AU2001264313A1 - Pyrazolopyridine compounds and use thereof as drugs - Google Patents

Pyrazolopyridine compounds and use thereof as drugs

Info

Publication number
AU2001264313A1
AU2001264313A1 AU2001264313A AU6431301A AU2001264313A1 AU 2001264313 A1 AU2001264313 A1 AU 2001264313A1 AU 2001264313 A AU2001264313 A AU 2001264313A AU 6431301 A AU6431301 A AU 6431301A AU 2001264313 A1 AU2001264313 A1 AU 2001264313A1
Authority
AU
Australia
Prior art keywords
drugs
pyrazolopyridine compounds
pyrazolopyridine
compounds
Prior art date
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
Abandoned
Application number
AU2001264313A
Inventor
Hisashi Kawasaki
Koichi Ozawa
Kazuhiko Yamamoto
Current Assignee (The listed assignees may be inaccurate. Google has not performed a legal analysis and makes no representation or warranty as to the accuracy of the list.)
Japan Tobacco Inc
Original Assignee
Japan Tobacco Inc
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Priority claimed from JP2000185067A external-priority patent/JP2004123537A/en
Priority claimed from JP2001070593A external-priority patent/JP2004123539A/en
Application filed by Japan Tobacco Inc filed Critical Japan Tobacco Inc
Publication of AU2001264313A1 publication Critical patent/AU2001264313A1/en
Abandoned legal-status Critical Current

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D471/00—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00
    • C07D471/02—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00 in which the condensed system contains two hetero rings
    • C07D471/04—Ortho-condensed systems
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P1/00—Drugs for disorders of the alimentary tract or the digestive system
    • A61P1/16—Drugs for disorders of the alimentary tract or the digestive system for liver or gallbladder disorders, e.g. hepatoprotective agents, cholagogues, litholytics
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P11/00—Drugs for disorders of the respiratory system
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P13/00—Drugs for disorders of the urinary system
    • A61P13/12—Drugs for disorders of the urinary system of the kidneys
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P43/00—Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P9/00—Drugs for disorders of the cardiovascular system
    • A61P9/10—Drugs for disorders of the cardiovascular system for treating ischaemic or atherosclerotic diseases, e.g. antianginal drugs, coronary vasodilators, drugs for myocardial infarction, retinopathy, cerebrovascula insufficiency, renal arteriosclerosis
AU2001264313A 2000-06-20 2001-06-18 Pyrazolopyridine compounds and use thereof as drugs Abandoned AU2001264313A1 (en)

Applications Claiming Priority (5)

Application Number Priority Date Filing Date Title
JP2000185067A JP2004123537A (en) 2000-06-20 2000-06-20 Pyrazolopyridine compound and its pharmaceutical application
JP2000-185067 2000-06-20
JP2001-070593 2001-03-13
JP2001070593A JP2004123539A (en) 2001-03-13 2001-03-13 New pyrazolopyridine compound and medicinal application
PCT/JP2001/005187 WO2001098301A1 (en) 2000-06-20 2001-06-18 Pyrazolopyridine compounds and use thereof as drugs

Publications (1)

Publication Number Publication Date
AU2001264313A1 true AU2001264313A1 (en) 2002-01-02

Family

ID=26594297

Family Applications (1)

Application Number Title Priority Date Filing Date
AU2001264313A Abandoned AU2001264313A1 (en) 2000-06-20 2001-06-18 Pyrazolopyridine compounds and use thereof as drugs

Country Status (2)

Country Link
AU (1) AU2001264313A1 (en)
WO (1) WO2001098301A1 (en)

