IL73534A
(en)
|
1983-11-18 |
1990-12-23 |
Riker Laboratories Inc |
1h-imidazo(4,5-c)quinoline-4-amines,their preparation and pharmaceutical compositions containing certain such compounds
|
JP2890448B2
(ja)
|
1988-04-26 |
1999-05-17 |
日産化学工業株式会社 |
ピラゾロピリジン系メバロノラクトン類
|
US5658889A
(en)
|
1989-01-24 |
1997-08-19 |
Gensia Pharmaceuticals, Inc. |
Method and compounds for aica riboside delivery and for lowering blood glucose
|
US4994468A
(en)
|
1989-03-07 |
1991-02-19 |
Kyowa Hakko Kogyo Co., Ltd. |
Imidazoquinolone derivatives
|
US5721356A
(en)
*
|
1989-09-15 |
1998-02-24 |
Gensia, Inc. |
Orally active adenosine kinase inhibitors
|
US5763596A
(en)
|
1989-09-15 |
1998-06-09 |
Metabasis Therapeutics, Inc. |
C-4' modified adenosine kinase inhibitors
|
US5864033A
(en)
|
1989-09-15 |
1999-01-26 |
Metabasis Therapeutics, Inc. |
Adenosine kinase inhibitors
|
US5795977A
(en)
|
1989-09-15 |
1998-08-18 |
Metabasis Therapeutics, Inc. |
Water soluble adenosine kinase inhibitors
|
US5763597A
(en)
|
1989-09-15 |
1998-06-09 |
Metabasis Therapeutics, Inc. |
Orally active adenosine kinase inhibitors
|
US5674998A
(en)
|
1989-09-15 |
1997-10-07 |
Gensia Inc. |
C-4' modified adenosine kinase inhibitors
|
US5726302A
(en)
|
1989-09-15 |
1998-03-10 |
Gensia Inc. |
Water soluble adenosine kinase inhibitors
|
US5646128A
(en)
|
1989-09-15 |
1997-07-08 |
Gensia, Inc. |
Methods for treating adenosine kinase related conditions
|
JPH03271289A
(ja)
|
1990-03-16 |
1991-12-03 |
Nissan Chem Ind Ltd |
ピラゾロピリジン誘導体の製造法及びジヒドロピラゾロピリジン誘導体
|
US5389640A
(en)
|
1991-03-01 |
1995-02-14 |
Minnesota Mining And Manufacturing Company |
1-substituted, 2-substituted 1H-imidazo[4,5-c]quinolin-4-amines
|
JP3130342B2
(ja)
|
1991-10-04 |
2001-01-31 |
日産化学工業株式会社 |
動脈硬化性血管内膜肥厚抑制薬
|
JP3271289B2
(ja)
|
1992-02-28 |
2002-04-02 |
スズキ株式会社 |
4サイクルエンジンのバルブ駆動装置
|
US5502187A
(en)
|
1992-04-03 |
1996-03-26 |
The Upjohn Company |
Pharmaceutically active bicyclic-heterocyclic amines
|
JPH08502721A
(ja)
|
1992-04-03 |
1996-03-26 |
ジ・アップジョン・カンパニー |
医薬的に活性な二環式‐複素環アミン
|
JPH05310700A
(ja)
|
1992-05-12 |
1993-11-22 |
Sagami Chem Res Center |
縮合ピリジン系メバロノラクトン中間体及びその製法
|
WO1995011898A1
(fr)
|
1992-05-12 |
1995-05-04 |
Nissan Chemical Industries Ltd. |
Intermediaire condense de synthese du mevalonolactone de type pyridine et procede de fabrication de cet intermediaire
|
JPH0641114A
(ja)
|
1992-05-25 |
1994-02-15 |
Nissan Chem Ind Ltd |
新規メバロノラクトン類とその製法
|
JPH06116239A
(ja)
|
1992-10-05 |
1994-04-26 |
Nissan Chem Ind Ltd |
7−置換−3,5−ジヒドロキシヘプタ−6−イン酸類
|
AU5161193A
(en)
|
1992-10-16 |
1994-05-09 |
Nippon Soda Co., Ltd. |
Pyrimidine derivative
|
DE69432629T3
(de)
|
1993-01-25 |
2008-01-17 |
Takeda Pharmaceutical Co. Ltd. |
Antikörper gegen beta-amyloid oder derivative davon und seine verwendung
|
WO1994018215A1
(fr)
|
1993-02-03 |
1994-08-18 |
Gensia, Inc. |
Inhibiteurs d'adenosine-kinase comprenant des derives de lyxofuranosyle
|
DE4304455A1
(de)
|
1993-02-15 |
1994-08-18 |
Bayer Ag |
Heterocyclisch substituierte Phenyl-cyclohexan-carbonsäurederivate
