PH11998002606B1 - Crystalline antifungal polymorph - Google Patents
Crystalline antifungal polymorphInfo
- Publication number
- PH11998002606B1 PH11998002606B1 PH11998002606A PH11998002606A PH11998002606B1 PH 11998002606 B1 PH11998002606 B1 PH 11998002606B1 PH 11998002606 A PH11998002606 A PH 11998002606A PH 11998002606 A PH11998002606 A PH 11998002606A PH 11998002606 B1 PH11998002606 B1 PH 11998002606B1
- Authority
- PH
- Philippines
- Prior art keywords
- polymorph
- antifungal
- crystalline
- crystalline antifungal
- antifungal polymorph
- Prior art date
Links
- 230000000843 anti-fungal effect Effects 0.000 title 1
- 229940121375 antifungal agent Drugs 0.000 title 1
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D405/00—Heterocyclic compounds containing both one or more hetero rings having oxygen atoms as the only ring hetero atoms, and one or more rings having nitrogen as the only ring hetero atom
- C07D405/14—Heterocyclic compounds containing both one or more hetero rings having oxygen atoms as the only ring hetero atoms, and one or more rings having nitrogen as the only ring hetero atom containing three or more hetero rings
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
- A61P31/10—Antimycotics
Landscapes
- Chemical & Material Sciences (AREA)
- Organic Chemistry (AREA)
- Health & Medical Sciences (AREA)
- Chemical Kinetics & Catalysis (AREA)
- Life Sciences & Earth Sciences (AREA)
- General Chemical & Material Sciences (AREA)
- Medicinal Chemistry (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- Communicable Diseases (AREA)
- Pharmacology & Pharmacy (AREA)
- Oncology (AREA)
- Animal Behavior & Ethology (AREA)
- General Health & Medical Sciences (AREA)
- Public Health (AREA)
- Veterinary Medicine (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Plural Heterocyclic Compounds (AREA)
- Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
- Agricultural Chemicals And Associated Chemicals (AREA)
Applications Claiming Priority (1)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| US94618397A | 1997-10-07 | 1997-10-07 |
Publications (1)
| Publication Number | Publication Date |
|---|---|
| PH11998002606B1 true PH11998002606B1 (en) | 2006-08-10 |
Family
ID=25484068
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| PH11998002606A PH11998002606B1 (en) | 1997-10-07 | 1998-10-06 | Crystalline antifungal polymorph |
Country Status (30)
| Country | Link |
|---|---|
| EP (1) | EP1021439B1 (enExample) |
| JP (4) | JP2001519346A (enExample) |
| KR (1) | KR100626109B1 (enExample) |
| CN (1) | CN1125067C (enExample) |
| AR (1) | AR015947A1 (enExample) |
| AT (1) | ATE263163T1 (enExample) |
| AU (1) | AU759982B2 (enExample) |
| BR (1) | BR9812866A (enExample) |
| CA (1) | CA2305803C (enExample) |
| CO (1) | CO4970829A1 (enExample) |
| CZ (1) | CZ299835B6 (enExample) |
| DE (1) | DE69822859T2 (enExample) |
| DK (1) | DK1021439T3 (enExample) |
| ES (1) | ES2217594T3 (enExample) |
| HU (1) | HU225233B1 (enExample) |
| ID (1) | ID29290A (enExample) |
| IL (1) | IL135331A (enExample) |
| IN (1) | IN1998CH02232A (enExample) |
| MX (1) | MX225999B (enExample) |
| MY (1) | MY130126A (enExample) |
| NO (1) | NO318827B1 (enExample) |
| NZ (1) | NZ503662A (enExample) |
| PE (1) | PE120499A1 (enExample) |
| PH (1) | PH11998002606B1 (enExample) |
| PL (1) | PL189317B1 (enExample) |
| PT (1) | PT1021439E (enExample) |
| SK (1) | SK285190B6 (enExample) |
| TW (1) | TW589310B (enExample) |
| WO (1) | WO1999018097A1 (enExample) |
| ZA (1) | ZA989063B (enExample) |
Families Citing this family (27)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| EP2130540A1 (en) | 2008-06-02 | 2009-12-09 | Sandoz AG | Pharmaceutical compositions containing a crystalline form of posaconazole |
| EP2141159A1 (en) | 2008-07-03 | 2010-01-06 | Sandoz AG | A Crystalline form of posaconazole |
