LT4477B - Fluoksetino enterinės piliulės - Google Patents
Fluoksetino enterinės piliulės Download PDFInfo
- Publication number
- LT4477B LT4477B LT98-058A LT98058A LT4477B LT 4477 B LT4477 B LT 4477B LT 98058 A LT98058 A LT 98058A LT 4477 B LT4477 B LT 4477B
- Authority
- LT
- Lithuania
- Prior art keywords
- fluoxetine
- layer
- enteric
- core
- hpmcas
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- 229920000523 polyvinylpolypyrrolidone Polymers 0.000 description 1
- 230000002028 premature Effects 0.000 description 1
- 238000002360 preparation method Methods 0.000 description 1
- 238000003825 pressing Methods 0.000 description 1
- 238000005086 pumping Methods 0.000 description 1
- 229920013730 reactive polymer Polymers 0.000 description 1
- 230000000306 recurrent effect Effects 0.000 description 1
- 230000004044 response Effects 0.000 description 1
- 229960002073 sertraline Drugs 0.000 description 1
- VGKDLMBJGBXTGI-SJCJKPOMSA-N sertraline Chemical compound C1([C@@H]2CC[C@@H](C3=CC=CC=C32)NC)=CC=C(Cl)C(Cl)=C1 VGKDLMBJGBXTGI-SJCJKPOMSA-N 0.000 description 1
- 231100000872 sexual dysfunction Toxicity 0.000 description 1
- 229960004029 silicic acid Drugs 0.000 description 1
- 235000019333 sodium laurylsulphate Nutrition 0.000 description 1
- 241000894007 species Species 0.000 description 1
- 238000003860 storage Methods 0.000 description 1
- 125000002730 succinyl group Chemical group C(CCC(=O)*)(=O)* 0.000 description 1
- 238000009495 sugar coating Methods 0.000 description 1
- 230000002459 sustained effect Effects 0.000 description 1
- 238000013268 sustained release Methods 0.000 description 1
- 239000012730 sustained-release form Substances 0.000 description 1
- 239000007916 tablet composition Substances 0.000 description 1
- 229940033134 talc Drugs 0.000 description 1
- 238000002560 therapeutic procedure Methods 0.000 description 1
- 239000010936 titanium Substances 0.000 description 1
- 229910052719 titanium Inorganic materials 0.000 description 1
- 235000010215 titanium dioxide Nutrition 0.000 description 1
- 238000004448 titration Methods 0.000 description 1
- 230000003245 working effect Effects 0.000 description 1
Classifications
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/13—Amines
- A61K31/135—Amines having aromatic rings, e.g. ketamine, nortriptyline
- A61K31/138—Aryloxyalkylamines, e.g. propranolol, tamoxifen, phenoxybenzamine
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K9/00—Medicinal preparations characterised by special physical form
- A61K9/48—Preparations in capsules, e.g. of gelatin, of chocolate
- A61K9/50—Microcapsules having a gas, liquid or semi-solid filling; Solid microparticles or pellets surrounded by a distinct coating layer, e.g. coated microspheres, coated drug crystals
- A61K9/5073—Microcapsules having a gas, liquid or semi-solid filling; Solid microparticles or pellets surrounded by a distinct coating layer, e.g. coated microspheres, coated drug crystals having two or more different coatings optionally including drug-containing subcoatings
- A61K9/5078—Microcapsules having a gas, liquid or semi-solid filling; Solid microparticles or pellets surrounded by a distinct coating layer, e.g. coated microspheres, coated drug crystals having two or more different coatings optionally including drug-containing subcoatings with drug-free core
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/24—Antidepressants
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/26—Psychostimulants, e.g. nicotine, cocaine
Landscapes
- Health & Medical Sciences (AREA)
- Engineering & Computer Science (AREA)
- Bioinformatics & Cheminformatics (AREA)
- Chemical & Material Sciences (AREA)
- Medicinal Chemistry (AREA)
- Pharmacology & Pharmacy (AREA)
- Life Sciences & Earth Sciences (AREA)
- Animal Behavior & Ethology (AREA)
- General Health & Medical Sciences (AREA)