|
JP3119758B2
(ja)
|
1993-02-24 |
2000-12-25 |
日清製粉株式会社 |
7−アザインドール誘導体及びこれを有効成分とする抗潰瘍薬
|
JP3350739B2
(ja)
|
1993-06-10 |
2002-11-25 |
コニカ株式会社 |
黒白ハロゲン化銀写真感光材料の現像処理方法
|
CN1102644A
(zh)
|
1993-11-11 |
1995-05-17 |
财团法人相模中央化学研究所 |
缩合吡啶型甲羟戊酸内酯中间体及其制备方法
|
JPH07281365A
(ja)
|
1994-04-07 |
1995-10-27 |
Konica Corp |
写真感光材料の処理方法
|
ATE159257T1
(de)
|
1994-05-03 |
1997-11-15 |
Ciba Geigy Ag |
Pyrrolopyrimidinderivate mit antiproliferativer wirkung
|
JP3448724B2
(ja)
|
1995-11-29 |
2003-09-22 |
コニカ株式会社 |
ハロゲン化銀写真感光材料用現像剤及びその処理方法
|
GB9604361D0
(en)
|
1996-02-29 |
1996-05-01 |
Pharmacia Spa |
4-Substituted pyrrolopyrimidine compounds as tyrosine kinase inhibitors
|
KR20000064601A
(ko)
*
|
1996-03-15 |
2000-11-06 |
한스 루돌프 하우스, 헨리테 브룬너, 베아트리체 귄터 |
신규의n-7-헤테로시클릴피롤로[2,3-d]피리딘및�그의용도
|
JPH10213887A
(ja)
|
1996-11-26 |
1998-08-11 |
Konica Corp |
黒白ハロゲン化銀写真感光材料の処理方法
|
IL129825A0
(en)
*
|
1996-11-27 |
2000-02-29 |
Pfizer |
Fused bicyclic pyrimidine derivatives
|
EP0846981A1
(fr)
|
1996-12-03 |
1998-06-10 |
Konica Corporation |
Procédé de traitement d'un produit photographique noir et blanc à l'halogénure d'argent sensible à la lumière
|
JP3543249B2
(ja)
|
1996-12-18 |
2004-07-14 |
コニカミノルタホールディングス株式会社 |
黒白ハロゲン化銀写真感光材料の処理方法
|
EP2305709A1
(fr)
|
1997-04-09 |
2011-04-06 |
Intellect Neurosciences, Inc. |
Anticorps recombinants spécifiques à des fins bêta-amyloïdes, codage ADN et procédés d'utilisation associés
|
US8173127B2
(en)
|
1997-04-09 |
2012-05-08 |
Intellect Neurosciences, Inc. |
Specific antibodies to amyloid beta peptide, pharmaceutical compositions and methods of use thereof
|
US6929808B2
(en)
|
2000-11-03 |
2005-08-16 |
Proteotech, Inc. |
Methods of isolating amyloid-inhibiting compounds and use of compounds isolated from Uncaria tomentosa and related plants
|
TWI239847B
(en)
|
1997-12-02 |
2005-09-21 |
Elan Pharm Inc |
N-terminal fragment of Abeta peptide and an adjuvant for preventing and treating amyloidogenic disease
|
US6905686B1
(en)
|
1997-12-02 |
2005-06-14 |
Neuralab Limited |
Active immunization for treatment of alzheimer's disease
|
CZ20004727A3
(cs)
|
1998-06-19 |
2002-03-13 |
Pfizer Products Inc. |
Deriváty pyrrolo[2,3-d] pyrimidinu
|
PA8474101A1
(es)
|
1998-06-19 |
2000-09-29 |
Pfizer Prod Inc |
Compuestos de pirrolo [2,3-d] pirimidina
|
YU25500A
(sh)
|
1999-05-11 |
2003-08-29 |
Pfizer Products Inc. |
Postupak za sintezu analoga nukleozida
|
US6309811B2
(en)
|
1999-07-21 |
2001-10-30 |
Eastman Kodak Company |
Color photographic element containing nitrogen heterocycle derivative and inhibitor releasing coupler
|
EP3070100B1
(fr)
|
2000-02-24 |
2021-07-07 |
Washington University St. Louis |
Anticorps humanisés qui séquestrent un peptide amyloïde beta
|
JP2001302515A
(ja)
|
2000-04-18 |
2001-10-31 |
Sumitomo Pharmaceut Co Ltd |
ポリ(adp−リボース)ポリメラーゼ阻害剤
|
AU2001264313A1
(en)
|
2000-06-20 |
2002-01-02 |
Japan Tobacco Inc. |
Pyrazolopyridine compounds and use thereof as drugs
|
EA200300717A1
(ru)
|
2000-12-22 |
2003-12-25 |
Уайт |