| EP2451805A1 (en) | 2009-07-09 | 2012-05-16 | Sandoz AG | A crystalline form of posaconazole |
| WO2011144656A1 (en) | 2010-05-19 | 2011-11-24 | Sandoz Ag | Preparation of posaconazole intermediates |
| CA2798010C (en) | 2010-05-19 | 2018-09-25 | Sandoz Ag | Purification of posaconazole and of posaconazole intermediates |
| WO2011144655A1 (en) | 2010-05-19 | 2011-11-24 | Sandoz Ag | Process for the preparation of chiral hydrazides |
| RU2585760C2 (ru) * | 2010-05-19 | 2016-06-10 | Сандоз Аг | Способ получения хиральных триазолонов |
| CN108329303A (zh) | 2011-06-16 | 2018-07-27 | 桑多斯股份公司 | 制备手性化合物的方法 |
| EP2758385B1 (en) * | 2011-09-19 | 2018-03-28 | MSN Laboratories Limited | Process for the preparation of triazole antifungal drug, its intermediates and polymorphs thereof |
| CN105579448B (zh) * | 2013-07-25 | 2018-12-21 | 桑多斯股份公司 | 制备泊沙康唑的晶型iv的改进方法 |
| ITMI20132118A1 (it) * | 2013-12-18 | 2015-06-19 | Djada Pharmaceutical Sa | Una forma cristallina di posaconazolo |
| ITMI20132115A1 (it) * | 2013-12-18 | 2015-06-19 | Djada Pharmaceutical Sa | Una forma cristallina di posaconazolo |
| ITMI20132114A1 (it) * | 2013-12-18 | 2015-06-19 | Djada Pharmaceutical Sa | Una forma cristallina di posaconazolo |
| ITMI20132117A1 (it) * | 2013-12-18 | 2015-06-19 | Djada Pharmaceutical Sa | Una forma cristallina di posaconazolo |
| CN104387374A (zh) * | 2014-10-21 | 2015-03-04 | 江苏恒盛药业有限公司 | 泊沙康唑晶型i的制备工艺 |
| CN104370894A (zh) * | 2014-10-21 | 2015-02-25 | 江苏恒盛药业有限公司 | 无定型泊沙康唑的制备工艺 |
| LT3209647T (lt) | 2014-10-21 | 2020-09-25 | Ariad Pharmaceuticals, Inc. | Kristalinės 5-chlor-n4-[-2-(dimetilfosforil)fenil]-n2-{2-metoksi-4-[4-(4-metilpiperazin-1-il) piperidin-1-il]pirimidin-2,4-diamino formos |
| EP3590505B1 (en) | 2015-08-08 | 2024-11-06 | Alfred E. Tiefenbacher (GmbH & Co. KG) | Gastro-resistant formulation containing posaconazole |
| EA039213B1 (ru) | 2015-12-24 | 2021-12-17 | Такеда Фармасьютикал Компани Лимитед | Сокристалл, способ его получения и лекарственное средство, содержащее сокристалл |
| EP4424308A3 (en) | 2016-02-26 | 2024-12-04 | Alfred E. Tiefenbacher (GmbH & Co. KG) | Gastro-resistant formulation containing posaconazole and a polymeric precipitation inhibitor |
| CN105949278B (zh) * | 2016-03-30 | 2019-12-06 | 南京曼杰生物科技有限公司 | 一种取代的四氢呋喃水溶性衍生物及其应用 |
| WO2017032908A1 (en) | 2016-07-08 | 2017-03-02 | Synthon B.V. | Pharmaceutical composition comprising amorphous posaconazole |
| TR201620462A2 (tr) | 2016-12-31 | 2018-07-23 | Abdi Ibrahim Ilac Sanayi Ve Ticaret Anonim Sirketi | POSAKONAZOL İÇEREN FARMASÖTİK BİLEŞİMLER ve ÜRETİM YÖNTEMİ |
| TR201722493A2 (tr) | 2017-12-28 | 2019-07-22 | Sanovel Ilac Sanayi Ve Ticaret Anonim Sirketi | Posakonazol i̇çeren kati farmasöti̇k kompozi̇syon |
| WO2022034232A1 (en) | 2020-08-13 | 2022-02-17 | Alfred E. Tiefenbacher (Gmbh & Co. Kg) | Gastro-resistant high-strength formulation containing posaconazole |
| WO2023012378A1 (en) | 2021-11-25 | 2023-02-09 | Alfred E. Tiefenbacher (Gmbh Und Co. Kg) | Granules containing posaconazole |
| EP4091604B1 (en) | 2021-11-25 | 2024-04-03 | Alfred E. Tiefenbacher (GmbH & Co. KG) | Granules containing posaconazole |
Family Cites Families (5)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| IL103558A0 (en) * | 1991-10-30 | 1993-03-15 | Schering Corp | Tri-substituted tetrahydrofuran antifungals |
| AU681753B2 (en) * | 1993-12-21 | 1997-09-04 | Merck Sharp & Dohme Corp. | Tetrahydrofuran antifungals |
| PT741737E (pt) * | 1994-01-24 | 2000-04-28 | Janssen Pharmaceutica Nv | Antifungicos do tipo azole soluveis em agua |
| US5625064A (en) * | 1995-04-19 | 1997-04-29 | Schering Corporation | Process for the preparation of triazolones |
| IL118464A (en) * | 1995-06-02 | 2000-08-13 | Schering Corp | (2R-cis)-4-¬4-¬4-¬4¬¬-5-(2',4 dihalophenyl)-tetrahydro-5-(1-H-1,2,4,triazol-1-yl-methyl)furan-3-yl(methoxy¾phenyl¾-1-piperazinyl¬phenyl2,4,dihydro2¬(5)-1-ethyl-2-(5)hydroxy propyl¾-3H-1,2,4-triazol-3-one and pharmaceutical compositions comprising them |