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EP2308562B1 (en) 2003-12-25 2015-02-25 Ono Pharmaceutical Co., Ltd. Azetidine ring compounds and drugs comprising the same
KR20060114022A (en) 2004-02-27 2006-11-03 에프. 호프만-라 로슈 아게 Indazole derivatives and pharmaceutical compositions containing them
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AU2005219525B2 (en) 2004-02-27 2011-08-18 F. Hoffmann-La Roche Ag Fused derivatives of pyrazole
DK1772145T3 (en) 2004-07-16 2011-05-30 Kyorin Seiyaku Kk Method of effective use of medicine and method of preventing side effects
ES2563034T3 (en) 2004-10-12 2016-03-10 Kyorin Pharmaceutical Co., Ltd. Process for producing 2-amino-2- [2- [4- (3-benzyloxyphenylthio) -2-chlorophenyl] ethyl] -1,3-propanediol hydrochloride and hydrates thereof, and intermediates for the production thereof
CA2620105A1 (en) 2005-08-25 2007-03-01 F. Hoffman-La Roche Ag P38 map kinase inhibitors and methods for using the same
BRPI0617077A2 (en) 2005-10-07 2015-01-06 Kyorin Seiyaku Kk THERAPEUTIC AGENT FOR TREATMENT OF LIVER DISEASES CONTAINING 2-AMINE-1, 3-PROPANEDIOL DERIVATIVE AS ACTIVE INGREDIENT, AND METHOD FOR TREATMENT OF LIVER DISEASES
TWI389683B (en) 2006-02-06 2013-03-21 Kyorin Seiyaku Kk A therapeutic agent for an inflammatory bowel disease or an inflammatory bowel disease treatment using a 2-amino-1,3-propanediol derivative as an active ingredient
CN101460458A (en) 2006-02-15 2009-06-17 阿勒根公司 Indole-3-carboxylic acid amide, ester, thioamide and thiol ester compounds bearing aryl or heteroaryl groups having sphingosine-1-phosphate (S1P) receptor antagonist biological activity
JP2009526863A (en) * 2006-02-15 2009-07-23 アラーガン、インコーポレイテッド Sphingosine-1-phosphate (S1P) receptor antagonists Indole-3-carboxylic acid amide, ester, thioamide and thiol ester compounds having aryl or heteroaryl groups with biological activity
CA2645137A1 (en) 2006-03-07 2007-09-13 James F. Blake Heterobicyclic pyrazole compounds and methods of use
RS53080B (en) 2006-08-08 2014-06-30 Kyorin Pharmaceutical Co. Ltd. Aminophosporic acid ester derivative and s1p receptor modulator containing the same as active ingredient
KR20090041424A (en) 2006-08-08 2009-04-28 교린 세이야꾸 가부시키 가이샤 Aminoalcohol derivative and immunosuppressant containing the same as active ingredient
KR20090101307A (en) 2007-01-11 2009-09-24 알러간, 인코포레이티드 6-substituted indole-3-carboxylic acid amide compounds having sphingosine-1-phosphate (s1p) receptor antagonist biological activity
US8524917B2 (en) 2007-01-11 2013-09-03 Allergan, Inc. 6-substituted indole-3-carboxylic acid amide compounds having sphingosine-1-phosphate (S1P) receptor antagonist biological activity
WO2008154470A1 (en) * 2007-06-08 2008-12-18 University Of Connecticut Nhibitor of the receptor activity of the s1p2 receptor for inhibiting pathological angiogenesis in the eye
WO2009085847A1 (en) 2008-01-03 2009-07-09 Allergan, Inc. Tetrahydroindoles having sphingosine-1-phosphate receptor activity
US20100068200A1 (en) * 2008-09-12 2010-03-18 The University Of Connecticut Methods and Compositions for Inhibiting Atherosclerosis and Vascular Inflammation
GB0908394D0 (en) 2009-05-15 2009-06-24 Univ Leuven Kath Novel viral replication inhibitors
GB0913636D0 (en) 2009-08-05 2009-09-16 Univ Leuven Kath Novel viral replication inhibitors
AU2010300791A1 (en) 2009-09-29 2012-04-19 Allergan, Inc. Condensed ring pyridine compounds as subtype-selective modulators of sphingosine-1-phosphate-2 (S1P2) receptors
