NI201000136A - Inhibidores macrocíclicos de serina proteasa. - Google Patents

Inhibidores macrocíclicos de serina proteasa.

Info

Publication number
NI201000136A
NI201000136A NI201000136A NI201000136A NI201000136A NI 201000136 A NI201000136 A NI 201000136A NI 201000136 A NI201000136 A NI 201000136A NI 201000136 A NI201000136 A NI 201000136A NI 201000136 A NI201000136 A NI 201000136A
Authority
NI
Nicaragua
Prior art keywords
serine protease
macrocyclic inhibitors
macrocyclic
inhibitors
compounds
Prior art date
Application number
NI201000136A
Other languages
English (en)
Spanish (es)
Inventor
Claude Parsy Christophe
Surleraux Dominique
Alexandre Francois-Rene
Derock Michel
Leroy Frederic
Original Assignee
Idenix Pharmaceuticals Inc
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Idenix Pharmaceuticals Inc filed Critical Idenix Pharmaceuticals Inc
Publication of NI201000136A publication Critical patent/NI201000136A/es

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D487/00—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00
    • C07D487/02—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00 in which the condensed system contains two hetero rings
    • C07D487/08—Bridged systems
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • A61P31/12—Antivirals
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • A61P31/12—Antivirals
    • A61P31/14—Antivirals for RNA viruses
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P43/00—Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00

Landscapes

  • Organic Chemistry (AREA)
  • Health & Medical Sciences (AREA)
  • Chemical & Material Sciences (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • General Chemical & Material Sciences (AREA)
  • Public Health (AREA)
  • Medicinal Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Virology (AREA)
  • Animal Behavior & Ethology (AREA)
  • General Health & Medical Sciences (AREA)
  • Veterinary Medicine (AREA)
  • Communicable Diseases (AREA)
  • Oncology (AREA)
  • Engineering & Computer Science (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Molecular Biology (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
  • Nitrogen Condensed Heterocyclic Rings (AREA)
  • Peptides Or Proteins (AREA)
NI201000136A 2008-02-04 2010-08-03 Inhibidores macrocíclicos de serina proteasa. NI201000136A (es)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
US2608608P 2008-02-04 2008-02-04
US8386708P 2008-07-25 2008-07-25

Publications (1)

Publication Number Publication Date
NI201000136A true NI201000136A (es) 2011-03-23

Family

ID=40568607

Family Applications (1)

Application Number Title Priority Date Filing Date
NI201000136A NI201000136A (es) 2008-02-04 2010-08-03 Inhibidores macrocíclicos de serina proteasa.

Country Status (21)

Country Link
US (2) US8003659B2 (enExample)
EP (1) EP2250174B1 (enExample)
JP (1) JP5574982B2 (enExample)
KR (1) KR20100118991A (enExample)
CN (1) CN101977915B (enExample)
AR (1) AR070413A1 (enExample)
AU (1) AU2009210789B2 (enExample)
BR (1) BRPI0908021A2 (enExample)
CA (1) CA2712971A1 (enExample)
CO (1) CO6501153A2 (enExample)
CR (1) CR11618A (enExample)
EC (1) ECSP10010413A (enExample)
ES (1) ES2437147T3 (enExample)
IL (1) IL207333A0 (enExample)
MX (1) MX2010008523A (enExample)
NI (1) NI201000136A (enExample)
NZ (1) NZ587133A (enExample)
RU (1) RU2490272C2 (enExample)
TW (1) TW200936131A (enExample)
WO (1) WO2009099596A2 (enExample)
ZA (1) ZA201005318B (enExample)

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AU2009210789B2 (en) 2014-01-30
EP2250174B1 (en) 2013-08-28
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