Гетероциклилиндазольные и -азаиндазольные соединения в качестве 5-гидрокситриптамин-6-лигандов
|
GB0111186D0
(en)
|
2001-05-08 |
2001-06-27 |
Smithkline Beecham Plc |
Novel compounds
|
WO2003000187A2
(fr)
*
|
2001-06-21 |
2003-01-03 |
Ariad Pharmaceuticals, Inc. |
Nouvelles pyrazolo-pyrimidines et pyrrolo-pyrimidines et leur utilisation
|
JP2005503789A
(ja)
|
2001-08-17 |
2005-02-10 |
イーライ・リリー・アンド・カンパニー |
抗Aβ抗体
|
US20030195205A1
(en)
|
2001-11-02 |
2003-10-16 |
Pfizer Inc. |
PDE9 inhibitors for treating cardiovascular disorders
|
AU2002339230A1
(en)
|
2002-03-08 |
2003-09-22 |
Decode Genetics Ehf. |
A susceptibility gene for late-onset idiopathic parkinson's disease
|
CA2495216A1
(fr)
|
2002-08-12 |
2004-02-19 |
Sugen, Inc. |
3-pyrrolyl-pyridopyrazoles et 3-pyrrolyl-indazoles utilises en tant que nouveaux inhibiteurs de la proteine kinase
|
SE0202463D0
(sv)
|
2002-08-14 |
2002-08-14 |
Astrazeneca Ab |
Novel compounds
|
DE10238723A1
(de)
|
2002-08-23 |
2004-03-11 |
Bayer Ag |
Phenyl-substituierte Pyrazolyprimidine
|
DE10238724A1
(de)
|
2002-08-23 |
2004-03-04 |
Bayer Ag |
Alkyl-substituierte Pyrazolpyrimidine
|
MXPA05003621A
(es)
|
2002-10-09 |
2005-10-19 |
Rinat Neuroscience Corp |
Metodos de tratamiento de la enfermedad de alzheimer usando anticuerpos dirigidos contra el peptido beta amiloide y composiciones de los mismos.
|
DE10259382A1
(de)
|
2002-12-18 |
2004-07-01 |
Abbott Gmbh & Co. Kg |
3-Substituierte 3,4-Dihydro-thieno[2,3-d]pyrimidin-4-on-Derivate, ihre Herstellung und Verwendung
|
US20040220186A1
(en)
|
2003-04-30 |
2004-11-04 |
Pfizer Inc. |
PDE9 inhibitors for treating type 2 diabetes,metabolic syndrome, and cardiovascular disease
|
WO2004110996A1
(fr)
|
2003-06-19 |
2004-12-23 |
Pfizer Products Inc. |
Antagoniste de nk1
|
CA2538220A1
(fr)
|
2003-09-09 |
2005-03-24 |
Takeda Pharmaceutical Company Limited |
Utilisation d'un anticorps
|
WO2005044181A2
(fr)
|
2003-09-09 |
2005-05-19 |
Temple University-Of The Commonwealth System Of Higher Education |
Protection de tissus et de cellules des effets cytotoxiques d'un rayonnement ionisant par des inhibiteurs abl
|
PL1696920T3
(pl)
|
2003-12-19 |
2015-03-31 |
Plexxikon Inc |
Związki i sposoby opracowywania modulatorów Ret
|
US20050187389A1
(en)
*
|
2004-01-13 |
2005-08-25 |
Ambit Biosciences Corporation |
Pyrrolopyrimidine derivatives and analogs and their use in the treatment and prevention of diseases
|
JP2007519707A
(ja)
|
2004-02-02 |
2007-07-19 |
ファイザー・プロダクツ・インク |
ヒスタミン−3受容体モジュレーター
|
BRPI0509298A
(pt)
|
2004-04-01 |
2007-09-18 |
Lilly Co Eli |
composto, composição farmacêutica, métodos de inibir receptor h3 de histamina em um mamìfero, para tratar ou prevenir um distúrbio do sistema nervoso, obesidade, e um distúrbio ou doença, e, uso de um composto
|
AU2005236002A1
(en)
|
2004-04-02 |
2005-11-03 |
Vertex Pharmaceuticals Incorporated |
Azaindoles useful as inhibitors of rock and other protein kinases
|
US7456164B2
(en)
|
2004-05-07 |
2008-11-25 |
Pfizer, Inc |
3- or 4-monosubtituted phenol and thiophenol derivatives useful as H3 ligands
