TNSN07244A1 - Dipeptidyl peptidase-iv inhibitors - Google Patents

Dipeptidyl peptidase-iv inhibitors

Info

Publication number
TNSN07244A1
TNSN07244A1 TNP2007000244A TNSN07244A TNSN07244A1 TN SN07244 A1 TNSN07244 A1 TN SN07244A1 TN P2007000244 A TNP2007000244 A TN P2007000244A TN SN07244 A TNSN07244 A TN SN07244A TN SN07244 A1 TNSN07244 A1 TN SN07244A1
Authority
TN
Tunisia
Prior art keywords
dpp
inhibitors
compounds
dipeptidyl peptidase
present
Prior art date
Application number
TNP2007000244A
Other languages
English (en)
French (fr)
Inventor
Heiko Kroth
Tim Feuerstein
Frank Richter
Jurgen Boer
Michael Essers
Bert Nolte
Matthias Schneider
Matthias Hochguertel
Fritz-Frieder Frickel
Arthur Taveras
Original Assignee
Alantos Pharmaceuticals Inc
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Family has litigation
First worldwide family litigation filed litigation Critical https://patents.darts-ip.com/?family=36694223&utm_source=google_patent&utm_medium=platform_link&utm_campaign=public_patent_search&patent=TNSN07244(A1) "Global patent litigation dataset” by Darts-ip is licensed under a Creative Commons Attribution 4.0 International License.
Application filed by Alantos Pharmaceuticals Inc filed Critical Alantos Pharmaceuticals Inc
Publication of TNSN07244A1 publication Critical patent/TNSN07244A1/fr

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D207/00—Heterocyclic compounds containing five-membered rings not condensed with other rings, with one nitrogen atom as the only ring hetero atom
    • C07D207/02—Heterocyclic compounds containing five-membered rings not condensed with other rings, with one nitrogen atom as the only ring hetero atom with only hydrogen or carbon atoms directly attached to the ring nitrogen atom
    • C07D207/04—Heterocyclic compounds containing five-membered rings not condensed with other rings, with one nitrogen atom as the only ring hetero atom with only hydrogen or carbon atoms directly attached to the ring nitrogen atom having no double bonds between ring members or between ring members and non-ring members
    • C07D207/10—Heterocyclic compounds containing five-membered rings not condensed with other rings, with one nitrogen atom as the only ring hetero atom with only hydrogen or carbon atoms directly attached to the ring nitrogen atom having no double bonds between ring members or between ring members and non-ring members with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
    • C07D207/16—Carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals
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    • A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/41—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having five-membered rings with two or more ring hetero atoms, at least one of which being nitrogen, e.g. tetrazole
    • A61K31/415—1,2-Diazoles
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    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D209/00—Heterocyclic compounds containing five-membered rings, condensed with other rings, with one nitrogen atom as the only ring hetero atom
    • C07D209/02—Heterocyclic compounds containing five-membered rings, condensed with other rings, with one nitrogen atom as the only ring hetero atom condensed with one carbocyclic ring
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    • C07D209/00—Heterocyclic compounds containing five-membered rings, condensed with other rings, with one nitrogen atom as the only ring hetero atom
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    • C—CHEMISTRY; METALLURGY
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    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D401/00—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom
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    • C07D401/12—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings linked by a chain containing hetero atoms as chain links
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    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D403/00—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, not provided for by group C07D401/00
    • C07D403/02—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, not provided for by group C07D401/00 containing two hetero rings
    • C07D403/12—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, not provided for by group C07D401/00 containing two hetero rings linked by a chain containing hetero atoms as chain links
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    • C07D413/02—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms containing two hetero rings
    • C07D413/12—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms containing two hetero rings linked by a chain containing hetero atoms as chain links
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    • C07D487/00—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00
    • C07D487/02—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00 in which the condensed system contains two hetero rings
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    • C07D495/00—Heterocyclic compounds containing in the condensed system at least one hetero ring having sulfur atoms as the only ring hetero atoms
    • C07D495/02—Heterocyclic compounds containing in the condensed system at least one hetero ring having sulfur atoms as the only ring hetero atoms in which the condensed system contains two hetero rings
    • C07D495/04—Ortho-condensed systems

