NL193376C - 16-Ledig pentacyclische macrolideverbindingen, preparaten die deze bevatten en gebruik ervan. - Google Patents
16-Ledig pentacyclische macrolideverbindingen, preparaten die deze bevatten en gebruik ervan. Download PDFInfo
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- NL193376C NL193376C NL8701322A NL8701322A NL193376C NL 193376 C NL193376 C NL 193376C NL 8701322 A NL8701322 A NL 8701322A NL 8701322 A NL8701322 A NL 8701322A NL 193376 C NL193376 C NL 193376C
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- 125000004432 carbon atom Chemical group C* 0.000 claims description 17
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- 238000000034 method Methods 0.000 claims description 12
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- 125000003342 alkenyl group Chemical group 0.000 claims description 4
- 125000001495 ethyl group Chemical group [H]C([H])([H])C([H])([H])* 0.000 claims description 4
- 238000003898 horticulture Methods 0.000 claims description 4
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Classifications
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- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D493/00—Heterocyclic compounds containing oxygen atoms as the only ring hetero atoms in the condensed system
- C07D493/22—Heterocyclic compounds containing oxygen atoms as the only ring hetero atoms in the condensed system in which the condensed system contains four or more hetero rings
-
- A—HUMAN NECESSITIES
- A01—AGRICULTURE; FORESTRY; ANIMAL HUSBANDRY; HUNTING; TRAPPING; FISHING
- A01N—PRESERVATION OF BODIES OF HUMANS OR ANIMALS OR PLANTS OR PARTS THEREOF; BIOCIDES, e.g. AS DISINFECTANTS, AS PESTICIDES OR AS HERBICIDES; PEST REPELLANTS OR ATTRACTANTS; PLANT GROWTH REGULATORS
- A01N43/00—Biocides, pest repellants or attractants, or plant growth regulators containing heterocyclic compounds
- A01N43/90—Biocides, pest repellants or attractants, or plant growth regulators containing heterocyclic compounds having two or more relevant hetero rings, condensed among themselves or with a common carbocyclic ring system
-
- A—HUMAN NECESSITIES
- A01—AGRICULTURE; FORESTRY; ANIMAL HUSBANDRY; HUNTING; TRAPPING; FISHING
- A01N—PRESERVATION OF BODIES OF HUMANS OR ANIMALS OR PLANTS OR PARTS THEREOF; BIOCIDES, e.g. AS DISINFECTANTS, AS PESTICIDES OR AS HERBICIDES; PEST REPELLANTS OR ATTRACTANTS; PLANT GROWTH REGULATORS
- A01N49/00—Biocides, pest repellants or attractants, or plant growth regulators, containing compounds containing the group, wherein m+n>=1, both X together may also mean —Y— or a direct carbon-to-carbon bond, and the carbon atoms marked with an asterisk are not part of any ring system other than that which may be formed by the atoms X, the carbon atoms in square brackets being part of any acyclic or cyclic structure, or the group, wherein A means a carbon atom or Y, n>=0, and not more than one of these carbon atoms being a member of the same ring system, e.g. juvenile insect hormones or mimics thereof
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
- A61P31/04—Antibacterial agents
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P33/00—Antiparasitic agents
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07H—SUGARS; DERIVATIVES THEREOF; NUCLEOSIDES; NUCLEOTIDES; NUCLEIC ACIDS
- C07H19/00—Compounds containing a hetero ring sharing one ring hetero atom with a saccharide radical; Nucleosides; Mononucleotides; Anhydro-derivatives thereof
- C07H19/01—Compounds containing a hetero ring sharing one ring hetero atom with a saccharide radical; Nucleosides; Mononucleotides; Anhydro-derivatives thereof sharing oxygen