|
EP1595881A1
(fr)
|
2004-05-12 |
2005-11-16 |
Pfizer Limited |
Dérivés de tetrahydronaphthyridine en tant que ligands de récepteur H3 d'histamine
|
UA84208C2
(en)
|
2004-05-25 |
2008-09-25 |
Пфайзер Продактс Инк. |
Tetraazabenzo(e)azulene derivatives and analogs thereof
|
CA2570043A1
(fr)
|
2004-06-08 |
2005-12-22 |
Chiron Corporation |
Complexes de polypeptides env et methodes d'utilisation correspondantes
|
CA2572314A1
(fr)
|
2004-06-29 |
2006-01-12 |
Christopher N. Farthing |
Pyrrolo [2, 3-d] pyrimidines qui modulent l'activite ack1 et lck
|
BRPI0513959A
(pt)
|
2004-07-30 |
2008-05-20 |
Rinat Neuroscience Corp |
anticorpos dirigidos contra o peptìdeo beta-amilóide, suas composições farmacêuticas, kit e métodos de fabricação dos mesmos
|
WO2006042102A2
(fr)
|
2004-10-05 |
2006-04-20 |
Neurogen Corporation |
Composes de pyrrolo-pyridine, de pyrrolo-pyrimidine et composes heterocycliques apparentes
|
DK1802749T3
(da)
|
2004-10-21 |
2012-11-26 |
Mayo Foundation |
KASPP (LRRK2)-gen, dets fremstilling og anvendelse til påvisning og behandling af neurodegenerative lidelser
|
US7511056B2
(en)
|
2004-11-10 |
2009-03-31 |
Eli Lilly And Company |
TGF-β inhibitors
|
DE102004054634A1
(de)
|
2004-11-12 |
2006-05-18 |
Schwarz Pharma Ag |
Azaindolcarboxamide
|
WO2006069081A2
(fr)
|
2004-12-22 |
2006-06-29 |
Washington University In St. Louis |
Utilisation d'anticorps anti-a$g(b) pour le traitement d'un traumatisme cerebral
|
AU2006216799A1
(en)
|
2005-02-23 |
2006-08-31 |
Coley Pharmaceutical Group, Inc. |
Hydroxyalkyl substituted imidazonaphthyridines
|
PE20061323A1
(es)
|
2005-04-29 |
2007-02-09 |
Rinat Neuroscience Corp |
Anticuerpos dirigidos contra el peptido amiloide beta y metodos que utilizan los mismos
|
WO2006136924A1
(fr)
|
2005-06-22 |
2006-12-28 |
Pfizer Products Inc. |
Antagonistes du recepteur 3 de l'histamine
|
US8158673B2
(en)
|
2005-10-27 |
2012-04-17 |
Pfizer Inc. |
Histamine-3 receptor antagonists
|
JP2009514846A
(ja)
|
2005-11-04 |
2009-04-09 |
ファイザー・リミテッド |
テトラヒドロナフチリジン誘導体
|
WO2007063385A2
(fr)
|
2005-12-01 |
2007-06-07 |
Pfizer Products Inc. |
Antagonistes des recepteurs de l'histamine 3 pour des amines spirocycliques
|
WO2007069053A1
(fr)
|
2005-12-14 |
2007-06-21 |
Pfizer Products Inc. |
Antagonistes benzimidazoliques du récepteur h-3
|
EP1968568A4
(fr)
|
2005-12-22 |
2011-04-13 |
Glaxosmithkline Llc |
INHIBITEURS D'ACTIVITE Akt
|
AU2006330587B2
(en)
|
2005-12-23 |
2012-12-13 |
Glaxosmithkline Llc |
Azaindole inhibitors of aurora kinases
|
WO2007088450A2
(fr)
|
2006-02-01 |
2007-08-09 |
Pfizer Products Inc. |
Chromane antagoniste du récepteur h-3
|
WO2007088462A1
(fr)
|
2006-02-01 |
2007-08-09 |
Pfizer Products Inc. |
Antagonistes du récepteur du h-3 à base de spirochromane
|
WO2007099423A1
(fr)
|
2006-03-02 |
2007-09-07 |
Pfizer Products Inc. |
Dérivés de 1-pyrrolidine indane en tant qu'antagonistes du récepteur d'histamine 3
|
EP2007749A2
(fr)
|
2006-03-13 |
2008-12-31 |
Pfizer Products Inc. |
