NO333722B1 - Farmasoytisk fremstilling omfattende en aktiv bestanddel dispergert pa en matrise - Google Patents
Farmasoytisk fremstilling omfattende en aktiv bestanddel dispergert pa en matrise Download PDFInfo
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- NO333722B1 NO333722B1 NO20032593A NO20032593A NO333722B1 NO 333722 B1 NO333722 B1 NO 333722B1 NO 20032593 A NO20032593 A NO 20032593A NO 20032593 A NO20032593 A NO 20032593A NO 333722 B1 NO333722 B1 NO 333722B1
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- active ingredient
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- 239000011976 maleic acid Substances 0.000 description 1
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- VQHSOMBJVWLPSR-WUJBLJFYSA-N maltitol Chemical compound OC[C@H](O)[C@@H](O)[C@@H]([C@H](O)CO)O[C@H]1O[C@H](CO)[C@@H](O)[C@H](O)[C@H]1O VQHSOMBJVWLPSR-WUJBLJFYSA-N 0.000 description 1
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- 150000007522 mineralic acids Chemical class 0.000 description 1
- 229940043348 myristyl alcohol Drugs 0.000 description 1
- WQEPLUUGTLDZJY-UHFFFAOYSA-N n-Pentadecanoic acid Natural products CCCCCCCCCCCCCCC(O)=O WQEPLUUGTLDZJY-UHFFFAOYSA-N 0.000 description 1
- GOQYKNQRPGWPLP-UHFFFAOYSA-N n-heptadecyl alcohol Natural products CCCCCCCCCCCCCCCCCO GOQYKNQRPGWPLP-UHFFFAOYSA-N 0.000 description 1
- 229910017604 nitric acid Inorganic materials 0.000 description 1
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- WLJNZVDCPSBLRP-UHFFFAOYSA-N pamoic acid Chemical compound C1=CC=C2C(CC=3C4=CC=CC=C4C=C(C=3O)C(=O)O)=C(O)C(C(O)=O)=CC2=C1 WLJNZVDCPSBLRP-UHFFFAOYSA-N 0.000 description 1
- 229940068065 phytosterols Drugs 0.000 description 1
- 229920000136 polysorbate Polymers 0.000 description 1
- 229910052700 potassium Inorganic materials 0.000 description 1
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- 230000002335 preservative effect Effects 0.000 description 1
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- 235000010232 propyl p-hydroxybenzoate Nutrition 0.000 description 1
- QELSKZZBTMNZEB-UHFFFAOYSA-N propylparaben Chemical class CCCOC(=O)C1=CC=C(O)C=C1 QELSKZZBTMNZEB-UHFFFAOYSA-N 0.000 description 1
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- 229940126409 proton pump inhibitor Drugs 0.000 description 1
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- KZJWDPNRJALLNS-VJSFXXLFSA-N sitosterol Chemical compound C1C=C2C[C@@H](O)CC[C@]2(C)[C@@H]2[C@@H]1[C@@H]1CC[C@H]([C@H](C)CC[C@@H](CC)C(C)C)[C@@]1(C)CC2 KZJWDPNRJALLNS-VJSFXXLFSA-N 0.000 description 1
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- HEBKCHPVOIAQTA-SCDXWVJYSA-N xylitol Chemical compound OC[C@H](O)[C@@H](O)[C@H](O)CO HEBKCHPVOIAQTA-SCDXWVJYSA-N 0.000 description 1
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Classifications
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K9/00—Medicinal preparations characterised by special physical form
- A61K9/20—Pills, tablets, discs, rods
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K9/00—Medicinal preparations characterised by special physical form
- A61K9/20—Pills, tablets, discs, rods
- A61K9/2072—Pills, tablets, discs, rods characterised by shape, structure or size; Tablets with holes, special break lines or identification marks; Partially coated tablets; Disintegrating flat shaped forms
