KR860008189A - 7-아미노-3- 프로페닐 세팔로스포란산 및 그 에스텔 - Google Patents

7-아미노-3- 프로페닐 세팔로스포란산 및 그 에스텔 Download PDF

Info

Publication number
KR860008189A
KR860008189A KR1019860003085A KR860003085A KR860008189A KR 860008189 A KR860008189 A KR 860008189A KR 1019860003085 A KR1019860003085 A KR 1019860003085A KR 860003085 A KR860003085 A KR 860003085A KR 860008189 A KR860008189 A KR 860008189A
Authority
KR
South Korea
Prior art keywords
compound
group
salt
lithium
amino
Prior art date
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
Ceased
Application number
KR1019860003085A
Other languages
English (en)
Korean (ko)
Inventor
호시 히데끼
오쿠무라 준
아베 요시오
나이또 다까유끼
아부라끼 심페리
Original Assignee
이삭 쟈코브스키
브리스톨 마이어즈 컴파니
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by 이삭 쟈코브스키, 브리스톨 마이어즈 컴파니 filed Critical 이삭 쟈코브스키
Publication of KR860008189A publication Critical patent/KR860008189A/ko
Priority to KR1019900002094A priority Critical patent/KR900004930B1/ko
Ceased legal-status Critical Current

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D501/00—Heterocyclic compounds containing 5-thia-1-azabicyclo [4.2.0] octane ring systems, i.e. compounds containing a ring system of the formula:, e.g. cephalosporins; Such ring systems being further condensed, e.g. 2,3-condensed with an oxygen-, nitrogen- or sulfur-containing hetero ring
    • C07D501/14—Compounds having a nitrogen atom directly attached in position 7
    • C07D501/16—Compounds having a nitrogen atom directly attached in position 7 with a double bond between positions 2 and 3
    • C07D501/18—7-Aminocephalosporanic or substituted 7-aminocephalosporanic acids
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D501/00—Heterocyclic compounds containing 5-thia-1-azabicyclo [4.2.0] octane ring systems, i.e. compounds containing a ring system of the formula:, e.g. cephalosporins; Such ring systems being further condensed, e.g. 2,3-condensed with an oxygen-, nitrogen- or sulfur-containing hetero ring
    • C07D501/14—Compounds having a nitrogen atom directly attached in position 7
    • C07D501/16—Compounds having a nitrogen atom directly attached in position 7 with a double bond between positions 2 and 3
    • C07D501/20—7-Acylaminocephalosporanic or substituted 7-acylaminocephalosporanic acids in which the acyl radicals are derived from carboxylic acids
    • C07D501/22—7-Acylaminocephalosporanic or substituted 7-acylaminocephalosporanic acids in which the acyl radicals are derived from carboxylic acids with radicals containing only hydrogen and carbon atoms, attached in position 3
    • Y—GENERAL TAGGING OF NEW TECHNOLOGICAL DEVELOPMENTS; GENERAL TAGGING OF CROSS-SECTIONAL TECHNOLOGIES SPANNING OVER SEVERAL SECTIONS OF THE IPC; TECHNICAL SUBJECTS COVERED BY FORMER USPC CROSS-REFERENCE ART COLLECTIONS [XRACs] AND DIGESTS
    • Y02—TECHNOLOGIES OR APPLICATIONS FOR MITIGATION OR ADAPTATION AGAINST CLIMATE CHANGE
    • Y02P—CLIMATE CHANGE MITIGATION TECHNOLOGIES IN THE PRODUCTION OR PROCESSING OF GOODS
    • Y02P20/00—Technologies relating to chemical industry
    • Y02P20/50—Improvements relating to the production of bulk chemicals
    • Y02P20/55—Design of synthesis routes, e.g. reducing the use of auxiliary or protecting groups

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Cephalosporin Compounds (AREA)
KR1019860003085A 1985-04-22 1986-04-22 7-아미노-3- 프로페닐 세팔로스포란산 및 그 에스텔 Ceased KR860008189A (ko)

Priority Applications (1)

Application Number Priority Date Filing Date Title
KR1019900002094A KR900004930B1 (ko) 1985-04-22 1990-02-21 7-아미노-3-프로페닐 세팔로스포란산 및 그 에스텔의 제조방법

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
US72587185A 1985-04-22 1985-04-22
US725,871 1985-04-22

Related Child Applications (1)

Application Number Title Priority Date Filing Date
KR1019900002094A Division KR900004930B1 (ko) 1985-04-22 1990-02-21 7-아미노-3-프로페닐 세팔로스포란산 및 그 에스텔의 제조방법

