PL219017B1 - Pochodna benzazepiny, zawierająca ją kompozycja oraz jej zastosowanie - Google Patents

Pochodna benzazepiny, zawierająca ją kompozycja oraz jej zastosowanie

Info

Publication number
PL219017B1
PL219017B1 PL391779A PL39177903A PL219017B1 PL 219017 B1 PL219017 B1 PL 219017B1 PL 391779 A PL391779 A PL 391779A PL 39177903 A PL39177903 A PL 39177903A PL 219017 B1 PL219017 B1 PL 219017B1
Authority
PL
Poland
Prior art keywords
benzazepine
tetrahydro
methyl
methoxy
bromo
Prior art date
Application number
PL391779A
Other languages
English (en)
Polish (pl)
Inventor
Jeffrey Smith
Brian Smith
Original Assignee
Arena Pharmaceuticals
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Family has litigation
First worldwide family litigation filed litigation Critical https://patents.darts-ip.com/?family=29255581&utm_source=google_patent&utm_medium=platform_link&utm_campaign=public_patent_search&patent=PL219017(B1) "Global patent litigation dataset” by Darts-ip is licensed under a Creative Commons Attribution 4.0 International License.
Application filed by Arena Pharmaceuticals filed Critical Arena Pharmaceuticals
Publication of PL219017B1 publication Critical patent/PL219017B1/pl

Links

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    • A—HUMAN NECESSITIES
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    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00—Medicinal preparations containing organic active ingredients
    • A61K31/33—Heterocyclic compounds
    • A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/55—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having seven-membered rings, e.g. azelastine, pentylenetetrazole
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    • A—HUMAN NECESSITIES
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    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D223/00—Heterocyclic compounds containing seven-membered rings having one nitrogen atom as the only ring hetero atom
    • C07D223/14—Heterocyclic compounds containing seven-membered rings having one nitrogen atom as the only ring hetero atom condensed with carbocyclic rings or ring systems
    • C07D223/16—Benzazepines; Hydrogenated benzazepines
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D403/00—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, not provided for by group C07D401/00
    • C07D403/02—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, not provided for by group C07D401/00 containing two hetero rings
    • C07D403/04—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, not provided for by group C07D401/00 containing two hetero rings directly linked by a ring-member-to-ring-member bond
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D409/00—Heterocyclic compounds containing two or more hetero rings, at least one ring having sulfur atoms as the only ring hetero atoms
    • C07D409/02—Heterocyclic compounds containing two or more hetero rings, at least one ring having sulfur atoms as the only ring hetero atoms containing two hetero rings
    • C07D409/04—Heterocyclic compounds containing two or more hetero rings, at least one ring having sulfur atoms as the only ring hetero atoms containing two hetero rings directly linked by a ring-member-to-ring-member bond
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D491/00—Heterocyclic compounds containing in the condensed ring system both one or more rings having oxygen atoms as the only ring hetero atoms and one or more rings having nitrogen atoms as the only ring hetero atoms, not provided for by groups C07D451/00 - C07D459/00, C07D463/00, C07D477/00 or C07D489/00
    • C07D491/02—Heterocyclic compounds containing in the condensed ring system both one or more rings having oxygen atoms as the only ring hetero atoms and one or more rings having nitrogen atoms as the only ring hetero atoms, not provided for by groups C07D451/00 - C07D459/00, C07D463/00, C07D477/00 or C07D489/00 in which the condensed system contains two hetero rings
    • C07D491/04—Ortho-condensed systems

Landscapes

  • Health & Medical Sciences (AREA)
  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Animal Behavior & Ethology (AREA)
  • Medicinal Chemistry (AREA)
  • Veterinary Medicine (AREA)
  • Public Health (AREA)
  • General Health & Medical Sciences (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Engineering & Computer Science (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • General Chemical & Material Sciences (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Biomedical Technology (AREA)
  • Neurosurgery (AREA)
  • Neurology (AREA)
  • Diabetes (AREA)
  • Psychiatry (AREA)
  • Ophthalmology & Optometry (AREA)
  • Addiction (AREA)
  • Endocrinology (AREA)
  • Obesity (AREA)
  • Urology & Nephrology (AREA)
  • Pain & Pain Management (AREA)
  • Reproductive Health (AREA)
  • Hematology (AREA)
  • Cardiology (AREA)
  • Heart & Thoracic Surgery (AREA)
  • Epidemiology (AREA)
  • Pulmonology (AREA)
  • Gynecology & Obstetrics (AREA)
  • Vascular Medicine (AREA)
  • Gastroenterology & Hepatology (AREA)
  • Pregnancy & Childbirth (AREA)
  • Anesthesiology (AREA)
  • Emergency Medicine (AREA)
  • Child & Adolescent Psychology (AREA)
  • Hospice & Palliative Care (AREA)
PL391779A 2002-04-12 2003-04-11 Pochodna benzazepiny, zawierająca ją kompozycja oraz jej zastosowanie PL219017B1 (pl)

Applications Claiming Priority (4)

Application Number Priority Date Filing Date Title
US37205802P 2002-04-12 2002-04-12
US40549502P 2002-08-23 2002-08-23
US43460702P 2002-12-18 2002-12-18
US10/410,991 US6953787B2 (en) 2002-04-12 2003-04-10 5HT2C receptor modulators

Publications (1)

Publication Number Publication Date
PL219017B1 true PL219017B1 (pl) 2015-02-27

Family

ID=29255581

Family Applications (4)