- A61K9/2077—Tablets comprising drug-containing microparticles in a substantial amount of supporting matrix; Multiparticulate tablets
- A61K9/2081—Tablets comprising drug-containing microparticles in a substantial amount of supporting matrix; Multiparticulate tablets with microcapsules or coated microparticles according to A61K9/50
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/33—Heterocyclic compounds
- A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
- A61K31/435—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom
- A61K31/44—Non condensed pyridines; Hydrogenated derivatives thereof
- A61K31/4427—Non condensed pyridines; Hydrogenated derivatives thereof containing further heterocyclic ring systems
- A61K31/4439—Non condensed pyridines; Hydrogenated derivatives thereof containing further heterocyclic ring systems containing a five-membered ring with nitrogen as a ring hetero atom, e.g. omeprazole
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K9/00—Medicinal preparations characterised by special physical form
- A61K9/14—Particulate form, e.g. powders, Processes for size reducing of pure drugs or the resulting products, Pure drug nanoparticles
- A61K9/16—Agglomerates; Granulates; Microbeadlets ; Microspheres; Pellets; Solid products obtained by spray drying, spray freeze drying, spray congealing,(multiple) emulsion solvent evaporation or extraction
- A61K9/1605—Excipients; Inactive ingredients
- A61K9/1617—Organic compounds, e.g. phospholipids, fats
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K9/00—Medicinal preparations characterised by special physical form
- A61K9/48—Preparations in capsules, e.g. of gelatin, of chocolate
- A61K9/4841—Filling excipients; Inactive ingredients
- A61K9/4858—Organic compounds
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P11/00—Drugs for disorders of the respiratory system
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P37/00—Drugs for immunological or allergic disorders
Landscapes
- Health & Medical Sciences (AREA)
- Life Sciences & Earth Sciences (AREA)
- Animal Behavior & Ethology (AREA)
- Chemical & Material Sciences (AREA)
- Veterinary Medicine (AREA)
- Medicinal Chemistry (AREA)
- Public Health (AREA)
- General Health & Medical Sciences (AREA)
- Pharmacology & Pharmacy (AREA)
- Epidemiology (AREA)
- Engineering & Computer Science (AREA)
- Bioinformatics & Cheminformatics (AREA)
- General Chemical & Material Sciences (AREA)
- Organic Chemistry (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- Chemical Kinetics & Catalysis (AREA)
- Biophysics (AREA)
- Molecular Biology (AREA)
- Pulmonology (AREA)
- Immunology (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Medicinal Preparation (AREA)
- Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
- Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
- Medicines Containing Material From Animals Or Micro-Organisms (AREA)
Applications Claiming Priority (2)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| EP00126847 | 2000-12-07 | ||
| PCT/EP2001/014307 WO2002045693A1 (fr) | 2000-12-07 | 2001-12-06 | Preparation pharmaceutique comprenant un principe actif disperse sur une matrice |
Publications (3)
| Publication Number | Publication Date |
|---|---|
| NO20032593D0 NO20032593D0 (no) | 2003-06-06 |
| NO20032593L NO20032593L (no) | 2003-08-05 |
| NO333722B1 true NO333722B1 (no) | 2013-09-02 |
Family
ID=8170601
