NZ563444A - Pyrrolo(2,3-b)pyridine derivatives as protein kinase inhibitors - Google Patents
Pyrrolo(2,3-b)pyridine derivatives as protein kinase inhibitorsInfo
- Publication number
- NZ563444A NZ563444A NZ563444A NZ56344406A NZ563444A NZ 563444 A NZ563444 A NZ 563444A NZ 563444 A NZ563444 A NZ 563444A NZ 56344406 A NZ56344406 A NZ 56344406A NZ 563444 A NZ563444 A NZ 563444A
- Authority
- NZ
- New Zealand
- Prior art keywords
- optionally substituted
- group
- lower alkyl
- fluoro
- nhc
- Prior art date
Links
- MVXVYAKCVDQRLW-UHFFFAOYSA-N 1h-pyrrolo[2,3-b]pyridine Chemical class C1=CN=C2NC=CC2=C1 MVXVYAKCVDQRLW-UHFFFAOYSA-N 0.000 title description 2
- 229940045988 antineoplastic drug protein kinase inhibitors Drugs 0.000 title 1
- 239000003909 protein kinase inhibitor Substances 0.000 title 1
- 150000001875 compounds Chemical class 0.000 claims abstract description 299
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Classifications
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- A61K31/4353—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom ortho- or peri-condensed with heterocyclic ring systems
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Landscapes
- Health & Medical Sciences (AREA)
- Chemical & Material Sciences (AREA)
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- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Nitrogen Condensed Heterocyclic Rings (AREA)
Applications Claiming Priority (6)
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| US68205105P | 2005-05-17 | 2005-05-17 | |
| US68204205P | 2005-05-17 | 2005-05-17 | |
| US68206305P | 2005-05-17 | 2005-05-17 | |
| US69275005P | 2005-06-22 | 2005-06-22 | |
| US69296005P | 2005-06-22 | 2005-06-22 | |
| PCT/US2006/018726 WO2007013896A2 (en) | 2005-05-17 | 2006-05-16 | Pyrrol (2,3-b) pyridine derivatives protein kinase inhibitors |
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| NZ563444A true NZ563444A (en) | 2011-04-29 |
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| NZ563444A NZ563444A (en) | 2005-05-17 | 2006-05-16 | Pyrrolo(2,3-b)pyridine derivatives as protein kinase inhibitors |
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| CN1925855B (zh) | 2003-12-19 | 2010-06-16 | 普莱希科公司 | 开发Ret调节剂的化合物和方法 |
| US7498342B2 (en) * | 2004-06-17 | 2009-03-03 | Plexxikon, Inc. | Compounds modulating c-kit activity |
| EP1797881B1 (en) | 2004-09-17 | 2009-04-15 | Eisai R&D Management Co., Ltd. | Medicinal composition with improved stability and reduced gelation properties |
| MX2007014377A (es) * | 2005-05-17 | 2008-02-06 | Plexxikon Inc | Inhibidores de proteina cinasa de derivados de pirrol (2,3-b) piridina. |
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- 2006-05-16 EP EP06813186A patent/EP1885723A2/en not_active Withdrawn
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- 2006-05-16 CA CA002608733A patent/CA2608733A1/en not_active Abandoned
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Also Published As
| Publication number | Publication date |
|---|---|
| WO2007013896A2 (en) | 2007-02-01 |
| US20070032519A1 (en) | 2007-02-08 |
| KR20080027775A (ko) | 2008-03-28 |
| CA2608733A1 (en) | 2007-02-01 |
| EP1885723A2 (en) | 2008-02-13 |
| NO20075992L (no) | 2008-02-13 |
| US7846941B2 (en) | 2010-12-07 |
| MX2007014377A (es) | 2008-02-06 |
| AU2006272951A1 (en) | 2007-02-01 |
| JP2008545652A (ja) | 2008-12-18 |
| CR9591A (es) | 2008-03-26 |
| WO2007013896A3 (en) | 2007-05-31 |
| BRPI0610066A2 (pt) | 2010-05-25 |
| ECSP077985A (es) | 2008-01-23 |
| US20110166174A1 (en) | 2011-07-07 |
| IL187344A0 (en) | 2008-04-13 |
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