Tétralines en tant qu'antagonistes du récepteur h-3
|
CN101426927B
(zh)
|
2006-03-14 |
2012-05-23 |
塞尔卓姆股份公司 |
鉴定lrrk2相互作用分子和纯化lrrk2的方法
|
WO2007124096A2
(fr)
|
2006-04-21 |
2007-11-01 |
The Trustees Of Columbia University In The City Of New York |
Régulation de la morphologie des processus neuronaux par lrrk2
|
GB0610317D0
(en)
|
2006-05-24 |
2006-07-05 |
Medical Res Council |
Antiparasitic compounds and compositions
|
WO2007138431A2
(fr)
|
2006-05-30 |
2007-12-06 |
Pfizer Products Inc. |
Antagonistes de l'éther histamine-3 azabicyclique
|
BRPI0713738A2
(pt)
|
2006-06-20 |
2014-06-24 |
Novartis Ag |
Biomarcadores para a progressão de doença alzheimer
|
US8466163B2
(en)
|
2006-12-11 |
2013-06-18 |
Bionomics Limited |
Furo[2,3-d]pyrimidines and related compounds and methods for treating disease states by inhibiting tubulin polymerization
|
WO2008075007A1
(fr)
*
|
2006-12-21 |
2008-06-26 |
Cancer Research Technology Limited |
Composé bicyclohétéroarylés substitué par morpholino et leur utilisation en tant qu'agents anti-cancer
|
CN101631545B
(zh)
|
2007-01-22 |
2013-03-13 |
辉瑞产品公司 |
治疗性化合物的甲苯磺酸盐及其药物组合物
|
WO2008091799A2
(fr)
|
2007-01-22 |
2008-07-31 |
The Trustees Of Columbia University In The City Of New York |
Procédés basés sur des cellules, destinés à identifier des inhibiteurs de mutants lrrk2 associés à la maladie de parkinson
|
FR2912744B1
(fr)
|
2007-02-16 |
2012-09-07 |
Centre Nat Rech Scient |
Composes pyrrolo°2,3-b!pyridine,composes azaindoles utiles dans la synthese de ces composes pyrrolo°2,3-b!pyridine, leurs procedes de fabrication et leurs utilisations.
|
GB0706709D0
(en)
|
2007-04-05 |
2007-05-16 |
Medical Res Council |
Methods
|
CN101679313A
(zh)
*
|
2007-04-13 |
2010-03-24 |
休普基因公司 |
用于治疗癌症或过度增殖性疾病的axl激酶抑制剂
|
BRPI0811280B8
(pt)
|
2007-05-11 |
2021-05-25 |
Pfizer |
compostos amino-heterocíclicos, composição farmacêutica que os compreende e usos dos referidos compostos
|
TW200908968A
(en)
|
2007-05-29 |
2009-03-01 |
Sgx Pharmaceuticals Inc |
Substituted pyrrolopyridines and pyrazolopyridines as kinase modulators
|
DE102007028515A1
(de)
|
2007-06-21 |
2008-12-24 |
Merck Patent Gmbh |
6-(Pyrrolopyridinyl)-pyrimidinyl-2-amin-derivate
|
WO2009000319A1
(fr)
|
2007-06-22 |
2008-12-31 |
Schulz Hans M |
Dispositif d'entrée manuel
|
US20100186098A1
(en)
|
2007-06-27 |
2010-07-22 |
Cornell University |
Transgenic animal models of parkinson's disease
|
WO2009030270A1
(fr)
|
2007-09-03 |
2009-03-12 |
Novartis Ag |
Dérivés dhydroindoles utilisés pour traiter la maladie de parkinson
|
US8288383B2
(en)
|
2007-09-14 |
2012-10-16 |
Sanofi |
3-methyl-2- ( (2S) -2- (4- (3-methyl-L, 2, 4-oxadiazol-5-YL) phenyl) morpholino) -6- (pyrim-idin-4-yl) pyrimidin-4 (3H) -one as tau protein kinase inhibitor
|
US20090118276A1
(en)
|
2007-11-02 |
2009-05-07 |
Wyeth |
Thienopyrimidines, thienopyridines, and pyrrolopyrimidines as b-raf inhibitors
|
ATE535241T1
(de)
|
2007-12-05 |
2011-12-15 |
Univ Mainz Johannes Gutenberg |
Verwendung von 3-(indolyl)- oder 3-(azaindolyl)-4-arylmaleimid-derivaten bei der behandlung von leukämie