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| NO20032593A NO333722B1 (no) | 2000-12-07 | 2003-06-06 | Farmasoytisk fremstilling omfattende en aktiv bestanddel dispergert pa en matrise |
Country Status (28)
| Country | Link |
|---|---|
| US (2) | US7175854B2 (fr) |
| EP (1) | EP1341527B1 (fr) |
| JP (1) | JP4950409B2 (fr) |
| KR (1) | KR20030072557A (fr) |
| CN (2) | CN101810592A (fr) |
| AT (1) | ATE519481T1 (fr) |
| AU (2) | AU2002216073B2 (fr) |
| BR (1) | BR0115987A (fr) |
| CA (1) | CA2430828C (fr) |
| CY (1) | CY1112333T1 (fr) |
| CZ (1) | CZ20031881A3 (fr) |
| DK (1) | DK1341527T3 (fr) |
| EA (1) | EA007151B1 (fr) |
| EE (1) | EE05256B1 (fr) |
| ES (1) | ES2371060T3 (fr) |
| HR (1) | HRP20030493B1 (fr) |
| HU (1) | HUP0400566A3 (fr) |
| IL (2) | IL155964A0 (fr) |
| MX (1) | MXPA03005092A (fr) |
| NO (1) | NO333722B1 (fr) |
| NZ (1) | NZ526015A (fr) |
| PL (1) | PL206595B1 (fr) |
| PT (1) | PT1341527E (fr) |
| SG (1) | SG148028A1 (fr) |
| SI (1) | SI1341527T1 (fr) |
| UA (1) | UA80393C2 (fr) |
| WO (1) | WO2002045693A1 (fr) |
| ZA (1) | ZA200305114B (fr) |
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| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| FR2754177B1 (fr) * | 1996-10-07 | 1999-08-06 | Sanofi Sa | Microspheres pharmaceutiques d'acide valproique pour administration orale |
| KR20030059318A (ko) * | 2000-12-07 | 2003-07-07 | 알타나 파마 아게 | 산 불안정성 활성 성분을 포함하는 현탁액 형태의 약학 제제 |
| SI1341524T1 (sl) * | 2000-12-07 | 2012-02-29 | Nycomed Gmbh | Farmacevtski pripravek v obliki paste, ki obsega kislinsko labilno učinkovino |
| UA80393C2 (uk) * | 2000-12-07 | 2007-09-25 | Алтана Фарма Аг | Фармацевтична композиція, яка містить інгібітор фде 4, диспергований в матриці |
| FR2818552B1 (fr) * | 2000-12-26 | 2003-02-07 | Servier Lab | Compositions pharmaceutique solide thermoformable pour la liberation controlee d'ivabradine |
| AU2002342917A1 (en) * | 2001-11-19 | 2003-06-10 | Altana Pharma Ag | Reversible proton pump inhibitors for the treatment of airway disorders |
| FR2834894B1 (fr) * | 2002-01-21 | 2004-02-27 | Servier Lab | Composition pharmaceutique orodispersible de piribedil |
| FR2834896B1 (fr) * | 2002-01-23 | 2004-02-27 | Servier Lab | Composition pharmaceutique orodispersible d'ivabradine |
| FR2834890B1 (fr) * | 2002-01-23 | 2004-02-27 | Servier Lab | Composition pharmaceutique orodispersible d'agomelatine |
| MY140561A (en) | 2002-02-20 | 2009-12-31 | Nycomed Gmbh | Dosage form containing pde 4 inhibitor as active ingredient |
| ATE344026T1 (de) * | 2002-06-28 | 2006-11-15 | Speedel Pharma Ag | Pharmazeutische formulierung mit einem nichtpeptidischen renin-hemmer und surfactant |
| JP5148813B2 (ja) * | 2002-07-03 | 2013-02-20 | タケダ ファーマシューティカルズ ユー．エス．エー． インコーポレイティド | プロトンポンプ阻害剤の液体剤形 |
| US8877168B1 (en) | 2002-07-31 | 2014-11-04 | Senju Pharmaceuticals Co., Ltd. | Aqueous liquid preparations and light-stabilized aqueous liquid preparations |
| EP1525884B1 (fr) | 2002-07-31 | 2011-10-12 | Senju Pharmaceutical Co., Ltd. | Preparations liquides aqueuses et preparations liquides aqueuses photostabilisees |
| US20080081834A1 (en) | 2002-07-31 | 2008-04-03 | Lippa Arnold S | Methods and compositions employing bicifadine for treating disability or functional impairment associated with acute pain, chronic pain, or neuropathic disorders |
| US20040127541A1 (en) * | 2002-07-31 | 2004-07-01 | Janet Codd | Bicifadine formulation |
