NO20090723L - Kondenserte heterosykliske derivater og fremgangsmater for anvendelse - Google Patents

Kondenserte heterosykliske derivater og fremgangsmater for anvendelse

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Publication number
NO20090723L
NO20090723L NO20090723A NO20090723A NO20090723L NO 20090723 L NO20090723 L NO 20090723L NO 20090723 A NO20090723 A NO 20090723A NO 20090723 A NO20090723 A NO 20090723A NO 20090723 L NO20090723 L NO 20090723L
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NO
Norway
Prior art keywords
methods
diseases
condensed heterocyclic
heterocyclic derivatives
compounds
Prior art date
Application number
NO20090723A
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English (en)
Inventor
Steven Bellon
Tae-Seong Kim
Ning Xi
Jean-Christophe Harmange
Kevin Yang
Shon Booker
Deborah Choquette
David Bauer
Alessandro Boezio
Longbin Liu
Brian Albrecht
Christiane Bode
Amico Derin D
Satoko Hirai
Randall Hungate
Richard Lewis
Julia Lohman
Mark Norman
Michele Potashman
Aaron Siegmund
Original Assignee
Usstec Markian
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
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Publication date
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First worldwide family litigation filed litigation Critical https://patents.darts-ip.com/?family=38800918&utm_source=google_patent&utm_medium=platform_link&utm_campaign=public_patent_search&patent=NO20090723(L) "Global patent litigation dataset” by Darts-ip is licensed under a Creative Commons Attribution 4.0 International License.
Application filed by Usstec Markian filed Critical Usstec Markian
Publication of NO20090723L publication Critical patent/NO20090723L/no

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    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D471/00—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00
    • C07D471/02—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00 in which the condensed system contains two hetero rings
    • C07D471/04—Ortho-condensed systems
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00—Medicinal preparations containing organic active ingredients
    • A61K31/33—Heterocyclic compounds
    • A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/435—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom
    • A61K31/4353—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom ortho- or peri-condensed with heterocyclic ring systems
    • A61K31/437—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom ortho- or peri-condensed with heterocyclic ring systems the heterocyclic ring system containing a five-membered ring having nitrogen as a ring hetero atom, e.g. indolizine, beta-carboline
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    • A61P1/00—Drugs for disorders of the alimentary tract or the digestive system
    • A61P1/04—Drugs for disorders of the alimentary tract or the digestive system for ulcers, gastritis or reflux esophagitis, e.g. antacids, inhibitors of acid secretion, mucosal protectants
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    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
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    • A61P1/00—Drugs for disorders of the alimentary tract or the digestive system
    • A61P1/16—Drugs for disorders of the alimentary tract or the digestive system for liver or gallbladder disorders, e.g. hepatoprotective agents, cholagogues, litholytics
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P11/00—Drugs for disorders of the respiratory system
    • A—HUMAN NECESSITIES
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    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P11/00—Drugs for disorders of the respiratory system
    • A61P11/06—Antiasthmatics
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P15/00—Drugs for genital or sexual disorders; Contraceptives
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P17/00—Drugs for dermatological disorders
    • A61P17/02—Drugs for dermatological disorders for treating wounds, ulcers, burns, scars, keloids, or the like
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    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
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    • A61P7/10—Antioedematous agents; Diuretics
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P9/00—Drugs for disorders of the cardiovascular system
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P9/00—Drugs for disorders of the cardiovascular system
    • A61P9/10—Drugs for disorders of the cardiovascular system for treating ischaemic or atherosclerotic diseases, e.g. antianginal drugs, coronary vasodilators, drugs for myocardial infarction, retinopathy, cerebrovascula insufficiency, renal arteriosclerosis
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D487/00—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00
    • C07D487/02—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00 in which the condensed system contains two hetero rings
    • C07D487/04—Ortho-condensed systems