- Public Health (AREA)
- Veterinary Medicine (AREA)
- Epidemiology (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- Biomedical Technology (AREA)
- Neurology (AREA)
- Neurosurgery (AREA)
- Chemical Kinetics & Catalysis (AREA)
- General Chemical & Material Sciences (AREA)
- Organic Chemistry (AREA)
- Psychiatry (AREA)
- Pain & Pain Management (AREA)
- Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
- Medicinal Preparation (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Saccharide Compounds (AREA)
Applications Claiming Priority (1)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| US08/867,196 US5910319A (en) | 1997-05-29 | 1997-05-29 | Fluoxetine enteric pellets and methods for their preparation and use |
Publications (2)
| Publication Number | Publication Date |
|---|---|
| LT98058A LT98058A (en) | 1998-10-26 |
| LT4477B true LT4477B (lt) | 1999-03-25 |
Family
ID=25349313
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| LT98-058A LT4477B (lt) | 1997-05-29 | 1998-04-22 | Fluoksetino enterinės piliulės |
Country Status (45)
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| FR2752732B1 (fr) * | 1996-08-28 | 1998-11-20 | Pf Medicament | Forme galenique a liberation prolongee de milnacipran |
| CA2698347A1 (en) * | 1999-05-20 | 2000-11-30 | Elan Pharma International Limited | Multiparticulate controlled release selective serotonin reuptake inhibitor formulations |
| IE990406A1 (en) | 1999-05-20 | 2000-12-27 | Elan Corp Plc | Multiparticulate controlled release selective serotonin reuptake inhibitor formulations. |
| ES2162560B1 (es) * | 1999-06-25 | 2002-07-16 | Rodriguez Concepcion Pena | Uso de fluoxetina, paroxetina y otros isrs para la fabricacion de medicamentos con el fin de aumentar la capacidad de abstenerse de substancias o actividades que crean dependencia. |
| CZ299712B6 (cs) | 1999-09-03 | 2008-10-29 | Apbi Holdings, Llc | Použití dapoxetinu pro zvládnutí sexuální dysfunkce podáváním zpusobem podle potreby |
| CN1094347C (zh) * | 1999-11-15 | 2002-11-20 | 广东药学院药物研究所 | 一种治疗前列腺良性增生症的控释微丸及其制备方法 |
| US6273260B1 (en) | 2000-03-08 | 2001-08-14 | Eli Lilly And Company | Pharmaceutical packaging system |
| ES2185452B2 (es) * | 2000-08-01 | 2004-03-16 | Cinfa S A Lab | Composicion farmaceutica de fluoxetina en comprimido dispersable recubierto y su proceso de fabricacion. |
| JP4181738B2 (ja) * | 2000-08-25 | 2008-11-19 | 信越化学工業株式会社 | 腸溶性コーティング製剤の製造方法 |
| US6482440B2 (en) * | 2000-09-21 | 2002-11-19 | Phase 2 Discovery, Inc. | Long acting antidepressant microparticles |
| AU2002212102A1 (en) * | 2000-11-08 | 2002-05-21 | Aeromatic-Fielder Ag | A process for production of particles for pharmaceutical compositions having increased bioavailability |
| US20040170688A1 (en) * | 2001-08-06 | 2004-09-02 | Deshmukh Abhijit Mukund | Enteric formulation of fluoxetin |
| WO2003013480A1 (en) | 2001-08-06 | 2003-02-20 | Dr. Reddy's Laboratories Ltd. | Improved enteric formulation of fluoxetin |
| US20040220153A1 (en) * | 2002-09-24 | 2004-11-04 | Jost-Price Edward Roydon | Methods and reagents for the treatment of diseases and disorders associated with increased levels of proinflammatory cytokines |
| WO2004058228A1 (en) * | 2002-12-24 | 2004-07-15 | Lupin Limited | Enteric coated fluoxetine composition |
| US8614247B2 (en) * | 2003-04-10 | 2013-12-24 | Institut National De La Sante Et De La Recherche Medicale | Methods for preventing, attenuating or treating pulmonary hypertension using a serotonin transporter inhibitor, and pharmaceutical compositions for the treatment thereof |
| JP4901474B2 (ja) | 2003-05-30 | 2012-03-21 | ランバクシー ラボラトリーズ リミテッド | 置換ピロール誘導体 |
| US20050176693A1 (en) * | 2003-08-12 | 2005-08-11 | Boissonneault Roger M. | Method of intermittent administration of a pharmaceutical for the treatment of conditions associated with a female's menstrual cycle |
