SMT201500224B - Derivati purinici per l'uso nel trattamento di malattie allergiche, infiammatorie e infettive - Google Patents

Derivati purinici per l'uso nel trattamento di malattie allergiche, infiammatorie e infettive

Info

Publication number
SMT201500224B
SMT201500224B SM201500224T SM201500224T SMT201500224B SM T201500224 B SMT201500224 B SM T201500224B SM 201500224 T SM201500224 T SM 201500224T SM 201500224 T SM201500224 T SM 201500224T SM T201500224 B SMT201500224 B SM T201500224B
Authority
SM
San Marino
Prior art keywords
allergic
inflammatory
treatment
infectious diseases
purine derivatives
Prior art date
Application number
SM201500224T
Other languages
English (en)
Italian (it)
Inventor
Keith Biggadike
Diane Mary Coe
Xiao Qing Lewell
Charlotte Jane Mitchell
Naimisha Trivedi
Stephen Alan Smith
Original Assignee
Glaxosmithkline Llc
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Family has litigation
First worldwide family litigation filed litigation Critical https://patents.darts-ip.com/?family=41187189&utm_source=google_patent&utm_medium=platform_link&utm_campaign=public_patent_search&patent=SMT201500224(B) "Global patent litigation dataset” by Darts-ip is licensed under a Creative Commons Attribution 4.0 International License.
Application filed by Glaxosmithkline Llc filed Critical Glaxosmithkline Llc
Publication of SMT201500224B publication Critical patent/SMT201500224B/xx

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D473/00—Heterocyclic compounds containing purine ring systems
    • C07D473/02—Heterocyclic compounds containing purine ring systems with oxygen, sulphur, or nitrogen atoms directly attached in positions 2 and 6
    • C07D473/18—Heterocyclic compounds containing purine ring systems with oxygen, sulphur, or nitrogen atoms directly attached in positions 2 and 6 one oxygen and one nitrogen atom, e.g. guanine
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00—Medicinal preparations containing organic active ingredients
    • A61K31/33—Heterocyclic compounds
    • A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/495—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with two or more nitrogen atoms as the only ring heteroatoms, e.g. piperazine or tetrazines
    • A61K31/505—Pyrimidines; Hydrogenated pyrimidines, e.g. trimethoprim
    • A61K31/519—Pyrimidines; Hydrogenated pyrimidines, e.g. trimethoprim ortho- or peri-condensed with heterocyclic rings
    • A61K31/52—Purines, e.g. adenine
    • A61K31/522—Purines, e.g. adenine having oxo groups directly attached to the heterocyclic ring, e.g. hypoxanthine, guanine, acyclovir
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00—Medicinal preparations containing organic active ingredients
    • A61K31/33—Heterocyclic compounds
    • A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/55—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having seven-membered rings, e.g. azelastine, pentylenetetrazole
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K45/00—Medicinal preparations containing active ingredients not provided for in groups A61K31/00 - A61K41/00
    • A61K45/06—Mixtures of active ingredients without chemical characterisation, e.g. antiphlogistics and cardiaca
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00—Medicinal preparations characterised by special physical form
    • A61K9/0012—Galenical forms characterised by the site of application
    • A61K9/0043—Nose
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P29/00—Non-central analgesic, antipyretic or antiinflammatory agents, e.g. antirheumatic agents; Non-steroidal antiinflammatory drugs [NSAID]
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P35/00—Antineoplastic agents
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P37/00—Drugs for immunological or allergic disorders
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D473/00—Heterocyclic compounds containing purine ring systems
    • C07D473/02—Heterocyclic compounds containing purine ring systems with oxygen, sulphur, or nitrogen atoms directly attached in positions 2 and 6
    • C07D473/16—Heterocyclic compounds containing purine ring systems with oxygen, sulphur, or nitrogen atoms directly attached in positions 2 and 6 two nitrogen atoms

Landscapes

  • Health & Medical Sciences (AREA)
  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Veterinary Medicine (AREA)
  • Medicinal Chemistry (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • General Health & Medical Sciences (AREA)
  • Public Health (AREA)
  • General Chemical & Material Sciences (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Epidemiology (AREA)
  • Pain & Pain Management (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Immunology (AREA)
  • Communicable Diseases (AREA)
  • Oncology (AREA)
  • Engineering & Computer Science (AREA)
  • Rheumatology (AREA)
  • Otolaryngology (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
  • Medicines Containing Antibodies Or Antigens For Use As Internal Diagnostic Agents (AREA)
  • Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
  • Preparation Of Compounds By Using Micro-Organisms (AREA)
SM201500224T 2008-08-11 2015-09-22 Derivati purinici per l'uso nel trattamento di malattie allergiche, infiammatorie e infettive SMT201500224B (it)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
US8777708P 2008-08-11 2008-08-11
PCT/EP2009/060265 WO2010018133A1 (en) 2008-08-11 2009-08-07 Purine derivatives for use in the treatment of allergic, inflammatory and infectious diseases

Publications (1)

Publication Number Publication Date
SMT201500224B true SMT201500224B (it) 2015-10-30

Family

ID=41187189

Family Applications (1)

Application Number Title Priority Date Filing Date
SM201500224T SMT201500224B (it) 2008-08-11 2015-09-22 Derivati purinici per l'uso nel trattamento di malattie allergiche, infiammatorie e infettive

Country Status (38)

Country Link
US (7) US8067426B2 (ko)
EP (3) EP2324026B1 (ko)
JP (1) JP5529867B2 (ko)
KR (1) KR101669939B1 (ko)
CN (2) CN102177159B (ko)
AU (1) AU2009281197B2 (ko)
BR (1) BRPI0917138A2 (ko)
CA (1) CA2733749C (ko)
CL (1) CL2011000301A1 (ko)
CO (1) CO6351791A2 (ko)
CR (1) CR20110116A (ko)
CY (1) CY1119992T1 (ko)
DK (2) DK2324026T3 (ko)
DO (1) DOP2011000048A (ko)
EA (1) EA020631B1 (ko)
ES (2) ES2661671T3 (ko)
HK (3) HK1157770A1 (ko)
HR (2) HRP20150938T1 (ko)
HU (2) HUE036570T2 (ko)
IL (1) IL210757A (ko)
LT (1) LT3000813T (ko)
MA (1) MA32624B1 (ko)
ME (1) ME02274B (ko)
MX (2) MX2011001666A (ko)
MY (1) MY162538A (ko)
NO (1) NO3000813T3 (ko)
NZ (2) NZ602812A (ko)
PE (1) PE20110674A1 (ko)
PL (2) PL3000813T3 (ko)
PT (2) PT3000813T (ko)
RS (2) RS56984B1 (ko)
SG (1) SG192547A1 (ko)
SI (2) SI2324026T1 (ko)
SM (1) SMT201500224B (ko)
TR (1) TR201802648T4 (ko)
UA (1) UA103195C2 (ko)
WO (1) WO2010018133A1 (ko)
ZA (1) ZA201100845B (ko)

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