Publications (1)

Publication Number Publication Date
KR860008189A true KR860008189A (ko) 1986-11-12

Family

ID=24916301

Family Applications (1)

Application Number Title Priority Date Filing Date
KR1019860003085A Ceased KR860008189A (ko) 1985-04-22 1986-04-22 7-아미노-3- 프로페닐 세팔로스포란산 및 그 에스텔

Country Status (38)

Country Link
JP (1) JPS61249989A (enrdf_load_stackoverflow)
KR (1) KR860008189A (enrdf_load_stackoverflow)
CN (1) CN1015714B (enrdf_load_stackoverflow)
AR (1) AR242581A1 (enrdf_load_stackoverflow)
AT (1) AT392072B (enrdf_load_stackoverflow)
AU (1) AU589170B2 (enrdf_load_stackoverflow)
BE (1) BE904646A (enrdf_load_stackoverflow)
CA (1) CA1273629A (enrdf_load_stackoverflow)
CH (1) CH671399A5 (enrdf_load_stackoverflow)
CS (1) CS270435B2 (enrdf_load_stackoverflow)
CY (1) CY1571A (enrdf_load_stackoverflow)
DD (1) DD244557A5 (enrdf_load_stackoverflow)
DE (1) DE3613365A1 (enrdf_load_stackoverflow)
DK (1) DK163584C (enrdf_load_stackoverflow)
EG (1) EG18001A (enrdf_load_stackoverflow)
ES (1) ES8800236A1 (enrdf_load_stackoverflow)
FI (1) FI84268C (enrdf_load_stackoverflow)
FR (1) FR2580652B1 (enrdf_load_stackoverflow)
GB (1) GB2173798B (enrdf_load_stackoverflow)
GR (1) GR861065B (enrdf_load_stackoverflow)
HK (1) HK106290A (enrdf_load_stackoverflow)
HU (1) HU195223B (enrdf_load_stackoverflow)
IE (1) IE59014B1 (enrdf_load_stackoverflow)
IT (1) IT1228241B (enrdf_load_stackoverflow)
LU (1) LU86402A1 (enrdf_load_stackoverflow)
MY (1) MY100694A (enrdf_load_stackoverflow)
NL (1) NL192205C (enrdf_load_stackoverflow)
NO (1) NO164659C (enrdf_load_stackoverflow)
NZ (1) NZ215717A (enrdf_load_stackoverflow)
OA (1) OA08245A (enrdf_load_stackoverflow)
PT (1) PT82436B (enrdf_load_stackoverflow)
SE (1) SE500217C2 (enrdf_load_stackoverflow)
SG (1) SG90890G (enrdf_load_stackoverflow)
SU (1) SU1435155A3 (enrdf_load_stackoverflow)
YU (1) YU43697B (enrdf_load_stackoverflow)
ZA (1) ZA862985B (enrdf_load_stackoverflow)
ZM (1) ZM4286A1 (enrdf_load_stackoverflow)
ZW (1) ZW9086A1 (enrdf_load_stackoverflow)

Families Citing this family (12)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US4708955A (en) * 1985-06-24 1987-11-24 Bristol-Myers Company 3-(substituted)propenyl-7-aminothiazol-ylcephalosporanic acids and esters thereof
US4870168A (en) * 1987-02-26 1989-09-26 Bristol-Myers Company 3-Unsaturated alkyl cephems from 3-triflyl cephems
DE3933934A1 (de) * 1989-10-03 1991-04-11 Bayer Ag Verfahren zur herstellung von 7-amino-3-((z)-1-propen-1-yl)-3-cephem-4-carbonsaeure
DK0503453T3 (da) * 1991-03-08 2001-07-16 Biochemie Gmbh Fremgangsmåde til fremstilling af cephalosporiner og mellemprodukter i denne fremgangsmåde
DK0630380T3 (da) * 1992-02-05 2001-12-10 Biochemie Gmbh Fremgangsmåde til rensning af et 3-cephem-4-carboxylsyrederivat
AT399876B (de) * 1992-02-05 1995-08-25 Biochemie Gmbh Verfahren zur abreicherung von 7-amino-3-((e)-1- propen-1-yl)-3-cephem-4-carbonsäure
JPH07173168A (ja) * 1993-07-14 1995-07-11 Sumitomo Chem Co Ltd セフェム系化合物、その製法、およびそれのセフェム系抗生物質製造への利用
US20060173176A1 (en) * 2002-10-08 2006-08-03 Yatendra Kumar Process for the preparation of (z)-isomer enriched 7-amino-3-propen-1-yl-3-cephem-4-carboxylic acid
US7544797B2 (en) 2003-10-30 2009-06-09 Cj Cheiljedang Corporation Processes for the preparation of cephem derivatives
JP4046708B2 (ja) * 2004-06-04 2008-02-13 明治製菓株式会社 ３−アルケニルセフェム化合物の製造方法
ATE457990T1 (de) 2004-11-01 2010-03-15 Hetero Drugs Ltd Neues verfahren zur herstellung eines cefprozil- zwischenprodukts
CN103183686B (zh) * 2011-12-30 2016-06-29 浙江新和成股份有限公司 7β-氨基-7α-甲氧基-3-头孢烯化合物的制备方法