|
WO2009127642A2
(fr)
|
2008-04-15 |
2009-10-22 |
Cellzome Limited |
Utilisation d’inhibiteurs de lrrk2 pour maladies neurodégénératives
|
AU2009238590A1
(en)
|
2008-04-22 |
2009-10-29 |
Portola Pharmaceuticals, Inc. |
Inhibitors of protein kinases
|
CA2722220C
(fr)
|
2008-04-30 |
2016-06-07 |
National Health Research Institutes |
Composes de pyrimidine bicycliques fusionnes en tant qu'inhibiteurs d'aurora kinase
|
DE102008025751A1
(de)
|
2008-05-29 |
2009-12-03 |
Merck Patent Gmbh |
4-(1H-Pyrrolo[2,3-b]pyridin-3-yl)-pyridin-2-ylamin-derivate
|
AR072008A1
(es)
|
2008-06-13 |
2010-07-28 |
Merck & Co Inc |
Compuestos heterobiciclicos como agentes de inhibicion de quinasa p38
|
DE102008031517A1
(de)
|
2008-07-03 |
2010-01-07 |
Merck Patent Gmbh |
Pyrrolopyridinyl-pyrimidin-2-yl-amin-derivate
|
US20110201599A1
(en)
|
2008-07-03 |
2011-08-18 |
Exelixis, Inc. |
CDK Modulators
|
DE102008038221A1
(de)
|
2008-08-18 |
2010-02-25 |
Merck Patent Gmbh |
7-Azaindolderivate
|
FR2935712A1
(fr)
|
2008-09-05 |
2010-03-12 |
Ct Hospitalier Regional Univer |
Methode de detection de l'expression differentielle d'un ensemble de marqueurs moleculaires associee a la maladie de parkinson
|
GB2463656B
(en)
|
2008-09-18 |
2010-10-13 |
Medical Res Council |
Substrate of LRRK2 and methods of assessing LRRK2 activity
|
EP2346508B1
(fr)
|
2008-09-26 |
2016-08-24 |
Intellikine, LLC |
Inhibiteurs hétérocycliques de kinases
|
US20100175140A1
(en)
|
2008-12-19 |
2010-07-08 |
The Johns Hopkins University |
Leucine-rich repeat kinase (LRRK2) drosophila model for parkinson's disease: wildtype1 (WT1) and G2019S mutant flies
|
EP3828185A3
(fr)
|
2009-01-06 |
2021-09-01 |
Dana Farber Cancer Institute, Inc. |
Composés d'échafaudage de kinase pyrimido-diazépinone et procédés de traitement de troubles
|
EP2210887A1
(fr)
|
2009-01-14 |
2010-07-28 |
Isdin, S.A. |
Dérivés de bis-résorcinyl triazine en tant qu'agents de protection contre le rayonnement UV
|
WO2010085799A2
(fr)
|
2009-01-26 |
2010-07-29 |
Tautatis, Inc. |
Compositions et méthode pour le traitement de la maladie de parkinson
|
WO2010093191A2
(fr)
|
2009-02-13 |
2010-08-19 |
Lg Life Sciences Ltd. |
Nouveaux composés efficaces en tant qu'inhibiteurs de xanthine oxydase, leur procédé de préparation et composition pharmaceutique les contenant
|
JP5732036B2
(ja)
*
|
2009-03-19 |
2015-06-10 |
メディカル リサーチ カウンシル テクノロジーMedical Research Council Technology |
化合物
|
TW201040191A
(en)
|
2009-03-27 |
2010-11-16 |
Abbott Gmbh & Co Kg |
Heterocyclic compounds and their use as glycogen synthase kinase-3 inhibitors
|
KR20100116765A
(ko)
|
2009-04-23 |
2010-11-02 |
인제대학교 산학협력단 |
파킨슨병 치료제 스크리닝 방법
|
WO2010129053A2
(fr)
|
2009-05-05 |
2010-11-11 |
Dana Farber Cancer Institute |
Inhibiteurs d'egfr et procédés de traitement de troubles
|
DE102009019962A1
(de)
|
2009-05-05 |
2010-11-11 |
Merck Patent Gmbh |
3-([1,2,3]Triazol-4-yl)-pyrrolo[2,3-b]pyridinderivate
|
US20120083476A1
(en)
|
2009-06-05 |
2012-04-05 |