Landscapes
- Chemical & Material Sciences (AREA)
- Life Sciences & Earth Sciences (AREA)
- Organic Chemistry (AREA)
- Health & Medical Sciences (AREA)
- General Health & Medical Sciences (AREA)
- Engineering & Computer Science (AREA)
- Plant Pathology (AREA)
- Pest Control & Pesticides (AREA)
- Dentistry (AREA)
- Agronomy & Crop Science (AREA)
- Wood Science & Technology (AREA)
- Zoology (AREA)
- Environmental Sciences (AREA)
- Veterinary Medicine (AREA)
- Genetics & Genomics (AREA)
- Insects & Arthropods (AREA)
- Biochemistry (AREA)
- Molecular Biology (AREA)
- Biotechnology (AREA)
- Public Health (AREA)
- Chemical Kinetics & Catalysis (AREA)
- General Chemical & Material Sciences (AREA)
- Medicinal Chemistry (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- Pharmacology & Pharmacy (AREA)
- Animal Behavior & Ethology (AREA)
- Oncology (AREA)
- Communicable Diseases (AREA)
- Tropical Medicine & Parasitology (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Agricultural Chemicals And Associated Chemicals (AREA)
- Heterocyclic Carbon Compounds Containing A Hetero Ring Having Oxygen Or Sulfur (AREA)
- Saccharide Compounds (AREA)
- Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
Applications Claiming Priority (6)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| GB868613790A GB8613790D0 (en) | 1986-06-06 | 1986-06-06 | Chemical compounds |
| GB8613790 | 1986-06-06 | ||
| GB8625854 | 1986-10-29 | ||
| GB868625854A GB8625854D0 (en) | 1986-10-29 | 1986-10-29 | Chemical process |
| GB8708423 | 1987-04-08 | ||
| GB878708423A GB8708423D0 (en) | 1987-04-08 | 1987-04-08 | Chemical compounds |
Publications (3)
| Publication Number | Publication Date |
|---|---|
| NL8701322A NL8701322A (nl) | 1988-01-04 |
| NL193376B NL193376B (nl) | 1999-04-01 |
| NL193376C true NL193376C (nl) | 1999-08-03 |
Family
ID=27263057
Family Applications (2)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| NL8701322A NL193376C (nl) | 1986-06-06 | 1987-06-05 | 16-Ledig pentacyclische macrolideverbindingen, preparaten die deze bevatten en gebruik ervan. |
| NL990026C NL990026I2 (nl) | 1986-06-06 | 1999-08-18 | 16-Ledig pentacyclische macrolideverbindingen, preparaten die deze bevatten en gebruik ervan. |
Family Applications After (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| NL990026C NL990026I2 (nl) | 1986-06-06 | 1999-08-18 | 16-Ledig pentacyclische macrolideverbindingen, preparaten die deze bevatten en gebruik ervan. |
Country Status (35)
| Country | Link |
|---|---|
| US (1) | US4900753A (pl) |
| JP (1) | JP2648147B2 (pl) |
| KR (1) | KR950010077B1 (pl) |
| CN (1) | CN1023858C (pl) |
| AR (1) | AR244691A1 (pl) |
| AT (1) | AT398571B (pl) |
| AU (1) | AU609399B2 (pl) |
| BE (1) | BE1000201A4 (pl) |
| BR (1) | BR8702866A (pl) |
| CA (1) | CA1296329C (pl) |
| CH (1) | CH677670A5 (pl) |
| DE (3) | DE3718926C2 (pl) |
| DK (1) | DK166498B1 (pl) |
| EG (1) | EG18752A (pl) |
| ES (1) | ES2006479A6 (pl) |
| FI (2) | FI90663C (pl) |
| FR (1) | FR2599742B1 (pl) |
| GB (1) | GB2192630B (pl) |
| GE (1) | GEP19981388B (pl) |
| GR (1) | GR870891B (pl) |
| HU (1) | HU199847B (pl) |
| IE (1) | IE60411B1 (pl) |
| IL (1) | IL82776A (pl) |
| IT (1) | IT1206015B (pl) |
| LU (2) | LU86908A1 (pl) |
| LV (2) | LV10280A (pl) |
| NL (2) | NL193376C (pl) |
| NZ (1) | NZ220587A (pl) |
| OA (1) | OA08606A (pl) |
| PH (1) | PH23948A (pl) |
| PL (3) | PL155723B1 (pl) |
| PT (1) | PT85018B (pl) |
| SE (1) | SE503399C2 (pl) |
| TR (1) | TR28970A (pl) |
| UA (1) | UA45300C2 (pl) |
Families Citing this family (19)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| ES2058082T3 (es) * | 1986-09-12 | 1994-11-01 | American Cyanamid Co | Derivados 23-oxo (ceto) y 23-imino de compuestos ll-f28249. |
