NO20003245D0 - <Kappa>-reseptor-opoid-peptider - Google Patents

<Kappa>-reseptor-opoid-peptider

Info

Publication number
NO20003245D0
NO20003245D0 NO20003245A NO20003245A NO20003245D0 NO 20003245 D0 NO20003245 D0 NO 20003245D0 NO 20003245 A NO20003245 A NO 20003245A NO 20003245 A NO20003245 A NO 20003245A NO 20003245 D0 NO20003245 D0 NO 20003245D0
Authority
NO
Norway
Prior art keywords
kappa
opioid peptides
receptor opioid
receptor
peptides
Prior art date
Application number
NO20003245A
Other languages
English (en)
Other versions
NO20003245L (no
NO327080B1 (no
Inventor
Jean Louis Junien
Pierre J M Riviere
Claudio D Schteingart
Javier Sueiras Diaz
Jerzy A Trojnar
Todd W Vanderah
Original Assignee
Ferring Bv
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Ferring Bv filed Critical Ferring Bv
Publication of NO20003245D0 publication Critical patent/NO20003245D0/no
Publication of NO20003245L publication Critical patent/NO20003245L/no
Publication of NO327080B1 publication Critical patent/NO327080B1/no

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07K—PEPTIDES
    • C07K5/00—Peptides containing up to four amino acids in a fully defined sequence; Derivatives thereof
    • C07K5/04—Peptides containing up to four amino acids in a fully defined sequence; Derivatives thereof containing only normal peptide links
    • C07K5/10—Tetrapeptides
    • C07K5/1027—Tetrapeptides containing heteroatoms different from O, S, or N
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P1/00—Drugs for disorders of the alimentary tract or the digestive system
    • A61P1/04—Drugs for disorders of the alimentary tract or the digestive system for ulcers, gastritis or reflux esophagitis, e.g. antacids, inhibitors of acid secretion, mucosal protectants
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P1/00—Drugs for disorders of the alimentary tract or the digestive system
    • A61P1/14—Prodigestives, e.g. acids, enzymes, appetite stimulants, antidyspeptics, tonics, antiflatulents
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P13/00—Drugs for disorders of the urinary system
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P13/00—Drugs for disorders of the urinary system
    • A61P13/10—Drugs for disorders of the urinary system of the bladder
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00—Drugs for disorders of the nervous system
    • A61P25/04—Centrally acting analgesics, e.g. opioids
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P29/00—Non-central analgesic, antipyretic or antiinflammatory agents, e.g. antirheumatic agents; Non-steroidal antiinflammatory drugs [NSAID]
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P37/00—Drugs for immunological or allergic disorders
    • A61P37/02—Immunomodulators
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07K—PEPTIDES
    • C07K5/00—Peptides containing up to four amino acids in a fully defined sequence; Derivatives thereof
    • C07K5/04—Peptides containing up to four amino acids in a fully defined sequence; Derivatives thereof containing only normal peptide links
    • C07K5/10—Tetrapeptides
    • C07K5/1002—Tetrapeptides with the first amino acid being neutral
    • C07K5/1016—Tetrapeptides with the first amino acid being neutral and aromatic or cycloaliphatic
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07K—PEPTIDES
    • C07K5/00—Peptides containing up to four amino acids in a fully defined sequence; Derivatives thereof
    • C07K5/04—Peptides containing up to four amino acids in a fully defined sequence; Derivatives thereof containing only normal peptide links
    • C07K5/10—Tetrapeptides
    • C07K5/1024—Tetrapeptides with the first amino acid being heterocyclic
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K38/00—Medicinal preparations containing peptides

Landscapes

  • Health & Medical Sciences (AREA)
  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Medicinal Chemistry (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • General Health & Medical Sciences (AREA)
  • General Chemical & Material Sciences (AREA)
  • Veterinary Medicine (AREA)
  • Molecular Biology (AREA)
  • Proteomics, Peptides & Aminoacids (AREA)
  • Biophysics (AREA)
  • Genetics & Genomics (AREA)
  • Public Health (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Biochemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Animal Behavior & Ethology (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Engineering & Computer Science (AREA)
  • Immunology (AREA)
  • Urology & Nephrology (AREA)
  • Pain & Pain Management (AREA)
  • Biomedical Technology (AREA)
  • Neurology (AREA)
  • Neurosurgery (AREA)
  • Rheumatology (AREA)
  • Nutrition Science (AREA)
  • Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
  • Peptides Or Proteins (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
NO20003245A 1997-12-23 2000-06-21 Syntetisk opioidpeptidamid samt et farmasoytisk preparat NO327080B1 (no)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
US08/997,208 US5965701A (en) 1997-12-23 1997-12-23 Kappa receptor opioid peptides
PCT/US1998/027282 WO1999032510A1 (en) 1997-12-23 1998-12-22 Kappa receptor opioid peptides