| US20070141150A1 (en) * | 2003-12-30 | 2007-06-21 | Raghupathi Kandarapu | Pharmaceutical composition |
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| KR100920856B1 (ko) * | 2004-11-30 | 2009-10-09 | (주)아모레퍼시픽 | 선택적 세로토닌 재흡수 억제제의 연장방출 제제 및 그제조방법 |
| EP1730132A2 (de) * | 2004-12-23 | 2006-12-13 | Teva Pharmaceutical Industries Ltd | Verfahren zur herstellung pharmazeutisch unbedenklicher salze von duloxetin und zwischenprodukten davon |
| AU2006274565B2 (en) * | 2005-08-02 | 2012-05-17 | Lupin Limited | Novel controlled release compositions of selective serotonin reuptake inhibitors |
| KR101329112B1 (ko) | 2005-11-08 | 2013-11-14 | 랜박시 래보러터리스 리미티드 | (3ｒ,5ｒ)-7-〔2-(4-플루오로페닐)-5-이소프로필-3-페닐-4-〔(4-히드록시 메틸 페닐 아미노)카르보닐〕-피롤-1-일〕-3,5-디히드록시 헵탄산 헤미 칼슘염의 제조 방법 |
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| CN101057837B (zh) * | 2006-04-20 | 2010-12-22 | 湖南九典制药有限公司 | 一种右旋酮洛芬肠溶微丸及制备方法 |
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| EP2026768B1 (de) * | 2006-06-01 | 2018-02-28 | Dexcel Pharma Technologies Ltd. | Pharmazeutische formulierung auf mehreren einheiten |
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| KR101612146B1 (ko) | 2008-07-16 | 2016-04-12 | 리히터 게데온 닐트. | 도파민 수용체 리간드를 함유하는 약학적 제형 |
| WO2010026993A1 (ja) * | 2008-09-03 | 2010-03-11 | 武田薬品工業株式会社 | 製剤における吸収性改善方法および吸収性が改善された製剤 |
| CN101804145B (zh) * | 2009-02-12 | 2012-11-14 | 杭州赛利药物研究所有限公司 | 一种大蒜油肠溶微丸胶囊及其制备方法 |
| JP2013504562A (ja) * | 2009-09-17 | 2013-02-07 | カディラ・ヘルスケア・リミテッド | アルコールで誘発される用量ダンピングを低減するための医薬組成物 |
| WO2011102504A1 (ja) * | 2010-02-22 | 2011-08-25 | 第一三共株式会社 | 経口用徐放性固形製剤 |
| RU2442572C1 (ru) * | 2010-12-23 | 2012-02-20 | Ольга Львовна Титова | Энтеросолюбильная оболочка и композиция для ее получения |
| ES2728850T3 (es) * | 2012-05-02 | 2019-10-29 | Capsugel Belgium Nv | Dispersiones acuosas de acetato acetato succinato de hidroxipropilmetilcelulosa (HPMCAS) |
| CN102716084B (zh) * | 2012-06-29 | 2013-09-25 | 海南美大制药有限公司 | 盐酸氟西汀脂质体固体制剂 |
| KR102127625B1 (ko) | 2012-09-03 | 2020-06-29 | 다이이찌 산쿄 가부시키가이샤 | 하이드로모르폰염산염 함유의 경구용 서방성 의약 조성물 |
| EP2919788A4 (de) | 2012-11-14 | 2016-05-25 | Univ Johns Hopkins | Verfahren und zusammensetzungen zur behandlung von schizophrenie |
| WO2015179072A1 (en) | 2014-05-20 | 2015-11-26 | Dow Global Technologies Llc | Dispersion comprising a partially neutralized esterified cellulose ether |
| US9782356B2 (en) | 2014-05-20 | 2017-10-10 | Dow Global Technologies Llc | Capsule shells comprising an esterified cellulose ether |
| US10564114B2 (en) * | 2014-06-07 | 2020-02-18 | Structure-Ase Incorporated | Method for the detection and/or diagnosis of eating disorders and malnutrition using X-ray diffraction |
| US10471152B2 (en) | 2014-08-29 | 2019-11-12 | Capsugel Belgium Nv | Colloidal dispersion comprising HPMCAS |
| US20170042806A1 (en) | 2015-04-29 | 2017-02-16 | Dexcel Pharma Technologies Ltd. | Orally disintegrating compositions |
| US10076494B2 (en) | 2016-06-16 | 2018-09-18 | Dexcel Pharma Technologies Ltd. | Stable orally disintegrating pharmaceutical compositions |
| US11274087B2 (en) | 2016-07-08 | 2022-03-15 | Richter Gedeon Nyrt. | Industrial process for the preparation of cariprazine |
| MA52457A (fr) | 2017-04-13 | 2021-03-10 | Chase Therapeutics Corp | Combinaison pharmaceutique et son utilisation pour le traitement de synucléinopathies |
| HUP1700253A1 (hu) | 2017-06-13 | 2019-01-28 | Richter Gedeon Nyrt | Szilárd orális gyógyszerkészítmények |
| CN107898942B (zh) * | 2017-11-24 | 2021-01-26 | 一力制药(罗定)有限公司 | 一种感冒清热胶囊及其制备方法 |
| US11547707B2 (en) | 2019-04-10 | 2023-01-10 | Richter Gedeon Nyrt. | Carbamoyl cyclohexane derivatives for treating autism spectrum disorder |
| JP7606825B2 (ja) * | 2020-06-15 | 2024-12-26 | 東和薬品株式会社 | エソメプラゾール顆粒ならびにその製造方法および用途 |
| WO2022115054A1 (en) * | 2020-11-27 | 2022-06-02 | Santa Farma Ilac Sanayii A.S. | Enteric coated duloxetine compositions |