Application Number Title Priority Date Filing Date
PL391779A PL219017B1 (pl) 2002-04-12 2003-04-11 Pochodna benzazepiny, zawierająca ją kompozycja oraz jej zastosowanie
PL391780A PL211333B1 (pl) 2002-04-12 2003-04-11 Hydrat lub solwat hydratu lub solwatu pochodnej benzazepiny, jego zastosowanie, zawierająca go kompozycja farmaceutyczna oraz sposób wytwarzania tej kompozycji
PL396873A PL231405B1 (pl) 2002-04-12 2003-04-11 Sposób wytwarzania kompozycji farmaceutycznej 8-chloro-1 -metylo-2,3,4,5-tetrahydro-1H-3- benzazepiny
PL373464A PL211314B1 (pl) 2002-04-12 2003-04-11 Pochodna benzazepiny, jej zastosowanie, zawierająca ją kompozycja farmaceutyczna oraz sposób wytwarzania tej kompozycji

Family Applications After (3)

Application Number Title Priority Date Filing Date
PL391780A PL211333B1 (pl) 2002-04-12 2003-04-11 Hydrat lub solwat hydratu lub solwatu pochodnej benzazepiny, jego zastosowanie, zawierająca go kompozycja farmaceutyczna oraz sposób wytwarzania tej kompozycji
PL396873A PL231405B1 (pl) 2002-04-12 2003-04-11 Sposób wytwarzania kompozycji farmaceutycznej 8-chloro-1 -metylo-2,3,4,5-tetrahydro-1H-3- benzazepiny
PL373464A PL211314B1 (pl) 2002-04-12 2003-04-11 Pochodna benzazepiny, jej zastosowanie, zawierająca ją kompozycja farmaceutyczna oraz sposób wytwarzania tej kompozycji

Country Status (28)

Country Link
US (11) US6953787B2 (enExample)
EP (4) EP1411881B9 (enExample)
JP (5) JP4155926B2 (enExample)
KR (3) KR100812925B1 (enExample)
CN (5) CN101486677B (enExample)
AT (1) ATE294781T1 (enExample)
AU (1) AU2003221866B2 (enExample)
BR (2) BR122017023795B8 (enExample)
CA (1) CA2481723C (enExample)
CR (2) CR7503A (enExample)
DE (1) DE60300610T2 (enExample)
DK (1) DK1411881T3 (enExample)
ES (2) ES2670568T3 (enExample)
GE (1) GEP20074197B (enExample)
IL (1) IL164162A0 (enExample)
IS (1) IS2134B (enExample)
MX (1) MXPA04009965A (enExample)
MY (1) MY141476A (enExample)
NO (1) NO323528B1 (enExample)
NZ (1) NZ535381A (enExample)
PL (4) PL219017B1 (enExample)
PT (1) PT1411881E (enExample)
RU (1) RU2317982C2 (enExample)
SI (1) SI1411881T1 (enExample)
TW (1) TWI252105B (enExample)
UA (1) UA77788C2 (enExample)
WO (1) WO2003086306A2 (enExample)
ZA (1) ZA200408506B (enExample)

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SE0200968D0 (sv) * 2002-03-26 2002-03-26 Lars Baltzer Novel polypeptide scaffolds and use thereof
US6953787B2 (en) * 2002-04-12 2005-10-11 Arena Pharmaceuticals, Inc. 5HT2C receptor modulators
TWI329111B (en) 2002-05-24 2010-08-21 X Ceptor Therapeutics Inc Azepinoindole and pyridoindole derivatives as pharmaceutical agents
US7595311B2 (en) 2002-05-24 2009-09-29 Exelixis, Inc. Azepinoindole derivatives as pharmaceutical agents
ES2333008T3 (es) 2002-12-20 2010-02-16 Glaxo Group Limited Derivados de benzo(d)azepina para el tratamiento de trastornos neurologicos.
MXPA05013364A (es) 2003-06-17 2006-03-17 Arena Pharm Inc Procedimiento para preparar 3-benzazepinas.
AU2004253888B2 (en) * 2003-06-17 2010-11-11 Arena Pharmaceuticals, Inc. Benzazepine derivatives useful for the treatment of 5HT2C receptor associated diseases
TW200510324A (en) * 2003-08-11 2005-03-16 Lilly Co Eli 6-(2,2,2-trifluoroethylamino)-7-chiloro-2, 3, 4, 5-tetrahydro-1h-benzo[d]azepine as a 5-ht2c receptor agonist
WO2005042490A1 (en) * 2003-10-22 2005-05-12 Arena Pharmaceuticals, Inc. Benzazepine derivatives and methods of prophylaxis or treatment of 5ht2c receptor associated diseases
WO2005042491A1 (en) * 2003-10-22 2005-05-12 Arena Pharmaceuticals, Inc. Benzazepine derivatives and methods of prophylaxis or treatment of 5ht2c receptor associated diseases
EP1680127B1 (en) * 2003-10-23 2008-10-15 F. Hoffmann-La Roche Ag Benzazepine derivatives as mao-b inhibitors
CN102311387A (zh) 2004-02-25 2012-01-11 伊莱利利公司 作为5-HT2C受体激动剂的6-取代的2,3,4,5-四氢-1H-苯并[d]氮杂䓬
EP2400300A1 (en) 2004-08-25 2011-12-28 Takeda Pharmaceutical Company Limited Method of screening preventives/remedies for stress urinary incontinence
WO2006028961A2 (en) * 2004-09-03 2006-03-16 Athersys, Inc. Tricyclic heteroaryl piperazines, pyrrolidines and azetidines as serotonin receptor modulators
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