Landscapes

  • Health & Medical Sciences (AREA)
  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Animal Behavior & Ethology (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Veterinary Medicine (AREA)
  • Public Health (AREA)
  • Medicinal Chemistry (AREA)
  • General Health & Medical Sciences (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • General Chemical & Material Sciences (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Engineering & Computer Science (AREA)
  • Immunology (AREA)
  • Ophthalmology & Optometry (AREA)
  • Physical Education & Sports Medicine (AREA)
  • Pulmonology (AREA)
  • Rheumatology (AREA)
  • Hematology (AREA)
  • Orthopedic Medicine & Surgery (AREA)
  • Diabetes (AREA)
  • Dermatology (AREA)
  • Cardiology (AREA)
  • Heart & Thoracic Surgery (AREA)
  • Neurology (AREA)
  • Oncology (AREA)
  • Biomedical Technology (AREA)
  • Endocrinology (AREA)
  • Neurosurgery (AREA)
  • Gastroenterology & Hepatology (AREA)
  • Urology & Nephrology (AREA)
  • Transplantation (AREA)
  • Vascular Medicine (AREA)
  • Pain & Pain Management (AREA)
  • Reproductive Health (AREA)
  • Epidemiology (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Nitrogen Condensed Heterocyclic Rings (AREA)

Abstract

Utvalgte forbindelser er effektive til profylakse og behandling av sykdommer, slik som HGF-formidlede sykdommer. Oppfinnelsen omfatter nye forbindelser, analoger, prolegemidler og farmasøytisk akseptable salter derav, farmasøytiske preparater og fremgangsmåter for profylakse og behandling av sykdommer og andre lidelser eller tilstander som involverer kreft og lignende. Den foreliggende oppfinnelse vedrører også fremgangsmåter for fremstilling av slike forbindelser, samt mellomprodukter som kan anvendes i slike fremgangsmåter.
NO20090723A 2006-07-14 2009-02-13 Kondenserte heterosykliske derivater og fremgangsmater for anvendelse NO20090723L (no)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
US83088206P 2006-07-14 2006-07-14
PCT/US2007/016068 WO2008008539A2 (en) 2006-07-14 2007-07-13 Fused heterocyclic derivatives useful as inhibitors of the hepatocyte growth factor receptor

Publications (1)

Publication Number Publication Date
NO20090723L true NO20090723L (no) 2009-02-13

Family

ID=38800918

Family Applications (2)

Application Number Title Priority Date Filing Date
NO20090723A NO20090723L (no) 2006-07-14 2009-02-13 Kondenserte heterosykliske derivater og fremgangsmater for anvendelse
NO20172002A NO20172002A1 (no) 2006-07-14 2017-12-15 Kondenserte heterosykliske derivater og fremgangsmåter for anvendelse

Family Applications After (1)

Application Number Title Priority Date Filing Date
NO20172002A NO20172002A1 (no) 2006-07-14 2017-12-15 Kondenserte heterosykliske derivater og fremgangsmåter for anvendelse

Country Status (24)

Country Link
US (1) US8212041B2 (no)
EP (3) EP2578583A1 (no)
JP (1) JP5532398B2 (no)
KR (2) KR101140474B1 (no)
CN (1) CN101528743B (no)
AR (1) AR062056A1 (no)
AU (1) AU2007272783B2 (no)
BR (1) BRPI0714387A2 (no)
CA (1) CA2657327A1 (no)
CL (1) CL2007002062A1 (no)
CR (1) CR10614A (no)
DK (1) DK2081931T3 (no)
EA (1) EA016028B1 (no)
ES (1) ES2592888T3 (no)
IL (1) IL196243A (no)
MX (1) MX2009000531A (no)
MY (1) MY167135A (no)
NO (2) NO20090723L (no)
NZ (1) NZ574002A (no)
PE (2) PE20080403A1 (no)
TW (1) TWI394755B (no)
UA (1) UA95965C2 (no)
WO (1) WO2008008539A2 (no)
ZA (1) ZA200900662B (no)

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