| US4886828A (en) * | 1986-09-12 | 1989-12-12 | American Cyanamid Company | Δ22 -derivatives of LL-F28249 compounds |
| EP0260537A1 (en) * | 1986-09-12 | 1988-03-23 | American Cyanamid Company | 13-Deoxy-23-oxo(keto) and 23-imino derivatives of 13-deoxy C-076-aglycone compounds |
| GB8721377D0 (en) * | 1987-09-11 | 1987-10-21 | Glaxo Group Ltd | Chemical compounds |
| GB8811036D0 (en) * | 1988-05-10 | 1988-06-15 | Glaxo Group Ltd | Chemical compounds |
| GB8813150D0 (en) * | 1988-06-03 | 1988-07-06 | American Cyanamid Co | Chemical compounds |
| GB8905605D0 (en) * | 1989-03-11 | 1989-04-26 | Beecham Group Plc | Novel compounds |
| NZ233680A (en) * | 1989-05-17 | 1995-02-24 | Beecham Group Plc | Avermectins and milbemycins and compositions thereof |
| US4988824A (en) * | 1989-09-11 | 1991-01-29 | Maulding Donald R | Process for the preparation of 23-(C1-C6 alkyloxime)-LL-F28249 compounds |
| CA2097918C (en) * | 1990-12-07 | 2002-07-16 | Frank N. Chang | Stabilized insect nematode compositions |
| JP2855181B2 (ja) | 1993-12-10 | 1999-02-10 | 敏雄 鈴木 | 松類の枯損防止用組成物及び防止方法 |
| EP1197215B1 (en) | 2000-10-10 | 2006-03-22 | Wyeth | Anthelmintic compositions |
| US7348417B2 (en) * | 2003-08-07 | 2008-03-25 | Wyeth | Method of purifying moxidectin through crystallization |
| WO2006119174A1 (en) | 2005-04-30 | 2006-11-09 | Ocular Surface Center, P.A. | Method for treating ocular demodex |
| JP4939025B2 (ja) * | 2005-09-30 | 2012-05-23 | 三菱電線工業株式会社 | 電熱ヒータ付きハンドル用グリップ部材 |
| EP1849363A1 (en) * | 2006-03-09 | 2007-10-31 | Cheminova A/S | Synergistic combination of glutamate- and GABA-gated chloride agonist pesticide and at least one of Vitamin E or Niacin |
| US8128968B2 (en) * | 2007-08-29 | 2012-03-06 | Tissuetech, Inc. | Compositions and methods for treating Demodex infestations |
| MX379693B (es) | 2011-12-02 | 2025-03-11 | Merial Ltd | Formulaciones de moxidectina inyectables de larga acción y formas de cristal de moxidectina novedosas. |
| FR2995605B1 (fr) * | 2012-09-18 | 2014-09-19 | Sanofi Sa | Derives de macrolides, leur preparation et leur application therapeutique. |
Family Cites Families (10)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| PH15982A (en) * | 1977-10-03 | 1983-05-18 | Merck & Co Inc | Selective hydrogenation producta of c-076 compounds and derivatives thereof |
| US4289760A (en) * | 1980-05-02 | 1981-09-15 | Merck & Co., Inc. | 23-Keto derivatives of C-076 compounds |
| US4423209A (en) * | 1982-02-26 | 1983-12-27 | Merck & Co., Inc. | Processes for the interconversion of avermectin compounds |
| JPS59108785A (ja) * | 1982-11-25 | 1984-06-23 | Sankyo Co Ltd | ミルベマイシン類の５−オキシム誘導体 |
| JPS60126289A (ja) * | 1983-11-14 | 1985-07-05 | Sankyo Co Ltd | ミルベマイシン類の５−カ−ボネ−ト誘導体 |
| PT80577B (pt) * | 1984-06-05 | 1987-09-18 | American Cyanamid Co | Processo para a producao de novos agentes macrolidos ll-f28249 uteis no tratamento de infeccoes helminticas por ectoparasitas artropodes e por acarideos |
| US4579864A (en) * | 1984-06-11 | 1986-04-01 | Merck & Co., Inc. | Avermectin and milbemycin 13-keto, 13-imino and 13-amino derivatives |
| GR852232B (pl) * | 1984-09-14 | 1986-01-14 | American Cyanamid Co | |
| ES8802229A1 (es) * | 1985-04-30 | 1988-04-16 | Glaxo Group Ltd | Un procedimiento para preparar nuevos derivados lactonicos macrociclicos. |
| ES2058082T3 (es) * | 1986-09-12 | 1994-11-01 | American Cyanamid Co | Derivados 23-oxo (ceto) y 23-imino de compuestos ll-f28249. |
-
1987
- 1987-05-26 CA CA000537979A patent/CA1296329C/en not_active Expired - Lifetime