Janssen Pharmaceutica Nv |
Heteroaryl-substituted spirocyclic diamine urea modulators of fatty acid amide hydrolase
|
ES2512727T3
(es)
|
2009-09-29 |
2014-10-24 |
Glaxo Group Limited |
Nuevos compuestos
|
FR2951172B1
(fr)
|
2009-10-13 |
2014-09-26 |
Pf Medicament |
Derives pyrazolopyridines en tant qu'agent anticancereux
|
SG10201407012XA
(en)
|
2009-10-29 |
2014-11-27 |
Genosco |
Kinase inhibitors
|
KR20110049217A
(ko)
|
2009-11-04 |
2011-05-12 |
다우어드밴스드디스플레이머티리얼 유한회사 |
신규한 유기 발광 화합물 및 이를 채용하고 있는 유기 전계 발광 소자
|
WO2011057204A2
(fr)
*
|
2009-11-06 |
2011-05-12 |
The Johns Hopkins University |
Toxicité neuronale médiée par lrrk2
|
CN102811619B
(zh)
|
2009-11-13 |
2015-04-22 |
金纳斯克公司 |
激酶抑制剂
|
EP2338486A1
(fr)
|
2009-12-18 |
2011-06-29 |
Johannes Gutenberg-Universität Mainz |
Dérivés de 3-(indolyl)- ou de 3-(azaindolyl)-4-arylmaléimide pour usage dans le traitement de l'adenocarcinome du colon et de l'estomac
|
PT3001903T
(pt)
|
2009-12-21 |
2017-12-18 |
Samumed Llc |
1h-pirazolo[3,4-b]piridinas e usos terapêuticos destas
|
WO2011106168A1
(fr)
|
2010-02-24 |
2011-09-01 |
Dcam Pharma Inc |
Composés de purine pour le traitement de maladies auto-immunes et démyélinisantes
|
US8367349B2
(en)
|
2010-04-19 |
2013-02-05 |
Medical Research Council |
Methods for identifying modulators of LRRK2
|
EP2563125A4
(fr)
|
2010-04-27 |
2013-10-02 |
Merck Sharp & Dohme |
Azaindoles comme inhibiteurs de janus kinase
|
GB201008134D0
(en)
|
2010-05-14 |
2010-06-30 |
Medical Res Council Technology |
Compounds
|
JP5863058B2
(ja)
|
2010-05-17 |
2016-02-16 |
ベーリンガー インゲルハイム インターナショナル ゲゼルシャフト ミット ベシュレンクテル ハフツング |
1H−イミダゾ[4,5−c]キノリン
|
WO2011149827A1
(fr)
|
2010-05-24 |
2011-12-01 |
Glaxosmithkline Llc |
Composés et procédés
|
US9303322B2
(en)
|
2010-05-24 |
2016-04-05 |
Integran Technologies Inc. |
Metallic articles with hydrophobic surfaces
|
CA2797947C
(fr)
|
2010-06-04 |
2019-07-09 |
Charles Baker-Glenn |
Derives d'aminopyrimidine au titre de modulateurs de lrrk2
|
KR101208198B1
(ko)
|
2010-08-27 |
2012-12-04 |
인제대학교 산학협력단 |
Lrrk2 인산화효소 억제 활성을 갖는 화합물을 유효성분으로 함유하는 파킨슨병 치료 또는 예방용 약학조성물
|
AR082827A1
(es)
|
2010-09-02 |
2013-01-09 |
Glaxo Group Ltd |
Compuestos de aril-metiloxi-benzamida, composicion farmaceutica que lo comprende y su uso para la fabricacion de un medicamento util para el tratamiento o la profilaxis de la enfermedad de parkinson
|
EP2616468A4
(fr)
|
2010-09-16 |
2014-02-26 |
Hutchison Medipharma Ltd |
Hétéroaryles condensés et leurs utilisations
|
GB201015949D0
(en)
|
2010-09-22 |
2010-11-03 |
Medical Res Council Technology |
Compounds
|
JP5310700B2
(ja)
|
2010-10-27 |
2013-10-09 |
パナソニック株式会社 |
Ledパッケージ製造システムおよびledパッケージ製造システムにおける樹脂塗布方法
|
WO2012058193A1
(fr)
|
2010-10-29 |
2012-05-03 |
Merck Sharp & Dohme Corp. |
Activité de l'enzyme kinase à répétition riche en leucine
|
ES2653967T3
(es)
|
2010-11-10 |
2018-02-09 |
Genentech, Inc. |
Derivados de pirazol aminopirimidina como moduladores de LRRK2
|
JP2014504362A
(ja)
|
2010-11-30 |
2014-02-20 |
ジェネンテック, インコーポレイテッド |
