RU2003117476A - Аминотиазолы и их применение в качестве антагонистов рецептора аденозина - Google Patents

Аминотиазолы и их применение в качестве антагонистов рецептора аденозина Download PDF

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RU2003117476A
RU2003117476A RU2003117476/04A RU2003117476A RU2003117476A RU 2003117476 A RU2003117476 A RU 2003117476A RU 2003117476/04 A RU2003117476/04 A RU 2003117476/04A RU 2003117476 A RU2003117476 A RU 2003117476A RU 2003117476 A RU2003117476 A RU 2003117476A
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compound
alkyl
hydrogen
phenyl
formula
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RU2003117476/04A
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English (en)
Russian (ru)
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Нейл Джон ПРЕСС (GB)
Нейл Джон ПРЕСС
Роджер Джон ТЕЙЛОР (GB)
Роджер Джон Тейлор
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Новартис АГ (CH)
Новартис Аг
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Publication of RU2003117476A publication Critical patent/RU2003117476A/ru

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    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D231/00—Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings
    • C07D231/02—Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings not condensed with other rings
    • C07D231/10—Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings not condensed with other rings having two or three double bonds between ring members or between ring members and non-ring members
    • C07D231/12—Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings not condensed with other rings having two or three double bonds between ring members or between ring members and non-ring members with only hydrogen atoms, hydrocarbon or substituted hydrocarbon radicals, directly attached to ring carbon atoms
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D417/00—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00
    • C07D417/02—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00 containing two hetero rings
    • C07D417/04—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00 containing two hetero rings directly linked by a ring-member-to-ring-member bond
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    • A61P1/04—Drugs for disorders of the alimentary tract or the digestive system for ulcers, gastritis or reflux esophagitis, e.g. antacids, inhibitors of acid secretion, mucosal protectants
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    • A61P27/14—Decongestants or antiallergics
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    • A61P3/00—Drugs for disorders of the metabolism
    • A61P3/08—Drugs for disorders of the metabolism for glucose homeostasis
    • A61P3/10—Drugs for disorders of the metabolism for glucose homeostasis for hyperglycaemia, e.g. antidiabetics
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    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P9/00—Drugs for disorders of the cardiovascular system
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    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D233/00—Heterocyclic compounds containing 1,3-diazole or hydrogenated 1,3-diazole rings, not condensed with other rings
    • C07D233/54—Heterocyclic compounds containing 1,3-diazole or hydrogenated 1,3-diazole rings, not condensed with other rings having two double bonds between ring members or between ring members and non-ring members
    • C07D233/56—Heterocyclic compounds containing 1,3-diazole or hydrogenated 1,3-diazole rings, not condensed with other rings having two double bonds between ring members or between ring members and non-ring members with only hydrogen atoms or radicals containing only hydrogen and carbon atoms, attached to ring carbon atoms
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D249/00—Heterocyclic compounds containing five-membered rings having three nitrogen atoms as the only ring hetero atoms
    • C07D249/02—Heterocyclic compounds containing five-membered rings having three nitrogen atoms as the only ring hetero atoms not condensed with other rings
    • C07D249/08—1,2,4-Triazoles; Hydrogenated 1,2,4-triazoles

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  • Health & Medical Sciences (AREA)
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  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Engineering & Computer Science (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • General Health & Medical Sciences (AREA)
  • Pulmonology (AREA)
  • Diabetes (AREA)
  • Dermatology (AREA)
  • Ophthalmology & Optometry (AREA)
  • Neurology (AREA)
  • Immunology (AREA)
  • Hematology (AREA)
  • Urology & Nephrology (AREA)
  • Physical Education & Sports Medicine (AREA)
  • Biomedical Technology (AREA)
  • Neurosurgery (AREA)
  • Endocrinology (AREA)
  • Otolaryngology (AREA)
  • Psychiatry (AREA)
  • Emergency Medicine (AREA)
  • Heart & Thoracic Surgery (AREA)
  • Obesity (AREA)
  • Pain & Pain Management (AREA)
  • Rheumatology (AREA)
  • Cardiology (AREA)
  • Hospice & Palliative Care (AREA)
  • Toxicology (AREA)
  • Gastroenterology & Hepatology (AREA)
  • Vascular Medicine (AREA)
  • Orthopedic Medicine & Surgery (AREA)
RU2003117476/04A 2000-11-21 2001-11-19 Аминотиазолы и их применение в качестве антагонистов рецептора аденозина RU2003117476A (ru)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
GB0028383.8 2000-11-21
GBGB0028383.8A GB0028383D0 (en) 2000-11-21 2000-11-21 Organic compounds

Publications (1)

Publication Number Publication Date
RU2003117476A true RU2003117476A (ru) 2005-02-10

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US (1) US7109202B2 (enExample)
EP (1) EP1339711B1 (enExample)
JP (1) JP3973556B2 (enExample)
KR (1) KR20040007412A (enExample)
CN (1) CN1244580C (enExample)
AR (1) AR035371A1 (enExample)
AT (1) ATE300536T1 (enExample)
AU (1) AU2002237221A1 (enExample)
BR (1) BR0115478A (enExample)
CA (1) CA2429442A1 (enExample)
CZ (1) CZ20031393A3 (enExample)
DE (1) DE60112322T2 (enExample)
EC (1) ECSP034611A (enExample)
ES (1) ES2246346T3 (enExample)
GB (1) GB0028383D0 (enExample)
HU (1) HUP0302079A2 (enExample)
IL (1) IL155712A0 (enExample)
MX (1) MXPA03004439A (enExample)
NO (1) NO20032277L (enExample)
NZ (1) NZ525875A (enExample)
PE (1) PE20020580A1 (enExample)
PL (1) PL361842A1 (enExample)
RU (1) RU2003117476A (enExample)
SK (1) SK6032003A3 (enExample)
WO (1) WO2002042298A1 (enExample)
ZA (1) ZA200303721B (enExample)

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