| CA2395931A1 (fr) * | 2002-08-07 | 2004-02-07 | Bernard Charles Sherman | Compositions solides comportant du gabapentin et ayant une meilleure stabilite |
| KR20040016202A (ko) * | 2002-08-16 | 2004-02-21 | 주식회사 제이알팜 | 쓴맛이 차폐된 히드로코르티손 경구용 약제 조성물 및 그제조방법 |
| AU2003276688A1 (en) * | 2002-09-02 | 2004-03-19 | Sun Pharmaceutical Industries Limited | Pharmaceutical composition of metaxalone with enhanced oral bioavailability |
| UA80991C2 (en) | 2002-10-07 | 2007-11-26 | Solid preparation containing an insulin resistance improving drug and an active ingredient useful as a remedy for diabetes | |
| US7704527B2 (en) * | 2002-10-25 | 2010-04-27 | Collegium Pharmaceutical, Inc. | Modified release compositions of milnacipran |
| US20060014801A1 (en) * | 2002-11-22 | 2006-01-19 | The Johns Hopkins University | Prevention and treatment of cognitive impairment using (R)-(-)-5-methyl-1-nicotynoyl-2-pyrazoline (MNP) and analogs |
| CA2503290C (fr) | 2003-03-10 | 2012-12-04 | Altana Pharma Ag | Nouveau procede de preparation de roflumilast |
| TW200503783A (en) * | 2003-04-11 | 2005-02-01 | Altana Pharma Ag | Oral pharmaceutical preparation for proton pump antagonists |
| TWI366442B (en) * | 2003-07-30 | 2012-06-21 | Novartis Ag | Palatable ductile chewable veterinary composition |
| US7838029B1 (en) * | 2003-07-31 | 2010-11-23 | Watson Laboratories, Inc. | Mirtazapine solid dosage forms |
| US7390503B1 (en) | 2003-08-22 | 2008-06-24 | Barr Laboratories, Inc. | Ondansetron orally disintegrating tablets |
| CA2545584C (fr) | 2003-11-17 | 2012-10-23 | Biomarin Pharmaceutical Inc. | Methodes et compositions destinees au traitement de troubles metaboliques |
| EP1696881A2 (fr) * | 2003-12-23 | 2006-09-06 | Sun Pharmaceutical Industries Limited | Composition orale stable |
| KR100629771B1 (ko) * | 2004-01-27 | 2006-09-28 | 씨제이 주식회사 | 결정성이 감소되거나 무정형화된 올티프라즈의 제조방법 |
| DE102004011512B4 (de) * | 2004-03-08 | 2022-01-13 | Boehringer Ingelheim Vetmedica Gmbh | Pharmazeutische Zubereitung enthaltend Pimobendan |
| PT1748756E (pt) | 2004-03-10 | 2009-07-20 | Bayer Schering Pharma Ag | Composições compreendendo drospirenona molecularmente dispersa |
| KR100681660B1 (ko) * | 2004-03-17 | 2007-02-09 | 주식회사종근당 | 방출제어 펠릿의 약제학적 조성물 |
| US8980894B2 (en) | 2004-03-25 | 2015-03-17 | Boehringer Ingelheim Vetmedica Gmbh | Use of PDE III inhibitors for the treatment of asymptomatic (occult) heart failure |
| EP1579862A1 (fr) | 2004-03-25 | 2005-09-28 | Boehringer Ingelheim Vetmedica Gmbh | Utilisation des inhibiteurs de PDE III pour la réduction de la taille du coeur chez des mammifères souffrant d'insufficances cardiaques |
| US20110008327A1 (en) | 2004-03-29 | 2011-01-13 | Cheng Jin Q | Compositions including triciribine and epidermal growth factor receptor inhibitor compounds or salts thereof and methods of use thereof |
| US20100009928A1 (en) * | 2004-03-29 | 2010-01-14 | Cheng Jin Q | Compositions including triciribine and taxanes and methods of use thereof |
| US20100173864A1 (en) | 2004-03-29 | 2010-07-08 | Cheng Jin Q | Compositions including triciribine and one or more platinum compounds and methods of use thereof |
| PL2574341T3 (pl) | 2004-03-29 | 2017-09-29 | University Of South Florida | Efektywne leczenie guzów i raka fosforanem tricyrybiny |
| US20100028339A1 (en) | 2004-03-29 | 2010-02-04 | Cheng Jin Q | Compositions including triciribine and trastuzumab and methods of use thereof |
