AR070413A1 - Inhibidores macrociclicos de proteasa de serina - Google Patents

Inhibidores macrociclicos de proteasa de serina

Info

Publication number
AR070413A1
AR070413A1 ARP090100353A ARP090100353A AR070413A1 AR 070413 A1 AR070413 A1 AR 070413A1 AR P090100353 A ARP090100353 A AR P090100353A AR P090100353 A ARP090100353 A AR P090100353A AR 070413 A1 AR070413 A1 AR 070413A1
Authority
AR
Argentina
Prior art keywords
heterocyclyl
alkyl
aryl
alkynyl
cycloalkyl
Prior art date
Application number
ARP090100353A
Other languages
English (en)
Spanish (es)
Original Assignee
Idenix Pharmaceuticals Inc
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Idenix Pharmaceuticals Inc filed Critical Idenix Pharmaceuticals Inc
Publication of AR070413A1 publication Critical patent/AR070413A1/es

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D487/00—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00
    • C07D487/02—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00 in which the condensed system contains two hetero rings
    • C07D487/08—Bridged systems
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • A61P31/12—Antivirals
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • A61P31/12—Antivirals
    • A61P31/14—Antivirals for RNA viruses
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P43/00—Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00

Landscapes

  • Chemical & Material Sciences (AREA)
  • Health & Medical Sciences (AREA)
  • Organic Chemistry (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Public Health (AREA)
  • Animal Behavior & Ethology (AREA)
  • Veterinary Medicine (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • General Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Virology (AREA)
  • Pharmacology & Pharmacy (AREA)
  • General Health & Medical Sciences (AREA)
  • Oncology (AREA)
  • Communicable Diseases (AREA)
  • Molecular Biology (AREA)
  • Engineering & Computer Science (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
  • Nitrogen Condensed Heterocyclic Rings (AREA)
  • Peptides Or Proteins (AREA)
ARP090100353A 2008-02-04 2009-02-03 Inhibidores macrociclicos de proteasa de serina AR070413A1 (es)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
US2608608P 2008-02-04 2008-02-04
US8386708P 2008-07-25 2008-07-25

Publications (1)

Publication Number Publication Date
AR070413A1 true AR070413A1 (es) 2010-04-07

Family

ID=40568607

Family Applications (1)

Application Number Title Priority Date Filing Date
ARP090100353A AR070413A1 (es) 2008-02-04 2009-02-03 Inhibidores macrociclicos de proteasa de serina

Country Status (21)

Country Link
US (2) US8003659B2 (enExample)
EP (1) EP2250174B1 (enExample)
JP (1) JP5574982B2 (enExample)
KR (1) KR20100118991A (enExample)
CN (1) CN101977915B (enExample)
AR (1) AR070413A1 (enExample)
AU (1) AU2009210789B2 (enExample)
BR (1) BRPI0908021A2 (enExample)
CA (1) CA2712971A1 (enExample)
CO (1) CO6501153A2 (enExample)
CR (1) CR11618A (enExample)
EC (1) ECSP10010413A (enExample)
ES (1) ES2437147T3 (enExample)
IL (1) IL207333A0 (enExample)
MX (1) MX2010008523A (enExample)
NI (1) NI201000136A (enExample)
NZ (1) NZ587133A (enExample)
RU (1) RU2490272C2 (enExample)
TW (1) TW200936131A (enExample)
WO (1) WO2009099596A2 (enExample)
ZA (1) ZA201005318B (enExample)

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US20170135990A1 (en) 2014-03-05 2017-05-18 Idenix Pharmaceuticals Llc Pharmaceutical compositions comprising a 5,5-fused heteroarylene flaviviridae inhibitor and their use for treating or preventing flaviviridae infection
US20170066779A1 (en) 2014-03-05 2017-03-09 Idenix Pharmaceuticals Llc Solid forms of a flaviviridae virus inhibitor compound and salts thereof
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CN109562107A (zh) 2016-05-10 2019-04-02 C4医药公司 用于靶蛋白降解的杂环降解决定子体
CN109790143A (zh) 2016-05-10 2019-05-21 C4医药公司 用于靶蛋白降解的胺连接的c3-戊二酰亚胺降解决定子体
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