Publications (3)

Publication Number Publication Date
NO20003245D0 true NO20003245D0 (no) 2000-06-21
NO20003245L NO20003245L (no) 2000-08-23
NO327080B1 NO327080B1 (no) 2009-04-20

Family

ID=25543752

Family Applications (1)

Application Number Title Priority Date Filing Date
NO20003245A NO327080B1 (no) 1997-12-23 2000-06-21 Syntetisk opioidpeptidamid samt et farmasoytisk preparat

Country Status (33)

Country Link
US (1) US5965701A (no)
EP (1) EP1042359B1 (no)
JP (1) JP4275852B2 (no)
KR (1) KR100629548B1 (no)
CN (1) CN1154655C (no)
AR (1) AR014167A1 (no)
AT (1) ATE301670T1 (no)
AU (1) AU747806B2 (no)
BR (2) BRPI9814499B8 (no)
CA (1) CA2315878C (no)
CR (1) CR5936A (no)
CZ (1) CZ297281B6 (no)
DE (1) DE69831176T2 (no)
DK (1) DK1042359T3 (no)
EE (1) EE04440B1 (no)
ES (1) ES2247735T3 (no)
HK (1) HK1029349A1 (no)
HR (1) HRP20000415B1 (no)
HU (1) HU227640B1 (no)
IL (3) IL136742A0 (no)
MY (1) MY117542A (no)
NO (1) NO327080B1 (no)
NZ (1) NZ505183A (no)
PL (1) PL195842B1 (no)
PT (1) PT1042359E (no)
RU (1) RU2217437C2 (no)
SK (1) SK286135B6 (no)
TR (1) TR200001985T2 (no)
TW (1) TW580502B (no)
UA (1) UA68366C2 (no)
UY (1) UY25327A1 (no)
WO (1) WO1999032510A1 (no)
ZA (1) ZA9811801B (no)

