UA80393C2 - Фармацевтична композиція, яка містить інгібітор фде 4, диспергований в матриці - Google Patents

Фармацевтична композиція, яка містить інгібітор фде 4, диспергований в матриці Download PDF

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Publication number
UA80393C2
UA80393C2 UA2003076286A UA2003076286A UA80393C2 UA 80393 C2 UA80393 C2 UA 80393C2 UA 2003076286 A UA2003076286 A UA 2003076286A UA 2003076286 A UA2003076286 A UA 2003076286A UA 80393 C2 UA80393 C2 UA 80393C2
Authority
UA
Ukraine
Prior art keywords
sodium
acid
composition according
droplets
excipients
Prior art date
Application number
UA2003076286A
Other languages
English (en)
Russian (ru)
Ukrainian (uk)
Inventor
Ранго Дітріх
Рудольф Ліндер
Хартмут Ней
Original Assignee
Алтана Фарма Аг
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Алтана Фарма Аг filed Critical Алтана Фарма Аг
Publication of UA80393C2 publication Critical patent/UA80393C2/uk

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Classifications

    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00Medicinal preparations characterised by special physical form
    • A61K9/20Pills, tablets, discs, rods
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00Medicinal preparations characterised by special physical form
    • A61K9/20Pills, tablets, discs, rods
    • A61K9/2072Pills, tablets, discs, rods characterised by shape, structure or size; Tablets with holes, special break lines or identification marks; Partially coated tablets; Disintegrating flat shaped forms
    • A61K9/2077Tablets comprising drug-containing microparticles in a substantial amount of supporting matrix; Multiparticulate tablets
    • A61K9/2081Tablets comprising drug-containing microparticles in a substantial amount of supporting matrix; Multiparticulate tablets with microcapsules or coated microparticles according to A61K9/50
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/33Heterocyclic compounds
    • A61K31/395Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/435Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom
    • A61K31/44Non condensed pyridines; Hydrogenated derivatives thereof
    • A61K31/4427Non condensed pyridines; Hydrogenated derivatives thereof containing further heterocyclic ring systems
    • A61K31/4439Non condensed pyridines; Hydrogenated derivatives thereof containing further heterocyclic ring systems containing a five-membered ring with nitrogen as a ring hetero atom, e.g. omeprazole
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00Medicinal preparations characterised by special physical form
    • A61K9/14Particulate form, e.g. powders, Processes for size reducing of pure drugs or the resulting products, Pure drug nanoparticles
    • A61K9/16Agglomerates; Granulates; Microbeadlets ; Microspheres; Pellets; Solid products obtained by spray drying, spray freeze drying, spray congealing,(multiple) emulsion solvent evaporation or extraction
    • A61K9/1605Excipients; Inactive ingredients
    • A61K9/1617Organic compounds, e.g. phospholipids, fats
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00Medicinal preparations characterised by special physical form
    • A61K9/48Preparations in capsules, e.g. of gelatin, of chocolate
    • A61K9/4841Filling excipients; Inactive ingredients
    • A61K9/4858Organic compounds
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P11/00Drugs for disorders of the respiratory system
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P37/00Drugs for immunological or allergic disorders

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  • Health & Medical Sciences (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • Chemical & Material Sciences (AREA)
  • Veterinary Medicine (AREA)
  • Medicinal Chemistry (AREA)
  • Public Health (AREA)
  • General Health & Medical Sciences (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Epidemiology (AREA)
  • Engineering & Computer Science (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • General Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Biophysics (AREA)
  • Molecular Biology (AREA)
  • Immunology (AREA)
  • Pulmonology (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Medicinal Preparation (AREA)
  • Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
  • Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
  • Medicines Containing Material From Animals Or Micro-Organisms (AREA)
UA2003076286A 2000-12-07 2001-06-12 Фармацевтична композиція, яка містить інгібітор фде 4, диспергований в матриці UA80393C2 (uk)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
EP00126847 2000-12-07
PCT/EP2001/014307 WO2002045693A1 (fr) 2000-12-07 2001-12-06 Preparation pharmaceutique comprenant un principe actif disperse sur une matrice

Publications (1)

Publication Number Publication Date
UA80393C2 true UA80393C2 (uk) 2007-09-25

Family

ID=8170601

Family Applications (1)

Application Number Title Priority Date Filing Date
UA2003076286A UA80393C2 (uk) 2000-12-07 2001-06-12 Фармацевтична композиція, яка містить інгібітор фде 4, диспергований в матриці

Country Status (28)

Country Link
US (2) US7175854B2 (fr)
EP (1) EP1341527B1 (fr)
JP (1) JP4950409B2 (fr)
KR (1) KR20030072557A (fr)
CN (2) CN1523980A (fr)
AT (1) ATE519481T1 (fr)
AU (2) AU2002216073B2 (fr)
BR (1) BR0115987A (fr)
CA (1) CA2430828C (fr)
CY (1) CY1112333T1 (fr)
CZ (1) CZ20031881A3 (fr)
DK (1) DK1341527T3 (fr)
EA (1) EA007151B1 (fr)
EE (1) EE05256B1 (fr)
ES (1) ES2371060T3 (fr)
HR (1) HRP20030493B1 (fr)
HU (1) HUP0400566A3 (fr)
IL (2) IL155964A0 (fr)
MX (1) MXPA03005092A (fr)
NO (1) NO333722B1 (fr)
NZ (1) NZ526015A (fr)
PL (1) PL206595B1 (fr)
PT (1) PT1341527E (fr)
SG (1) SG148028A1 (fr)
SI (1) SI1341527T1 (fr)
UA (1) UA80393C2 (fr)
WO (1) WO2002045693A1 (fr)
ZA (1) ZA200305114B (fr)

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