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  • Health & Medical Sciences (AREA)
  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Engineering & Computer Science (AREA)
  • Bioinformatics & Cheminformatics (AREA)
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  • Public Health (AREA)
  • General Health & Medical Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • Medicinal Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • General Chemical & Material Sciences (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Neurology (AREA)
  • Neurosurgery (AREA)
  • Biomedical Technology (AREA)
  • Psychiatry (AREA)
  • Addiction (AREA)
  • Immunology (AREA)
  • Diabetes (AREA)
  • Ophthalmology & Optometry (AREA)
  • Endocrinology (AREA)
  • Hematology (AREA)
  • Obesity (AREA)
  • Reproductive Health (AREA)
  • Heart & Thoracic Surgery (AREA)
  • Cardiology (AREA)
  • Urology & Nephrology (AREA)
  • Rheumatology (AREA)
  • Physical Education & Sports Medicine (AREA)
  • Orthopedic Medicine & Surgery (AREA)
  • Virology (AREA)
  • Oncology (AREA)
  • Psychology (AREA)
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  • AIDS & HIV (AREA)
  • Hospice & Palliative Care (AREA)
TNP2007000244A 2005-04-22 2007-06-26 Dipeptidyl peptidase-iv inhibitors TNSN07244A1 (en)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
US67415105P 2005-04-22 2005-04-22
PCT/US2006/015200 WO2006116157A2 (en) 2005-04-22 2006-04-21 Dipeptidyl peptidase-iv inhibitors

Publications (1)

Publication Number Publication Date
TNSN07244A1 true TNSN07244A1 (en) 2008-11-21

Family

ID=36694223

Family Applications (1)

Application Number Title Priority Date Filing Date
TNP2007000244A TNSN07244A1 (en) 2005-04-22 2007-06-26 Dipeptidyl peptidase-iv inhibitors

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US (3) US7553861B2 (cg-RX-API-DMAC7.html)
EP (1) EP1888562B1 (cg-RX-API-DMAC7.html)
JP (2) JP4568361B2 (cg-RX-API-DMAC7.html)
KR (1) KR20080000665A (cg-RX-API-DMAC7.html)
CN (1) CN101277949A (cg-RX-API-DMAC7.html)
AP (1) AP2007004234A0 (cg-RX-API-DMAC7.html)
AU (2) AU2006239929B2 (cg-RX-API-DMAC7.html)
BR (1) BRPI0608469A2 (cg-RX-API-DMAC7.html)
CA (1) CA2599419A1 (cg-RX-API-DMAC7.html)
CR (1) CR9462A (cg-RX-API-DMAC7.html)
EA (1) EA200702208A1 (cg-RX-API-DMAC7.html)
ES (1) ES2477868T3 (cg-RX-API-DMAC7.html)
IL (1) IL186607A0 (cg-RX-API-DMAC7.html)
MA (1) MA29387B1 (cg-RX-API-DMAC7.html)
MX (1) MX2007011453A (cg-RX-API-DMAC7.html)
NO (1) NO20075973L (cg-RX-API-DMAC7.html)
TN (1) TNSN07244A1 (cg-RX-API-DMAC7.html)
WO (1) WO2006116157A2 (cg-RX-API-DMAC7.html)
ZA (1) ZA200708179B (cg-RX-API-DMAC7.html)

Families Citing this family (73)

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Publication number Priority date Publication date Assignee Title
US7407955B2 (en) 2002-08-21 2008-08-05 Boehringer Ingelheim Pharma Gmbh & Co., Kg 8-[3-amino-piperidin-1-yl]-xanthines, the preparation thereof and their use as pharmaceutical compositions
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RU2394570C2 (ru) 2004-02-20 2010-07-20 Новартис Аг Ингибиторы dpp-iv для лечения нейродегенерации и когнитивных расстройств
KR100844593B1 (ko) * 2004-03-09 2008-07-07 내셔날 헬스 리서치 인스티튜트 피롤리딘 화합물
JP4568361B2 (ja) * 2005-04-22 2010-10-27 アラントス・ファーマシューティカルズ・ホールディング・インコーポレーテッド ジペプチジルペプチダーゼ−ｉｖ阻害剤

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BRPI0608469A2 (pt) 2010-01-05
CR9462A (es) 2008-04-16
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