SI20848A - Farmacevtska formulacija, ki vsebuje atorvastatin kalcij - Google Patents

Farmacevtska formulacija, ki vsebuje atorvastatin kalcij Download PDF

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Publication number
SI20848A
SI20848A SI200100069A SI200100069A SI20848A SI 20848 A SI20848 A SI 20848A SI 200100069 A SI200100069 A SI 200100069A SI 200100069 A SI200100069 A SI 200100069A SI 20848 A SI20848 A SI 20848A
Authority
SI
Slovenia
Prior art keywords
atorvastatin
pharmaceutical formulation
atorvastatin calcium
amorphous
calcium
Prior art date
Application number
SI200100069A
Other languages
English (en)
Slovenian (sl)
Inventor
Janez Ker
Mateja Salobir
Sa�a Bavec
Original Assignee
Lek, Tovarna Farmacevtskih In Kemijskih Izdelkov, D.D.
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Family has litigation
First worldwide family litigation filed litigation Critical https://patents.darts-ip.com/?family=20432850&utm_source=google_patent&utm_medium=platform_link&utm_campaign=public_patent_search&patent=SI20848(A) "Global patent litigation dataset” by Darts-ip is licensed under a Creative Commons Attribution 4.0 International License.
Application filed by Lek, Tovarna Farmacevtskih In Kemijskih Izdelkov, D.D. filed Critical Lek, Tovarna Farmacevtskih In Kemijskih Izdelkov, D.D.
Priority to SI200100069A priority Critical patent/SI20848A/sl
Priority to IL15753402A priority patent/IL157534A0/xx
Priority to YU69603A priority patent/RS51746B/sr
Priority to MXPA03008340A priority patent/MXPA03008340A/es
Priority to JP2002571032A priority patent/JP4295988B2/ja
Priority to US10/471,906 priority patent/US7030151B2/en
Priority to SK1136-2003A priority patent/SK287925B6/sk
Priority to PL396343A priority patent/PL217835B1/pl
Priority to MEP-2008-845A priority patent/ME00517B/me
Priority to RS20110313A priority patent/RS55021B1/sr
Priority to EP02702654A priority patent/EP1499297B1/en
Priority to CZ2003-2469A priority patent/CZ306128B6/cs
Priority to ES10183122T priority patent/ES2417881T3/es
Priority to CA002440331A priority patent/CA2440331C/en
Priority to BR0207880-5A priority patent/BR0207880A/pt
Priority to EP10183122.0A priority patent/EP2263655B1/en
Priority to RU2003130378/15A priority patent/RU2293555C2/ru
Priority to SI200230945T priority patent/SI1499297T1/sl
Priority to ES02702654T priority patent/ES2361609T3/es
Priority to KR1020037011535A priority patent/KR100905730B1/ko
Priority to PL371919A priority patent/PL211803B1/pl
Priority to AT02702654T priority patent/ATE500818T1/de
Priority to HU0303434A priority patent/HU230213B1/hu
Priority to DE60239425T priority patent/DE60239425D1/de
Priority to UA2003098317A priority patent/UA78201C2/xx
Priority to PCT/IB2002/000736 priority patent/WO2002072073A2/en
Priority to CN028064739A priority patent/CN1630510B/zh
Publication of SI20848A publication Critical patent/SI20848A/sl
Priority to IL157534A priority patent/IL157534A/en
Priority to ZA200306575A priority patent/ZA200306575B/en
Priority to HRP20030726AA priority patent/HRP20030726B1/hr
Priority to BG108175A priority patent/BG66339B1/bg