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-
1997
- 1997-05-29 US US08/867,196 patent/US5910319A/en not_active Ceased
-
1998
- 1998-04-13 IL IL12407398A patent/IL124073A/en not_active IP Right Cessation
- 1998-04-14 CA CA002234826A patent/CA2234826C/en not_active Expired - Lifetime
- 1998-04-14 RU RU98106998/14A patent/RU2164405C2/ru active
- 1998-04-14 RO RO98-00869A patent/RO120043B1/ro unknown
- 1998-04-15 GB GB9807939A patent/GB2325623B/en not_active Expired - Lifetime
- 1998-04-15 CZ CZ19981143A patent/CZ290582B6/cs not_active IP Right Cessation
- 1998-04-15 RS YUP-165/98A patent/RS49827B/sr unknown
- 1998-04-15 HU HU9800882A patent/HUP9800882A3/hu not_active Application Discontinuation
- 1998-04-15 UA UA98041929A patent/UA48193C2/uk unknown
- 1998-04-15 NZ NZ330192A patent/NZ330192A/xx not_active IP Right Cessation
- 1998-04-15 ZA ZA9803173A patent/ZA983173B/xx unknown
- 1998-04-16 MY MYPI98001702A patent/MY118139A/en unknown
- 1998-04-16 FI FI980846A patent/FI119971B/fi active IP Right Grant
- 1998-04-17 SE SE9801336A patent/SE522914C2/sv not_active IP Right Cessation
- 1998-04-17 SG SG1998000871A patent/SG72805A1/en unknown
- 1998-04-20 KR KR1019980014014A patent/KR100549473B1/ko not_active Expired - Lifetime
- 1998-04-22 LT LT98-058A patent/LT4477B/lt not_active IP Right Cessation
- 1998-04-24 CN CNB981087787A patent/CN1161109C/zh not_active Expired - Lifetime
- 1998-04-24 JP JP15350198A patent/JP3210288B2/ja not_active Expired - Lifetime
- 1998-04-28 SV SV1998000052A patent/SV1998000052A/es unknown
- 1998-04-28 ES ES009800899A patent/ES2161574B1/es not_active Expired - Fee Related
- 1998-04-28 IT IT98MI000908A patent/ITMI980908A1/it unknown
- 1998-04-29 SI SI9800128A patent/SI9800128B/sl unknown
- 1998-05-01 PL PL326134A patent/PL192293B1/pl unknown
- 1998-05-07 AR ARP980102130A patent/AR011728A1/es not_active Application Discontinuation
- 1998-05-08 PT PT102152A patent/PT102152B/pt active IP Right Grant
- 1998-05-11 TW TW087107241A patent/TWI239838B/zh not_active IP Right Cessation
- 1998-05-12 CO CO98026349A patent/CO4940407A1/es unknown
- 1998-05-13 FR FR9806040A patent/FR2763846B1/fr not_active Expired - Lifetime
- 1998-05-14 NO NO19982197A patent/NO317743B1/no not_active IP Right Cessation
- 1998-05-19 BR BR9801989-9A patent/BR9801989A/pt not_active Application Discontinuation
- 1998-05-20 LU LU90245A patent/LU90245B1/fr active
- 1998-05-20 BE BE9800383A patent/BE1011925A3/fr not_active IP Right Cessation
- 1998-05-25 LV LVP-98-121A patent/LV12176B/xx unknown
- 1998-05-26 NL NL1009259A patent/NL1009259C2/nl not_active IP Right Cessation
- 1998-05-26 CH CH01157/98A patent/CH693018A5/de not_active IP Right Cessation
- 1998-05-27 TR TR1998/00937A patent/TR199800937A2/xx unknown
- 1998-05-28 PE PE1998000430A patent/PE75399A1/es not_active Application Discontinuation
- 1998-05-28 GR GR980100188A patent/GR980100188A/el unknown
- 1998-05-28 DK DK199800728A patent/DK176776B1/da not_active IP Right Cessation
- 1998-05-28 AU AU69048/98A patent/AU726690B2/en not_active Expired
- 1998-05-28 DE DE19823940A patent/DE19823940B4/de not_active Expired - Lifetime
- 1998-05-28 ID IDP980791A patent/ID20343A/id unknown
- 1998-05-29 AT AT0093198A patent/AT408068B/de not_active IP Right Cessation
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1999
- 1999-03-10 US US09/265,610 patent/US5985322A/en not_active Expired - Lifetime
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2000
- 2000-07-25 CN CNB001222090A patent/CN1212834C/zh not_active Expired - Lifetime
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2002
- 2002-01-28 US US10/058,891 patent/USRE39030E1/en not_active Expired - Lifetime
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Legal Events
| Date | Code | Title | Description |
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| MK9A | Expiry of a patent |
Effective date: 20180422 |