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US9006175B2 (en) 1999-06-29 2015-04-14 Mannkind Corporation Potentiation of glucose elimination
WO2001036006A1 (en) * 1999-11-19 2001-05-25 Palatin Technologies, Inc. Opioid metallopeptide compositions and methods
DE10116978A1 (de) * 2001-04-05 2002-10-10 Merck Patent Gmbh Kappa-Opiatagonisten für die Behandlung von Erkrankungen der Blase
WO2002089845A1 (en) * 2001-05-08 2002-11-14 Toray Industries, Inc. Remedies for sepsis
ATE385193T1 (de) 2002-03-20 2008-02-15 Mannkind Corp Inhalationsgerät
AU2005277208B2 (en) 2004-08-20 2011-11-24 Mannkind Corporation Catalysis of diketopiperazine synthesis
DK1791542T3 (en) 2004-08-23 2015-06-15 Mannkind Corp Diketopiperazinsalte for pharmaceutical delivery
BRPI0615819B8 (pt) 2005-09-14 2021-05-25 Mannkind Corp processo para preparar uma composição de distribuição de fármaco compreendendo um agente ativo e uma micropartícula fumaril dicetopiperazina cristalina.
CN101389348A (zh) 2006-02-22 2009-03-18 曼金德公司 用于改善包含二酮哌嗪和活性剂的微粒的药物性质的方法
CN101454017A (zh) * 2006-05-26 2009-06-10 卡拉治疗学股份有限公司 提升哺乳动物催乳素的方法
CN101454338A (zh) * 2006-05-26 2009-06-10 卡拉治疗学股份有限公司 κ阿片样受体肽的N-氧化物
US8236766B2 (en) * 2006-11-10 2012-08-07 Cara Therapeutics, Inc. Uses of synthetic peptide amides
MX2009005000A (es) 2006-11-10 2009-10-12 Cara Therapeutics Inc Amidas de peptidos sinteticos.
US7842662B2 (en) * 2006-11-10 2010-11-30 Cara Therapeutics, Inc. Synthetic peptide amide dimers
US7713937B2 (en) * 2006-11-10 2010-05-11 Cara Therapeutics, Inc. Synthetic peptide amides and dimeric forms thereof
US8906859B2 (en) * 2006-11-10 2014-12-09 Cera Therapeutics, Inc. Uses of kappa opioid synthetic peptide amides
WO2008077194A1 (en) * 2006-12-22 2008-07-03 Xenome Ltd Receptor agonists
US8485180B2 (en) 2008-06-13 2013-07-16 Mannkind Corporation Dry powder drug delivery system
CA3086027C (en) 2008-06-13 2022-05-17 Mannkind Corporation A dry powder inhaler and system for drug delivery
MX2010014240A (es) 2008-06-20 2011-03-25 Mankind Corp Un metodo y aparato interactivo para perfilar en tiempo real esfuerzos de inhalacion.
TWI532497B (zh) 2008-08-11 2016-05-11 曼凱公司 超快起作用胰島素之用途
US8314106B2 (en) 2008-12-29 2012-11-20 Mannkind Corporation Substituted diketopiperazine analogs for use as drug delivery agents
DK2405963T3 (da) 2009-03-11 2013-12-16 Mannkind Corp Apparat, system og fremgangsmåde til at måle modstand i en inhalator
WO2010144789A2 (en) 2009-06-12 2010-12-16 Mannkind Corporation Diketopiperazine microparticles with defined specific surface areas
WO2011056889A1 (en) 2009-11-03 2011-05-12 Mannkind Corporation An apparatus and method for simulating inhalation efforts
KR20130117755A (ko) 2010-06-21 2013-10-28 맨카인드 코포레이션 건조 분말 약물 운반 시스템 및 방법
WO2012135765A2 (en) 2011-04-01 2012-10-04 Mannkind Corporation Blister package for pharmaceutical cartridges
WO2012174472A1 (en) 2011-06-17 2012-12-20 Mannkind Corporation High capacity diketopiperazine microparticles
MX2014004983A (es) * 2011-10-24 2014-09-22 Mannkid Corp Metodos y composiciones para tratar dolor.
CN104619369B (zh) 2012-07-12 2018-01-30 曼金德公司 干粉药物输送系统和方法
EP2911690A1 (en) 2012-10-26 2015-09-02 MannKind Corporation Inhalable influenza vaccine compositions and methods
WO2014144895A1 (en) 2013-03-15 2014-09-18 Mannkind Corporation Microcrystalline diketopiperazine compositions and methods
JP6491658B2 (ja) 2013-07-18 2019-03-27 マンカインド コーポレイション 熱安定性乾燥粉末医薬組成物及び方法
US11446127B2 (en) 2013-08-05 2022-09-20 Mannkind Corporation Insufflation apparatus and methods
WO2015148905A1 (en) 2014-03-28 2015-10-01 Mannkind Corporation Use of ultrarapid acting insulin
EP3162810B1 (en) * 2014-06-26 2019-02-13 Maruishi Pharmaceutical Co., Ltd. Method for producing synthetic pentapeptide
US10561806B2 (en) 2014-10-02 2020-02-18 Mannkind Corporation Mouthpiece cover for an inhaler
EP3294315A2 (en) 2015-05-11 2018-03-21 Cadila Healthcare Limited Novel short-chain peptides as kappa opioid receptors (kor) agonist
CN107098876B (zh) * 2016-02-23 2021-04-06 江苏恒瑞医药股份有限公司 苯基丙酰胺类衍生物、其制备方法及其在医药上的应用
EP3521301B1 (en) * 2016-09-27 2024-03-06 Sichuan Kelun-Biotech Biopharmaceutical Co., Ltd. Polyamide compound and use thereof
KR102375543B1 (ko) * 2017-07-21 2022-03-16 스촨 하이스코 파마수티컬 씨오., 엘티디 펩티드 아미드류 화합물 및 이의 제조 방법과 의약에서의 용도
TWI717664B (zh) 2017-12-06 2021-02-01 大陸商江蘇恒瑞醫藥股份有限公司 一種苯基丙醯胺類衍生物的鹽及其製備方法
BR112020023038A2 (pt) 2018-05-16 2021-02-02 Jiangsu Hengrui Medicine Co., Ltd. composição farmacêutica de agonista receptor kor
WO2021013085A1 (zh) * 2019-07-25 2021-01-28 四川海思科制药有限公司 一种肽酰胺盐及其制备方法和在医药上的用途
CN114127086B (zh) * 2019-07-25 2023-10-20 四川海思科制药有限公司 氘代肽酰胺类化合物及其制备方法和在医药上的用途
CN114615976A (zh) * 2019-08-07 2022-06-10 人福医药美国公司 κ阿片受体肽酰胺激动剂
US11492374B2 (en) 2020-06-25 2022-11-08 Humanwell Pharmaceutical US Peptides for treatment of medical disorders
TW202317533A (zh) 2021-07-02 2023-05-01 美商雅斯治療公司 奧沙奈坦(osanetant)之固體形式