Links

Classifications

    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00Medicinal preparations characterised by special physical form
    • A61K9/14Particulate form, e.g. powders, Processes for size reducing of pure drugs or the resulting products, Pure drug nanoparticles
    • A61K9/16Agglomerates; Granulates; Microbeadlets ; Microspheres; Pellets; Solid products obtained by spray drying, spray freeze drying, spray congealing,(multiple) emulsion solvent evaporation or extraction
    • A61K9/1605Excipients; Inactive ingredients
    • A61K9/1611Inorganic compounds
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/33Heterocyclic compounds
    • A61K31/395Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/40Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having five-membered rings with one nitrogen as the only ring hetero atom, e.g. sulpiride, succinimide, tolmetin, buflomedil
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00Medicinal preparations characterised by special physical form
    • A61K9/14Particulate form, e.g. powders, Processes for size reducing of pure drugs or the resulting products, Pure drug nanoparticles
    • A61K9/16Agglomerates; Granulates; Microbeadlets ; Microspheres; Pellets; Solid products obtained by spray drying, spray freeze drying, spray congealing,(multiple) emulsion solvent evaporation or extraction
    • A61K9/1605Excipients; Inactive ingredients
    • A61K9/1617Organic compounds, e.g. phospholipids, fats
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P3/00Drugs for disorders of the metabolism
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P3/00Drugs for disorders of the metabolism
    • A61P3/06Antihyperlipidemics
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P43/00Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P7/00Drugs for disorders of the blood or the extracellular fluid
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K47/00Medicinal preparations characterised by the non-active ingredients used, e.g. carriers or inert additives; Targeting or modifying agents chemically bound to the active ingredient
    • A61K47/02Inorganic compounds
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K47/00Medicinal preparations characterised by the non-active ingredients used, e.g. carriers or inert additives; Targeting or modifying agents chemically bound to the active ingredient
    • A61K47/06Organic compounds, e.g. natural or synthetic hydrocarbons, polyolefins, mineral oil, petrolatum or ozokerite
    • A61K47/16Organic compounds, e.g. natural or synthetic hydrocarbons, polyolefins, mineral oil, petrolatum or ozokerite containing nitrogen, e.g. nitro-, nitroso-, azo-compounds, nitriles, cyanates
    • A61K47/18Amines; Amides; Ureas; Quaternary ammonium compounds; Amino acids; Oligopeptides having up to five amino acids
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00Medicinal preparations characterised by special physical form
    • A61K9/14Particulate form, e.g. powders, Processes for size reducing of pure drugs or the resulting products, Pure drug nanoparticles
    • A61K9/16Agglomerates; Granulates; Microbeadlets ; Microspheres; Pellets; Solid products obtained by spray drying, spray freeze drying, spray congealing,(multiple) emulsion solvent evaporation or extraction
    • A61K9/1605Excipients; Inactive ingredients
    • A61K9/1629Organic macromolecular compounds
    • A61K9/1652Polysaccharides, e.g. alginate, cellulose derivatives; Cyclodextrin
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00Medicinal preparations characterised by special physical form
    • A61K9/20Pills, tablets, discs, rods
    • A61K9/2072Pills, tablets, discs, rods characterised by shape, structure or size; Tablets with holes, special break lines or identification marks; Partially coated tablets; Disintegrating flat shaped forms
    • A61K9/2077Tablets comprising drug-containing microparticles in a substantial amount of supporting matrix; Multiparticulate tablets
SI200100069A 2001-03-14 2001-03-14 Farmacevtska formulacija, ki vsebuje atorvastatin kalcij SI20848A (sl)

Priority Applications (31)