WO2011076744A1 (en) * 2009-12-21 2011-06-30 Novartis Ag Disubstituted heteroaryl-fused pyridines
WO2011159864A1 (en) * 2010-06-17 2011-12-22 Bracco Imaging S.P.A. Jte013 analogs and methods of making and using same
CN105859590B (en) 2010-10-12 2018-01-02 日本曹达株式会社 Aryloxy group carbamide compound and noxious organism control agent
AU2011331301A1 (en) 2010-11-15 2013-05-23 Katholieke Universiteit Leuven Antiviral condensed heterocyclic compounds
PL2762466T3 (en) 2011-09-29 2017-09-29 Ono Pharmaceutical Co., Ltd. Phenyl derivative
AU2013240139B2 (en) 2012-03-26 2017-02-23 Arroyo Biosciences L.L.C. Novel sphingosine 1-phosphate receptor antagonists
EP2858501A4 (en) * 2012-05-22 2015-12-09 Merck Sharp & Dohme TrkA KINASE INHIBITORS, COMPOSITIONS AND METHODS THEREOF
ES2637245T3 (en) 2012-06-29 2017-10-11 Pfizer Inc. New 4- (substituted amino) -7H-pyrrolo [2,3-d] pyrimidines as LRRK2 inhibitors
JP6264134B2 (en) 2013-03-26 2018-01-24 小野薬品工業株式会社 Pharmaceuticals containing phenyl derivatives
WO2014157158A1 (en) 2013-03-26 2014-10-02 小野薬品工業株式会社 Phenyl derivative
WO2015092592A1 (en) 2013-12-17 2015-06-25 Pfizer Inc. Novel 3,4-disubstituted-1h-pyrrolo[2,3-b]pyridines and 4,5-disubstituted-7h-pyrrolo[2,3-c]pyridazines as lrrk2 inhibitors
WO2015184541A1 (en) 2014-06-02 2015-12-10 Dalhousie University Treatment of familial exudative vitreoretinopathy through s1pr2 inhibition
AU2016273436B2 (en) * 2015-06-01 2021-01-28 Dalhousie University S1PR2 antagonists and uses therefor
US10487082B2 (en) 2015-06-01 2019-11-26 Dalhousie University S1PR2 antagonists and uses therefor
US10858358B2 (en) 2015-06-01 2020-12-08 Dalhousie University S1PR2 antagonists and uses therefor
CN108137586B (en) 2015-09-14 2021-04-13 辉瑞大药厂 Novel imidazo [4,5-c ] quinoline and imidazo [4,5-c ] [1,5] naphthyridine derivatives as LRRK2 inhibitors
JOP20190024A1 (en) 2016-08-26 2019-02-19 Gilead Sciences Inc Substituted pyrrolizine compounds and uses thereof
WO2019002624A1 (en) * 2017-06-30 2019-01-03 Kleuser, Burkhard Medicaments for treating inflammatory bowel diseases
CN111788204B (en) 2018-02-26 2023-05-05 吉利德科学公司 Substituted pyrrolizine compounds as inhibitors of HBV replication
EP3808176A4 (en) * 2018-05-25 2022-04-13 Kyoto University Method for suppressing freezing damage and composition for preventing freezing damage
WO2023283921A1 (en) * 2021-07-16 2023-01-19 北京深蓝泰医药科技有限公司 Dpd inhibitor, and pharmaceutical composition and use thereof
WO2024077036A1 (en) * 2022-10-07 2024-04-11 Scorpion Therapeutics, Inc. Methods for treating cancer

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US4260614A (en) * 1980-02-08 1981-04-07 E. R. Squibb & Sons, Inc. 4-(2-(1H-Imidazol-1-ylmethyl)-1,3-dioxolan-4-yl)methoxypyrazolo(3,4-b)pyridines
IT1154024B (en) * 1982-09-22 1987-01-21 Lepetit Spa PRIDINICAL DERIVATIVES AND PROCEDURE FOR THEIR PRODUCTION
US4822799A (en) * 1988-01-27 1989-04-18 Sandoz Pharm. Corp. Pyrazolopyridine analogs of mevalonolactone and derivatives thereof useful for inhibiting cholesterol biosynthesis in mammals
US5024999A (en) * 1988-04-26 1991-06-18 Nissan Chemical Industries Ltd. Pyrazolopyridine type mevalonolactones useful as pharmaeuticals
JP3130342B2 (en) * 1991-10-04 2001-01-31 日産化学工業株式会社 Atherosclerotic intimal thickening inhibitor
EP0920866A4 (en) * 1996-08-30 2001-08-22 Welfide Corp Preventives/remedies for muscle tissue degenerations

Also Published As

Publication number Publication date
WO2001098301A1 (en) 2001-12-27

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