HK1253532A1 - 用於治療變應性、炎性和感染性疾病的嘌呤衍生物 - Google Patents

用於治療變應性、炎性和感染性疾病的嘌呤衍生物

Info

Publication number
HK1253532A1
HK1253532A1 HK18112732.8A HK18112732A HK1253532A1 HK 1253532 A1 HK1253532 A1 HK 1253532A1 HK 18112732 A HK18112732 A HK 18112732A HK 1253532 A1 HK1253532 A1 HK 1253532A1
Authority
HK
Hong Kong
Prior art keywords
allergic
inflammatory
treatment
infectious diseases
purine derivatives
Prior art date
Application number
HK18112732.8A
Other languages
English (en)
Inventor
Keith Biggadike
Diane Mary Coe
Xiao Qing Lewell
Charlotte Jane Mitchell
Stephen Allan Smith
Naimisha Trivedi
Original Assignee
Glaxosmithkline Llc
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Family has litigation
First worldwide family litigation filed litigation Critical https://patents.darts-ip.com/?family=41187189&utm_source=google_patent&utm_medium=platform_link&utm_campaign=public_patent_search&patent=HK1253532(A1) "Global patent litigation dataset” by Darts-ip is licensed under a Creative Commons Attribution 4.0 International License.
Application filed by Glaxosmithkline Llc filed Critical Glaxosmithkline Llc
Publication of HK1253532A1 publication Critical patent/HK1253532A1/zh

Links

Classifications

    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00—Medicinal preparations containing organic active ingredients
    • A61K31/33—Heterocyclic compounds
    • A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/495—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with two or more nitrogen atoms as the only ring heteroatoms, e.g. piperazine or tetrazines
    • A61K31/505—Pyrimidines; Hydrogenated pyrimidines, e.g. trimethoprim
    • A61K31/519—Pyrimidines; Hydrogenated pyrimidines, e.g. trimethoprim ortho- or peri-condensed with heterocyclic rings
    • A61K31/52—Purines, e.g. adenine
    • A61K31/522—Purines, e.g. adenine having oxo groups directly attached to the heterocyclic ring, e.g. hypoxanthine, guanine, acyclovir
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00—Medicinal preparations containing organic active ingredients
    • A61K31/33—Heterocyclic compounds
    • A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/55—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having seven-membered rings, e.g. azelastine, pentylenetetrazole
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K45/00—Medicinal preparations containing active ingredients not provided for in groups A61K31/00 - A61K41/00
    • A61K45/06—Mixtures of active ingredients without chemical characterisation, e.g. antiphlogistics and cardiaca
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00—Medicinal preparations characterised by special physical form
    • A61K9/0012—Galenical forms characterised by the site of application
    • A61K9/0043—Nose
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P29/00—Non-central analgesic, antipyretic or antiinflammatory agents, e.g. antirheumatic agents; Non-steroidal antiinflammatory drugs [NSAID]
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P35/00—Antineoplastic agents
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P37/00—Drugs for immunological or allergic disorders
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D473/00—Heterocyclic compounds containing purine ring systems
    • C07D473/02—Heterocyclic compounds containing purine ring systems with oxygen, sulphur, or nitrogen atoms directly attached in positions 2 and 6
    • C07D473/16—Heterocyclic compounds containing purine ring systems with oxygen, sulphur, or nitrogen atoms directly attached in positions 2 and 6 two nitrogen atoms
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D473/00—Heterocyclic compounds containing purine ring systems
    • C07D473/02—Heterocyclic compounds containing purine ring systems with oxygen, sulphur, or nitrogen atoms directly attached in positions 2 and 6
    • C07D473/18—Heterocyclic compounds containing purine ring systems with oxygen, sulphur, or nitrogen atoms directly attached in positions 2 and 6 one oxygen and one nitrogen atom, e.g. guanine

Landscapes

  • Health & Medical Sciences (AREA)
  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Veterinary Medicine (AREA)
  • Public Health (AREA)
  • General Health & Medical Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • Medicinal Chemistry (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • General Chemical & Material Sciences (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Epidemiology (AREA)
  • Pain & Pain Management (AREA)
  • Engineering & Computer Science (AREA)
  • Communicable Diseases (AREA)
  • Oncology (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Immunology (AREA)
  • Rheumatology (AREA)
  • Otolaryngology (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
  • Medicines Containing Antibodies Or Antigens For Use As Internal Diagnostic Agents (AREA)
  • Preparation Of Compounds By Using Micro-Organisms (AREA)
  • Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
HK18112732.8A 2008-08-11 2018-10-05 用於治療變應性、炎性和感染性疾病的嘌呤衍生物 HK1253532A1 (zh)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
US8777708P 2008-08-11 2008-08-11

Publications (1)

Publication Number Publication Date
HK1253532A1 true HK1253532A1 (zh) 2019-06-21

Family

ID=41187189

Family Applications (3)

Application Number Title Priority Date Filing Date
HK11112171.3A HK1157770A1 (zh) 2008-08-11 2011-11-10 用於治療變應性、炎性和感染性疾病的嘌呤衍生物
HK16111100.6A HK1222857A1 (zh) 2008-08-11 2016-09-21 用於治療變應性、炎性和感染性疾病的嘌呤衍生物
HK18112732.8A HK1253532A1 (zh) 2008-08-11 2018-10-05 用於治療變應性、炎性和感染性疾病的嘌呤衍生物

Family Applications Before (2)

Application Number Title Priority Date Filing Date
HK11112171.3A HK1157770A1 (zh) 2008-08-11 2011-11-10 用於治療變應性、炎性和感染性疾病的嘌呤衍生物
HK16111100.6A HK1222857A1 (zh) 2008-08-11 2016-09-21 用於治療變應性、炎性和感染性疾病的嘌呤衍生物

Country Status (38)

Country Link
US (7) US8067426B2 (zh)
EP (3) EP3336089A1 (zh)
JP (1) JP5529867B2 (zh)
KR (1) KR101669939B1 (zh)
CN (2) CN104098568B (zh)
AU (1) AU2009281197B2 (zh)
BR (1) BRPI0917138A2 (zh)
CA (1) CA2733749C (zh)
CL (1) CL2011000301A1 (zh)
CO (1) CO6351791A2 (zh)
CR (1) CR20110116A (zh)
CY (1) CY1119992T1 (zh)
DK (2) DK2324026T3 (zh)
DO (1) DOP2011000048A (zh)
EA (1) EA020631B1 (zh)
ES (2) ES2661671T3 (zh)
HK (3) HK1157770A1 (zh)
HR (2) HRP20150938T1 (zh)
HU (2) HUE036570T2 (zh)
IL (1) IL210757A (zh)
LT (1) LT3000813T (zh)
MA (1) MA32624B1 (zh)
ME (1) ME02274B (zh)
MX (2) MX336345B (zh)
MY (1) MY162538A (zh)
NO (1) NO3000813T3 (zh)
NZ (2) NZ590782A (zh)
PE (1) PE20110674A1 (zh)
PL (2) PL3000813T3 (zh)
PT (2) PT3000813T (zh)
RS (2) RS56984B1 (zh)
SG (1) SG192547A1 (zh)
SI (2) SI2324026T1 (zh)
SM (1) SMT201500224B (zh)
TR (1) TR201802648T4 (zh)
UA (1) UA103195C2 (zh)
WO (1) WO2010018133A1 (zh)
ZA (1) ZA201100845B (zh)

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