-
1998
- 1998-10-05 DE DE69822859T patent/DE69822859T2/de not_active Expired - Lifetime
- 1998-10-05 PT PT98951994T patent/PT1021439E/pt unknown
- 1998-10-05 EP EP98951994A patent/EP1021439B1/en not_active Expired - Lifetime
- 1998-10-05 CZ CZ20001264A patent/CZ299835B6/cs not_active IP Right Cessation
- 1998-10-05 CO CO98057733A patent/CO4970829A1/es unknown
- 1998-10-05 BR BR9812866-3A patent/BR9812866A/pt not_active Application Discontinuation
- 1998-10-05 AU AU97803/98A patent/AU759982B2/en not_active Expired
- 1998-10-05 ZA ZA989063A patent/ZA989063B/xx unknown
- 1998-10-05 WO PCT/US1998/020476 patent/WO1999018097A1/en not_active Ceased
- 1998-10-05 IL IL13533198A patent/IL135331A/xx not_active IP Right Cessation
- 1998-10-05 NZ NZ503662A patent/NZ503662A/xx not_active IP Right Cessation
- 1998-10-05 PL PL98339659A patent/PL189317B1/pl unknown
- 1998-10-05 ES ES98951994T patent/ES2217594T3/es not_active Expired - Lifetime
- 1998-10-05 CA CA002305803A patent/CA2305803C/en not_active Expired - Lifetime
- 1998-10-05 DK DK98951994T patent/DK1021439T3/da active
- 1998-10-05 AT AT98951994T patent/ATE263163T1/de active
- 1998-10-05 ID IDW20000632A patent/ID29290A/id unknown
- 1998-10-05 KR KR20007003709A patent/KR100626109B1/ko not_active Expired - Lifetime
- 1998-10-05 HU HU0004899A patent/HU225233B1/hu unknown
- 1998-10-05 CN CN98811886A patent/CN1125067C/zh not_active Expired - Lifetime
- 1998-10-05 AR ARP980104957A patent/AR015947A1/es not_active Application Discontinuation
- 1998-10-05 PE PE1998000942A patent/PE120499A1/es not_active IP Right Cessation
- 1998-10-05 JP JP2000514908A patent/JP2001519346A/ja not_active Withdrawn
- 1998-10-05 SK SK512-2000A patent/SK285190B6/sk not_active IP Right Cessation
- 1998-10-06 PH PH11998002606A patent/PH11998002606B1/en unknown
- 1998-10-06 IN IN2232CH1998 patent/IN1998CH02232A/en unknown
- 1998-10-06 TW TW087116562A patent/TW589310B/zh not_active IP Right Cessation
- 1998-10-06 MY MYPI98004576A patent/MY130126A/en unknown
-
2000
- 2000-04-06 NO NO20001779A patent/NO318827B1/no not_active IP Right Cessation
- 2000-04-06 MX MXPA00003404 patent/MX225999B/es active IP Right Grant
-
2008
- 2008-01-04 JP JP2008000110A patent/JP2008106075A/ja not_active Withdrawn
-
2012
- 2012-05-18 JP JP2012114724A patent/JP2012153729A/ja active Pending
- 2012-05-18 JP JP2012114725A patent/JP2012153730A/ja active Pending
Also Published As
Similar Documents
| Publication | Publication Date | Title |
|---|---|---|
| ZA989063B (en) | Crystalline antifungal polymorph | |
| IL136824A0 (en) | Crystalline teriparatide | |
| GB9715892D0 (en) | Heterocyclic compounds | |
| PL345221A1 (en) | Crystalline efavirenz | |
| GB9706294D0 (en) | Heterocyclic compound | |
| GB9713732D0 (en) | Substituted triazinic compounds | |
| GB9724871D0 (en) | Crystalline fluoran compound | |
| PL336307A1 (en) | Crambescidin compounds | |
| AU9464398A (en) | Novel antifungal compounds | |
| PL327915A1 (en) | Crystalline progestagenes | |
| GB9702978D0 (en) | Compounds | |
| AU9592998A (en) | Crystalline antifungal glycine ester polymorph | |
| GB9721671D0 (en) | Fungicidal compounds | |
| CZ20002208A3 (cs) | Krystalický teriparatid | |
| GB9706309D0 (en) | Heterocyclic compound | |
| GB9712298D0 (en) | Crystallisation | |
| ZA989421B (en) | Heterocyclic compounds | |
| GB9801058D0 (en) | Heterocyclic compounds | |
| GB9702945D0 (en) | Heterocyclic compounds | |
| GB9715734D0 (en) | Heterocyclic compounds | |
| GB9719237D0 (en) | Heterocyclic compounds | |
| GB9716378D0 (en) | Heterocyclic compounds | |
| ZA981177B (en) | Heterocyclic compounds | |
| GB9715735D0 (en) | Heterocyclic compounds | |
| GB9704520D0 (en) | Compounds |