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GB2013689B (en) * 1977-12-15 1982-03-24 Reckitt & Colmann Prod Ltd Compounds
GB8801304D0 (en) * 1988-01-21 1988-02-17 Ici Plc Diamine compounds
US5367053A (en) * 1993-05-19 1994-11-22 Houghten Pharmaceuticals, Inc. Opioid peptide inhibitors
US5610271A (en) * 1995-06-07 1997-03-11 Torrey Pines Institute For Molecular Studies Kappa receptor selective opioid peptides

Also Published As

Publication number Publication date
HUP0100626A3 (en) 2001-12-28
ZA9811801B (en) 1999-06-22
WO1999032510A9 (en) 1999-09-23
TW580502B (en) 2004-03-21
BR9814499A (pt) 2000-10-10
KR100629548B1 (ko) 2006-09-27
UA68366C2 (en) 2004-08-16
PL195842B1 (pl) 2007-10-31
CZ20002382A3 (cs) 2000-12-13
ES2247735T3 (es) 2006-03-01
AU747806B2 (en) 2002-05-23
RU2217437C2 (ru) 2003-11-27
JP2001526295A (ja) 2001-12-18
EE04440B1 (et) 2005-02-15
CN1283201A (zh) 2001-02-07
WO1999032510A1 (en) 1999-07-01
NO20003245L (no) 2000-08-23
DE69831176D1 (de) 2005-09-15
SK9602000A3 (en) 2001-01-18
HU227640B1 (en) 2011-10-28
EP1042359A1 (en) 2000-10-11
IL178471A0 (en) 2007-02-11
HRP20000415B1 (en) 2004-06-30
IL136742A0 (en) 2001-06-14
HRP20000415A2 (en) 2000-12-31
NO327080B1 (no) 2009-04-20
PL341308A1 (en) 2001-04-09
TR200001985T2 (tr) 2000-11-21
PT1042359E (pt) 2005-11-30
EE200000370A (et) 2001-10-15
JP4275852B2 (ja) 2009-06-10
ATE301670T1 (de) 2005-08-15
BR9814499B1 (pt) 2014-10-21
KR20010033450A (ko) 2001-04-25
BRPI9814499A (pt) 2000-10-10
IL136742A (en) 2006-12-31
US5965701A (en) 1999-10-12
BRPI9814499B8 (pt) 2021-11-09
SK286135B6 (sk) 2008-04-07
BRPI9814499B1 (pt) 2014-10-21
AU1940299A (en) 1999-07-12
DK1042359T3 (da) 2005-11-28
CR5936A (es) 2006-08-18
CA2315878C (en) 2010-11-16
UY25327A1 (es) 2000-12-29
CN1154655C (zh) 2004-06-23
NZ505183A (en) 2001-09-28
HK1029349A1 (en) 2001-03-30
AR014167A1 (es) 2001-02-07
DE69831176T2 (de) 2006-04-20
EP1042359B1 (en) 2005-08-10
MY117542A (en) 2004-07-31
CZ297281B6 (cs) 2006-10-11
HUP0100626A2 (hu) 2001-08-28
CA2315878A1 (en) 1999-07-01

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Legal Events

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MM1K Lapsed by not paying the annual fees