SV2016005209A - Acrilamidas de pirrolo(2,3-d)pirimidinilo, pirrolo(2,3-b)pirazinilo y pirrolo(2,3-d)piridinilo - Google Patents

Acrilamidas de pirrolo(2,3-d)pirimidinilo, pirrolo(2,3-b)pirazinilo y pirrolo(2,3-d)piridinilo

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Publication number
SV2016005209A
SV2016005209A SV2016005209A SV2016005209A SV2016005209A SV 2016005209 A SV2016005209 A SV 2016005209A SV 2016005209 A SV2016005209 A SV 2016005209A SV 2016005209 A SV2016005209 A SV 2016005209A SV 2016005209 A SV2016005209 A SV 2016005209A
Authority
SV
El Salvador
Prior art keywords
pirrolo
pyrimidinyl
piridinyl
pyrazinyl
acrylic
Prior art date
Application number
SV2016005209A
Other languages
English (en)
Inventor
Matthew Frank Brown
Agustin Casimiro-Garcia
Ye Che
Jotham Wadsworth Coe
Jonathan David Langille
Jean-Baptiste Telliez
Atli Thorarensen
Rayomand Jal Unwalla
John I Trujillo
Mark Edward Flanagan
Adam Matthew Gilbert
Justin Ian Montgomery
Matthew Merrill Hayward
Original Assignee
Pfizer
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Family has litigation
First worldwide family litigation filed litigation Critical https://patents.darts-ip.com/?family=52144776&utm_source=google_patent&utm_medium=platform_link&utm_campaign=public_patent_search&patent=SV2016005209(A) "Global patent litigation dataset” by Darts-ip is licensed under a Creative Commons Attribution 4.0 International License.
Application filed by Pfizer filed Critical Pfizer
Publication of SV2016005209A publication Critical patent/SV2016005209A/es

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    • A61K31/4375Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom ortho- or peri-condensed with heterocyclic ring systems the heterocyclic ring system containing a six-membered ring having nitrogen as a ring heteroatom, e.g. quinolizines, naphthyridines, berberine, vincamine
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Abstract

LA PRESENTE INVENCIÓN PROVEE ACRILAMIDAS FARMACÉUTICAMENTE ACTIVAS DE PIRROLO[2,3-D]PIRIMIDINILO Y PIRROLO[2,3-D]PIRIDINILO Y ANÁLOGOS DE LAS MISMAS. DICHOS COMPUESTOS SON ÚTILES PARA INHIBIR QUINASA DE JANUS. ESTA INVENCIÓN TAMBIÉN ESTÁ DIRIGIDA A COMPOSICIONES QUE COMPRENDEN MÉTODOS PARA HACER DICHOS COMPUESTOS, Y MÉTODOS PARA TRATAR Y PREVENIR CONDICIONES MEDIADAS POR JAK
SV2016005209A 2013-12-05 2016-06-03 Acrilamidas de pirrolo(2,3-d)pirimidinilo, pirrolo(2,3-b)pirazinilo y pirrolo(2,3-d)piridinilo SV2016005209A (es)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
US201361912074P 2013-12-05 2013-12-05

Publications (1)

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SV2016005209A true SV2016005209A (es) 2018-04-11

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SV2016005209A SV2016005209A (es) 2013-12-05 2016-06-03 Acrilamidas de pirrolo(2,3-d)pirimidinilo, pirrolo(2,3-b)pirazinilo y pirrolo(2,3-d)piridinilo

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US (3) US9617258B2 (es)
EP (2) EP3318565B1 (es)
JP (2) JP6192839B2 (es)
KR (1) KR101930603B1 (es)
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AP (1) AP2016009269A0 (es)
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AU (1) AU2014358792C1 (es)
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CN106065017B (zh) 2013-09-18 2018-06-01 北京韩美药品有限公司 抑制btk和/或jak3激酶活性的化合物
SI3318565T1 (sl) * 2013-12-05 2021-07-30 Pfizer Inc. Pirolo(2,3-D)pirimidinil, pirolo(2,3-B)pirazinil in pirolo(2,3-D)piridinil akrilamidi
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