LT3318565T - Pirolo[2,3-d]pirimidinilo, pirolo[2,3-b]pirazinilo ir pirolo[2,3-d]piridinilo akrilamidai - Google Patents

Pirolo[2,3-d]pirimidinilo, pirolo[2,3-b]pirazinilo ir pirolo[2,3-d]piridinilo akrilamidai

Info

Publication number
LT3318565T
LT3318565T LTEP17200940.9T LT17200940T LT3318565T LT 3318565 T LT3318565 T LT 3318565T LT 17200940 T LT17200940 T LT 17200940T LT 3318565 T LT3318565 T LT 3318565T
Authority
LT
Lithuania
Prior art keywords
pyrrolo
pyrazinyl
pyrimidinyl
acrylamides
pyridinyl
Prior art date
Application number
LTEP17200940.9T
Other languages
English (en)
Inventor
Matthew Frank Brown
Agustin Casimiro-Garcia
Ye Che
Jotham Wadsworth Coe
Mark Edward Flanagan
Adam Matthew Gilbert
Matthew Merrill Hayward
Jonathan David LANGILLE
Justin Ian Montgomery
Jean-Baptiste Telliez
Atli Thorarensen
Rayomand Jal Unwalla
John I Trujillo
Original Assignee
Pfizer Inc.
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Family has litigation
First worldwide family litigation filed litigation Critical https://patents.darts-ip.com/?family=52144776&utm_source=google_patent&utm_medium=platform_link&utm_campaign=public_patent_search&patent=LT3318565(T) "Global patent litigation dataset” by Darts-ip is licensed under a Creative Commons Attribution 4.0 International License.
Application filed by Pfizer Inc. filed Critical Pfizer Inc.
Publication of LT3318565T publication Critical patent/LT3318565T/lt

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    • C07D487/00—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00
    • C07D487/02—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00 in which the condensed system contains two hetero rings
    • C07D487/04—Ortho-condensed systems
    • C—CHEMISTRY; METALLURGY
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    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D471/00—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00
    • C07D471/02—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00 in which the condensed system contains two hetero rings
    • C07D471/04—Ortho-condensed systems
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    • A61K31/33—Heterocyclic compounds
    • A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/435—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom
    • A61K31/4353—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom ortho- or peri-condensed with heterocyclic ring systems
    • A61K31/4375—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom ortho- or peri-condensed with heterocyclic ring systems the heterocyclic ring system containing a six-membered ring having nitrogen as a ring heteroatom, e.g. quinolizines, naphthyridines, berberine, vincamine
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    • A61K31/44—Non condensed pyridines; Hydrogenated derivatives thereof
    • A61K31/445—Non condensed piperidines, e.g. piperocaine
    • A61K31/4523—Non condensed piperidines, e.g. piperocaine containing further heterocyclic ring systems
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    • A61K31/505—Pyrimidines; Hydrogenated pyrimidines, e.g. trimethoprim
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LTEP17200940.9T 2013-12-05 2014-11-20 Pirolo[2,3-d]pirimidinilo, pirolo[2,3-b]pirazinilo ir pirolo[2,3-d]piridinilo akrilamidai LT3318565T (lt)

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US201361912074P 2013-12-05 2013-12-05

Publications (1)

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LT3318565T true LT3318565T (lt) 2021-06-25

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ID=52144776

Family Applications (2)

Application Number Title Priority Date Filing Date
LTEP14816404.9T LT3077395T (lt) 2013-12-05 2014-11-20 Pirolo[2,3-d]pirimidinilo, pirolo[2,3-b]pirazinilo ir pirolo[2,3-d]piridinilo akrilamidai
LTEP17200940.9T LT3318565T (lt) 2013-12-05 2014-11-20 Pirolo[2,3-d]pirimidinilo, pirolo[2,3-b]pirazinilo ir pirolo[2,3-d]piridinilo akrilamidai

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LTEP14816404.9T LT3077395T (lt) 2013-12-05 2014-11-20 Pirolo[2,3-d]pirimidinilo, pirolo[2,3-b]pirazinilo ir pirolo[2,3-d]piridinilo akrilamidai

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US (3) US9617258B2 (lt)
EP (2) EP3318565B1 (lt)
JP (2) JP6192839B2 (lt)
KR (1) KR101930603B1 (lt)
CN (2) CN106061973B (lt)
AP (1) AP2016009269A0 (lt)
AR (1) AR099363A1 (lt)
AU (1) AU2014358792C1 (lt)
BR (1) BR112016012262B1 (lt)
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