasis for hyperglycaemia, e.g. antidiabetics
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    • A61P5/48Drugs for disorders of the endocrine system of the pancreatic hormones
    • A61P5/50Drugs for disorders of the endocrine system of the pancreatic hormones for increasing or potentiating the activity of insulin
    • AHUMAN NECESSITIES
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    • A61P9/04Inotropic agents, i.e. stimulants of cardiac contraction; Drugs for heart failure
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    • A61P9/06Antiarrhythmics
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    • A61P9/10Drugs for disorders of the cardiovascular system for treating ischaemic or atherosclerotic diseases, e.g. antianginal drugs, coronary vasodilators, drugs for myocardial infarction, retinopathy, cerebrovascula insufficiency, renal arteriosclerosis
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    • A61P9/12Antihypertensives
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    • A61P9/14Vasoprotectives; Antihaemorrhoidals; Drugs for varicose therapy; Capillary stabilisers
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    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K2300/00Mixtures or combinations of active ingredients, wherein at least one active ingredient is fully defined in groups A61K31/00 - A61K41/00

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  • Health & Medical Sciences (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Veterinary Medicine (AREA)
  • Public Health (AREA)
  • Chemical & Material Sciences (AREA)
  • General Health & Medical Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • Medicinal Chemistry (AREA)
  • Engineering & Computer Science (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • General Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Diabetes (AREA)
  • Epidemiology (AREA)
  • Endocrinology (AREA)
  • Cardiology (AREA)
  • Obesity (AREA)
  • Hematology (AREA)
  • Heart & Thoracic Surgery (AREA)
  • Gastroenterology & Hepatology (AREA)
  • Immunology (AREA)
  • Proteomics, Peptides & Aminoacids (AREA)
  • Zoology (AREA)
  • Biomedical Technology (AREA)
  • Neurology (AREA)
  • Neurosurgery (AREA)
  • Emergency Medicine (AREA)
  • Urology & Nephrology (AREA)
  • Ophthalmology & Optometry (AREA)
  • Rheumatology (AREA)
  • Physical Education & Sports Medicine (AREA)
  • Reproductive Health (AREA)
  • Orthopedic Medicine & Surgery (AREA)
  • Hospice & Palliative Care (AREA)
  • Vascular Medicine (AREA)
  • Dermatology (AREA)
  • Pregnancy & Childbirth (AREA)
TW100122087A 2010-06-24 2011-06-23 糖尿病治療 TWI618537B (zh)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
??10167243.4 2010-06-24
EP10167243 2010-06-24

Publications (2)

Publication Number Publication Date
TW201212919A TW201212919A (en) 2012-04-01
TWI618537B true TWI618537B (zh) 2018-03-21

Family

ID=44509854

Family Applications (1)

Application Number Title Priority Date Filing Date
TW100122087A TWI618537B (zh) 2010-06-24 2011-06-23 糖尿病治療

Country Status (18)

Country Link
US (1) US9149478B2 (cg-RX-API-DMAC7.html)
EP (4) EP3124041A1 (cg-RX-API-DMAC7.html)
JP (3) JP5843855B2 (cg-RX-API-DMAC7.html)
KR (6) KR20200028498A (cg-RX-API-DMAC7.html)
CN (2) CN102971005A (cg-RX-API-DMAC7.html)
AR (1) AR082767A1 (cg-RX-API-DMAC7.html)
AU (1) AU2011268940B2 (cg-RX-API-DMAC7.html)
BR (1) BR112012032579B1 (cg-RX-API-DMAC7.html)
CA (2) CA2803504C (cg-RX-API-DMAC7.html)
CL (1) CL2012003393A1 (cg-RX-API-DMAC7.html)
EA (2) EA201991014A1 (cg-RX-API-DMAC7.html)
ES (2) ES2802243T3 (cg-RX-API-DMAC7.html)
IL (1) IL222778A0 (cg-RX-API-DMAC7.html)
MX (1) MX2012014247A (cg-RX-API-DMAC7.html)
NZ (1) NZ603319A (cg-RX-API-DMAC7.html)
PH (1) PH12012502524A1 (cg-RX-API-DMAC7.html)
TW (1) TWI618537B (cg-RX-API-DMAC7.html)
WO (1) WO2011161161A1 (cg-RX-API-DMAC7.html)

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CN107961377B (zh) 2010-05-05 2022-11-22 勃林格殷格翰国际有限公司 组合疗法
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