| US20100009929A1 (en) | 2004-03-29 | 2010-01-14 | Cheng Jin Q | Compositions including triciribine and bortezomib and derivatives thereof and methods of use thereof |
| CN100345544C (zh) * | 2004-06-10 | 2007-10-31 | 范敏华 | 一种尼麦角林口腔崩解片剂及其制备方法 |
| PE20060484A1 (es) * | 2004-07-14 | 2006-07-06 | Ucb Farchim Sa | Preparaciones farmaceuticas liquidas que comprenden un compuesto de benzhidril piperizina |
| AU2005291302A1 (en) * | 2004-10-05 | 2006-04-13 | Altana Pharma Ag | Oral pharmaceutical preparation comprising a proton pump antagonist and a basic excipient |
| KR101086254B1 (ko) | 2004-11-04 | 2011-11-24 | 에스케이케미칼주식회사 | 생체이용률이 개선된 프란루카스트 고체분산체 조성물 및그 고체분산체의 제조방법 |
| MX2007005039A (es) * | 2004-11-17 | 2007-06-19 | Biomarin Pharm Inc | Formulacion de tableta estable. |
| DE102005009241A1 (de) * | 2005-03-01 | 2006-09-07 | Bayer Healthcare Ag | Arzneiformen mit kontrollierter Bioverfügbarkeit |
| US20060204588A1 (en) * | 2005-03-10 | 2006-09-14 | Elan Pharma International Limited | Formulations of a nanoparticulate finasteride, dutasteride or tamsulosin hydrochloride, and mixtures thereof |
| CA2601250C (fr) * | 2005-03-16 | 2014-10-28 | Nycomed Gmbh | Forme posologique a gout masque |
| KR100706036B1 (ko) * | 2005-04-04 | 2007-04-11 | 대화제약 주식회사 | 염산 탐술로신 서방성 정제 및 그의 간단한 제조방법 |
| CA2612917A1 (fr) * | 2005-06-23 | 2007-01-04 | Schering Corporation | Formulations orales a absorption rapide d'inhibiteurs de la pde5 |
| CA2614187A1 (fr) * | 2005-07-15 | 2007-01-25 | Bayer Schering Pharma Aktiengesellschaft | Dispositifs d'administration d'un medicament transdermique contenant le drospirenone |
| EP1762179A1 (fr) | 2005-09-07 | 2007-03-14 | Boehringer Ingelheim Vetmedica Gmbh | Méthode pour l'amélioration de la qualité de diagnostic dans l'échocardiographie |
| KR20080056250A (ko) * | 2005-09-29 | 2008-06-20 | 바이엘 헬스케어 아게 | 비뇨기 장애의 치료를 위한 ｐｄｅ 억제제 및 이들의 조합 |
| CN1870631B (zh) * | 2005-11-11 | 2010-04-14 | 华为技术有限公司 | 媒体网关的门控方法 |
| PE20070698A1 (es) * | 2005-11-14 | 2007-08-17 | Teijin Pharma Ltd | Comprimido de disgregacion rapida intraoral que contiene hidrocloruro de ambroxol |
| JP5209492B2 (ja) * | 2005-12-21 | 2013-06-12 | ビーエーエスエフ ソシエタス・ヨーロピア | 速崩性錠剤製造のための医薬製剤 |
| JP2007210905A (ja) * | 2006-02-07 | 2007-08-23 | Asahi Breweries Ltd | 口腔内用顆粒、錠剤およびその製造方法 |
| CN1915233B (zh) * | 2006-08-30 | 2012-10-03 | 四川科瑞德制药有限公司 | 一种治疗焦虑症的药物组合物及其口崩制剂 |
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2001
- 2001-06-12 UA UA2003076286A patent/UA80393C2/uk unknown
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- 2001-12-06 SG SG200503573-8A patent/SG148028A1/en unknown
- 2001-12-06 WO PCT/EP2001/014307 patent/WO2002045693A1/fr active Application Filing
- 2001-12-06 ES ES01999359T patent/ES2371060T3/es not_active Expired - Lifetime
- 2001-12-06 MX MXPA03005092A patent/MXPA03005092A/es active IP Right Grant
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- 2001-12-06 AU AU2002216073A patent/AU2002216073B2/en not_active Ceased
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- 2001-12-06 AT AT01999359T patent/ATE519481T1/de active
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- 2001-12-06 CN CN201010149221A patent/CN101810592A/zh active Pending
- 2001-12-06 BR BR0115987-9A patent/BR0115987A/pt not_active Application Discontinuation
- 2001-12-06 CN CNA018223818A patent/CN1523980A/zh active Pending
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