- 1987-06-02 OA OA59131A patent/OA08606A/xx unknown
- 1987-06-04 FI FI872517A patent/FI90663C/fi not_active IP Right Cessation
- 1987-06-04 EG EG32487A patent/EG18752A/xx active
- 1987-06-04 DK DK290287A patent/DK166498B1/da not_active IP Right Cessation
- 1987-06-04 ES ES8701645A patent/ES2006479A6/es not_active Expired
- 1987-06-05 HU HU872583A patent/HU199847B/hu unknown
- 1987-06-05 AT AT0143887A patent/AT398571B/de not_active IP Right Cessation
- 1987-06-05 CN CN87104431A patent/CN1023858C/zh not_active Expired - Lifetime
- 1987-06-05 CH CH2150/87A patent/CH677670A5/de not_active IP Right Cessation
- 1987-06-05 DE DE3718926A patent/DE3718926C2/de not_active Expired - Lifetime
- 1987-06-05 FR FR878707915A patent/FR2599742B1/fr not_active Expired
- 1987-06-05 DE DE1998175029 patent/DE19875029I2/de active Active
- 1987-06-05 TR TR00392/87A patent/TR28970A/xx unknown
- 1987-06-05 PL PL1987282198A patent/PL155723B1/pl unknown
- 1987-06-05 BR BR8702866A patent/BR8702866A/pt not_active IP Right Cessation
- 1987-06-05 PL PL1987266100A patent/PL153226B1/pl unknown
- 1987-06-05 AR AR87307796A patent/AR244691A1/es active
- 1987-06-05 JP JP62140139A patent/JP2648147B2/ja not_active Expired - Lifetime
- 1987-06-05 NL NL8701322A patent/NL193376C/nl not_active IP Right Cessation
- 1987-06-05 GR GR870891A patent/GR870891B/el unknown
- 1987-06-05 PL PL1987283187A patent/PL153036B1/pl unknown
- 1987-06-05 DE DE3745133A patent/DE3745133C2/de not_active Expired - Lifetime
- 1987-06-05 PH PH35347A patent/PH23948A/en unknown
- 1987-06-05 SE SE8702361A patent/SE503399C2/sv not_active IP Right Cessation
- 1987-06-05 IE IE149687A patent/IE60411B1/en not_active IP Right Cessation
- 1987-06-05 PT PT85018A patent/PT85018B/pt unknown
- 1987-06-05 AU AU73873/87A patent/AU609399B2/en not_active Expired
- 1987-06-05 LU LU86908A patent/LU86908A1/fr active Protection Beyond IP Right Term
- 1987-06-05 GB GB8713239A patent/GB2192630B/en not_active Expired - Lifetime
- 1987-06-05 IT IT8748023A patent/IT1206015B/it active
- 1987-06-05 KR KR1019870005694A patent/KR950010077B1/ko not_active Expired - Lifetime
- 1987-06-05 NZ NZ220587A patent/NZ220587A/xx unknown
- 1987-06-05 US US07/058,856 patent/US4900753A/en not_active Expired - Lifetime
- 1987-06-05 BE BE8700626A patent/BE1000201A4/fr not_active IP Right Cessation
- 1987-06-05 IL IL82776A patent/IL82776A/xx not_active IP Right Cessation
-
1992
- 1992-07-30 FI FI923445A patent/FI90549C/fi not_active IP Right Cessation
- 1992-12-30 LV LV920561A patent/LV10280A/xx unknown
-
1993
- 1993-08-25 GE GEAP19931498A patent/GEP19981388B/en unknown
- 1993-09-15 UA UA93003885A patent/UA45300C2/uk unknown
- 1993-11-15 LV LVP-93-1233A patent/LV10781B/lv unknown
-
1996
- 1996-07-17 LU LU88790C patent/LU88790I2/fr unknown
-
1999
- 1999-08-18 NL NL990026C patent/NL990026I2/nl unknown
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Legal Events
| Date | Code | Title | Description |
|---|---|---|---|
| CNR | Transfer of rights (patent application after its laying open for public inspection) |
Free format text: AMERICAN CYANAMID COMPANY TE WAYNE |
|
| BA | A request for search or an international-type search has been filed | ||
| BB | A search report has been drawn up | ||
| BC | A request for examination has been filed | ||
| KC1 | Grant of a supplementary protection certificate |
Free format text: 990026, 20070605, EXPIRES: 20091229 |
|
| TNT | Modifications of names of proprietors of patents or applicants of examined patent applications |
Owner name: WYETH HOLDINGS CORPORATION |
|
| V4 | Discontinued because of reaching the maximum lifetime of a patent |
Effective date: 20070605 |