Lrrk2のためのアッセイ及びバイオマーカー
|
US20130338106A1
(en)
|
2011-02-28 |
2013-12-19 |
John A. McCauley |
Compounds inhibiting leucine-rich repeat kinase enzyme activity
|
US9493452B2
(en)
|
2011-03-24 |
2016-11-15 |
Southern Methodist University |
Compounds and derivatives of 2H-pyrido (3,2-b)(1, 4) oxazin 3)4H)-ones as raf kinase and LRRK2 inhibitors
|
GB201105137D0
(en)
|
2011-03-28 |
2011-05-11 |
Isis Innovation |
Therapeutic molecules for use in the suppression of Parkinson's disease
|
US8791112B2
(en)
|
2011-03-30 |
2014-07-29 |
Arrien Pharmaceuticals Llc |
Substituted 5-(pyrazin-2-yl)-1H-pyrazolo [3, 4-B] pyridine and pyrazolo [3, 4-B] pyridine derivatives as protein kinase inhibitors
|
EA034193B1
(ru)
|
2011-04-21 |
2020-01-15 |
Оригенис Гмбх |
Гетероциклические соединения в качестве ингибиторов киназ
|
SG194549A1
(en)
|
2011-04-21 |
2013-12-30 |
Origenis Gmbh |
Pyrazolo [4, 3-d] pyrimidines useful as kinase inhibitors
|
US9187567B2
(en)
|
2011-05-18 |
2015-11-17 |
Parkinson's Institute |
Assay to determine LRRK2 activity in parkinson's disease
|
EP2726465A1
(fr)
|
2011-05-23 |
2014-05-07 |
Elan Pharmaceuticals Inc. |
Inhibiteurs de l'activité lrrk2 kinase
|
WO2012178015A2
(fr)
|
2011-06-24 |
2012-12-27 |
Zenobia Therapeutics, Inc. |
Inhibiteurs de lrrk2
|
WO2013007768A1
(fr)
|
2011-07-13 |
2013-01-17 |
F. Hoffmann-La Roche Ag |
Composés hétérocycliques tricycliques, compositions et procédés d'utilisation de ces composés comme inhibiteurs des jak
|
CA2850350A1
(fr)
|
2011-09-30 |
2013-04-04 |
Ipsen Pharma S.A.S. |
Inhibiteurs macrocycliques de la kinase lrrk2
|
GB201204985D0
(en)
|
2012-03-21 |
2012-05-02 |
Genentech Inc |
Compounds
|
EP2844660B1
(fr)
|
2012-05-02 |
2017-11-01 |
Southern Research Institute |
Composés de triazolopyridazine, utilisation comme inhibiteurs de la kinase lrrk2, et procédés pour leur préparation
|
EP2844652B1
(fr)
|
2012-05-03 |
2019-03-13 |
Genentech, Inc. |
Dérivés de pyrazole aminopyrimidine en tant que modulateurs de lrrk2
|
KR20150027267A
(ko)
*
|
2012-06-29 |
2015-03-11 |
화이자 인코포레이티드 |
LRRK2 억제제로서의 4-(치환된-아미노)-7H-피롤로[2,3-d]피리미딘
|
WO2014060113A1
(fr)
|
2012-10-19 |
2014-04-24 |
Origenis Gmbh |
Nouveaux inhibiteurs de kinases
|
US9260426B2
(en)
|
2012-12-14 |
2016-02-16 |
Arrien Pharmaceuticals Llc |
Substituted 1H-pyrrolo [2, 3-b] pyridine and 1H-pyrazolo [3, 4-b] pyridine derivatives as salt inducible kinase 2 (SIK2) inhibitors
|
JP6116239B2
(ja)
|
2012-12-28 |
2017-04-19 |
キヤノン株式会社 |
被検体情報取得装置および被検体情報取得方法
|
EP2816840B1
(fr)
|
2013-03-21 |
2017-01-04 |
Huawei Device Co., Ltd. |
Procédé adaptive de transmission avec deux modes d'opération
|
WO2015022664A1
(fr)
|
2013-08-14 |
2015-02-19 |
Novartis Ag |
Composés et compositions utiles comme inhibiteurs de mek
|
WO2015092592A1
(fr)
|
2013-12-17 |
2015-06-25 |
Pfizer Inc. |
Nouvelles 1h-pyrrolo[2,3- b]pyridines 3,4-disubstituées et 7h-pyrrolo[2,3-c]pyridazines 4,5-disubstituées en tant qu'inhibiteurs de la lrrk2
|
CN115068134A
(zh)
|
2014-03-21 |
2022-09-20 |
阿莱恩技术有限公司 |
具有弹性体的分段的正畸矫正器
|