Application Number Priority Date Filing Date Title
SI200100069A SI20848A (sl) 2001-03-14 2001-03-14 Farmacevtska formulacija, ki vsebuje atorvastatin kalcij
IL15753402A IL157534A0 (en) 2001-03-14 2002-02-13 Atorvastatin calcium in a pharmaceutical form composition thereof, and pharmaceutical formulation comprising atorvastatin calcium
CN028064739A CN1630510B (zh) 2001-03-14 2002-03-13 药物形式的阿托伐他汀钙、其组合物和包含阿托伐他汀钙的药物制剂
BR0207880-5A BR0207880A (pt) 2001-03-14 2002-03-13 Formulação farmacêutica, processo para preparação da mesma e uso de formulação sólida
SI200230945T SI1499297T1 (sl) 2001-03-14 2002-03-13 Farmacevtska oblika, ki vsebuje atorvastatin kalcij
JP2002571032A JP4295988B2 (ja) 2001-03-14 2002-03-13 医薬形態のアトルバスタチンカルシウム、その構成物、及びアトルバスタチンカルシウムを含む医薬製剤
US10/471,906 US7030151B2 (en) 2001-03-14 2002-03-13 Atorvastatin calcium in a pharmaceutical form composition thereof and pharmaceutical formulation comprising atorvastatin calcium
SK1136-2003A SK287925B6 (sk) 2001-03-14 2002-03-13 Pharmaceutical formulation comprising atorvastatin calcium, method for the preparation and use
PL396343A PL217835B1 (pl) 2001-03-14 2002-03-13 Preparat farmaceutyczny zawierający sól wapniową atorwastatyny, sposób wytwarzania tego preparatu i jego zastosowanie do leczenia hipercholesterolemii i hiperlipidemii
MEP-2008-845A ME00517B (me) 2001-03-14 2002-03-13 Atorvastati kalcijum u farmaceutskom obliku, njegovoj smješi i farmaceutskoj formulaciji, koja sadrži atorvastatin kalcijum
RS20110313A RS55021B1 (sr) 2001-03-14 2002-03-13 Atorvastatin kalcijum u farmaceutskom obliku, njegovoj smeši i farmaceutskoj formulaciji, koja sadrži atorvastatin kalcijum
EP02702654A EP1499297B1 (en) 2001-03-14 2002-03-13 Pharmaceutical formulation comprising atorvastatin calcium
CZ2003-2469A CZ306128B6 (cs) 2001-03-14 2002-03-13 Kalcium-atorvastatin ve farmaceutické formě, prostředky obsahující tuto sloučeninu a farmaceutické přípravky obsahující kalcium-atorvastatin
ES10183122T ES2417881T3 (es) 2001-03-14 2002-03-13 Formulación farmacéutica que comprende atorvastatina cálcica
CA002440331A CA2440331C (en) 2001-03-14 2002-03-13 Atorvastatin calcium in a pharmaceutical form, composition thereof, and pharmaceutical formulation comprising atorvastatin calcium
YU69603A RS51746B (sr) 2001-03-14 2002-03-13 Atorvastatin kalcijum u farmaceutskom obliku, njegovoj smeši i farmaceutskoj formulaciji, koja sadrži atorvastatin kalcijum
EP10183122.0A EP2263655B1 (en) 2001-03-14 2002-03-13 Pharmaceutical formulation comprising atorvastatin calcium
RU2003130378/15A RU2293555C2 (ru) 2001-03-14 2002-03-13 Аторвастатин кальций в фармацевтической форме, его композиция и фармацевтическая рецептура, содержащая аторвастатин кальций
MXPA03008340A MXPA03008340A (es) 2001-03-14 2002-03-13 Calcio de atorvastatina en una forma farmaceutica, su composicion, y formulacion farmaceutica que comprende calcio de atorvastatina.
ES02702654T ES2361609T3 (es) 2001-03-14 2002-03-13 Formulación farmaceútica que comprende atorvastanina cálcica.
KR1020037011535A KR100905730B1 (ko) 2001-03-14 2002-03-13 약제학적 형태의 아토르바스타틴 칼슘, 이의 조성물 및아토르바스타틴 칼슘을 함유하는 약제학적 제형
PL371919A PL211803B1 (pl) 2001-03-14 2002-03-13 Preparat farmaceutyczny zawierający sól wapniową atorwastatyny, sposób wytwarzania tego preparatu i jego zastosowanie do leczenia hipercholesterolemii i hiperlipidemii
AT02702654T ATE500818T1 (de) 2001-03-14 2002-03-13 Kalziumatorvastatin enthaltende arzneiformulierung
HU0303434A HU230213B1 (hu) 2001-03-14 2002-03-13 Atorvasztatin-kalciumot tartalmazó gyógyszerkészítmény
DE60239425T DE60239425D1 (de) 2001-03-14 2002-03-13 Kalziumatorvastatin enthaltende arzneiformulierung
UA2003098317A UA78201C2 (en) 2001-03-14 2002-03-13 Pharmaceutical formulation containing amorphous micronized atorvastatin calcium and method for preparation thereof
PCT/IB2002/000736 WO2002072073A2 (en) 2001-03-14 2002-03-13 Pharmaceutical formulation comprising atorvastatin calcium
IL157534A IL157534A (en) 2001-03-14 2003-08-21 Atorvastatin calcium in a pharmaceutical form, composition thereof and pharmaceutical formulation comprising atorvastatin calcium
ZA200306575A ZA200306575B (en) 2001-03-14 2003-08-22 Atorvastatin calcium in a pharmaceutical form, composition thereof, and pharmaceutical formulation comprising atorvastatin calcium.
HRP20030726AA HRP20030726B1 (hr) 2001-03-14 2003-09-11 Atorvastatin kalcij u farmaceutskom obliku, njegova kompozicija i farmaceutska formulacija koja obuhvaä†a atorvastatin kalcij
BG108175A BG66339B1 (bg) 2001-03-14 2003-09-12 Фармацевтична форма съдържаща калциев аторвастатин

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
SI200100069A SI20848A (sl) 2001-03-14 2001-03-14 Farmacevtska formulacija, ki vsebuje atorvastatin kalcij

Publications (1)

Publication Number Publication Date
SI20848A true SI20848A (sl) 2002-10-31

Family

ID=20432850

Family Applications (2)

Application Number Title Priority Date Filing Date
SI200100069A SI20848A (sl) 2001-03-14 2001-03-14 Farmacevtska formulacija, ki vsebuje atorvastatin kalcij
SI200230945T SI1499297T1 (sl) 2001-03-14 2002-03-13 Farmacevtska oblika, ki vsebuje atorvastatin kalcij

Family Applications After (1)

Application Number Title Priority Date Filing Date
SI200230945T SI1499297T1 (sl) 2001-03-14 2002-03-13 Farmacevtska oblika, ki vsebuje atorvastatin kalcij

Country Status (25)

Country Link
US (1) US7030151B2 (hu)
EP (2) EP2263655B1 (hu)
JP (1) JP4295988B2 (hu)
KR (1) KR100905730B1 (hu)
CN (1) CN1630510B (hu)
AT (1) ATE500818T1 (hu)
BG (1) BG66339B1 (hu)
BR (1) BR0207880A (hu)
CA (1) CA2440331C (hu)
CZ (1) CZ306128B6 (hu)
DE (1) DE60239425D1 (hu)
ES (2) ES2361609T3 (hu)
HR (1) HRP20030726B1 (hu)
HU (1) HU230213B1 (hu)
IL (2) IL157534A0 (hu)
ME (1) ME00517B (hu)
MX (1) MXPA03008340A (hu)
PL (2) PL211803B1 (hu)
RS (2) RS55021B1 (hu)
RU (1) RU2293555C2 (hu)
SI (2) SI20848A (hu)
SK (1) SK287925B6 (hu)
UA (1) UA78201C2 (hu)
WO (1) WO2002072073A2 (hu)
ZA (1) ZA200306575B (hu)

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