Family Cites Families (7)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US3769277A (en) * 1970-01-23 1973-10-30 Glaxo Lab Ltd Preparation of delta3-4 carboxy cephalosporins having a 3-vinyl or substituted 3-vinyl group
US4110534A (en) * 1970-01-23 1978-08-29 Glaxo Laboratories Limited Process for the preparation of 3-vinyl and substituted vinyl cephalosporins
GB1342241A (en) * 1970-01-23 1974-01-03 Glaxo Lab Ltd Cephalosporin compounds
US4065620A (en) * 1971-06-14 1977-12-27 Eli Lilly And Company 3-(Substituted) vinyl cephalosporins
US4409214A (en) * 1979-11-19 1983-10-11 Fujisawa Pharmaceutical, Co., Ltd. 7-Acylamino-3-vinylcephalosporanic acid derivatives and processes for the preparation thereof
US4520022A (en) * 1983-01-28 1985-05-28 Bristol-Myers Company Substituted vinyl cephalosporins
AU566944B2 (en) * 1983-10-07 1987-11-05 Gist-Brocades N.V. Preparation of 3-cephem derivatives

Also Published As

Publication number Publication date
DE3613365C2 (enrdf_load_stackoverflow) 1989-06-15
AR242581A1 (es) 1993-04-30
JPS61249989A (ja) 1986-11-07
ES8800236A1 (es) 1987-10-16
CN86102630A (zh) 1987-02-04
HU195223B (en) 1988-04-28
ATA106786A (de) 1990-07-15
SE500217C2 (sv) 1994-05-09
IE861048L (en) 1986-10-22
NZ215717A (en) 1989-06-28
DE3613365A1 (de) 1987-01-02
JPH0327554B2 (enrdf_load_stackoverflow) 1991-04-16
IT8620162A0 (it) 1986-04-21
DK163584C (da) 1992-08-10
FR2580652B1 (fr) 1989-01-06
ZA862985B (en) 1986-12-30
YU43697B (en) 1989-10-31
FR2580652A1 (fr) 1986-10-24
DK182486D0 (da) 1986-04-21
SE8601825D0 (sv) 1986-04-21
CS287286A2 (en) 1989-11-14
FI861634L (fi) 1986-10-23
PT82436B (pt) 1988-11-30
SE8601825L (sv) 1986-10-23
DK163584B (da) 1992-03-16
YU65986A (en) 1987-12-31
GB2173798A (en) 1986-10-22
NL192205B (nl) 1996-11-01
NO164659C (no) 1990-10-31
DD244557A5 (de) 1987-04-08
AU589170B2 (en) 1989-10-05
IT1228241B (it) 1991-06-05
OA08245A (fr) 1987-10-30
CS270435B2 (en) 1990-06-13
BE904646A (fr) 1986-10-21
HK106290A (en) 1990-12-28
NL192205C (nl) 1997-03-04
AU5616886A (en) 1986-11-06
LU86402A1 (fr) 1986-11-05
IE59014B1 (en) 1993-12-15
NL8601011A (nl) 1986-11-17
SU1435155A3 (ru) 1988-10-30
SG90890G (en) 1991-01-18
PT82436A (en) 1986-05-01
FI84268C (fi) 1991-11-11
NO164659B (no) 1990-07-23
FI861634A0 (fi) 1986-04-17
GB2173798B (en) 1988-11-30
DK182486A (da) 1986-10-23
GB8609661D0 (en) 1986-05-29
HUT41033A (en) 1987-03-30
CH671399A5 (enrdf_load_stackoverflow) 1989-08-31
AT392072B (de) 1991-01-25
CY1571A (en) 1991-12-20
CN1015714B (zh) 1992-03-04
MY100694A (en) 1991-01-17
FI84268B (fi) 1991-07-31
NO861430L (no) 1986-10-23
ZM4286A1 (en) 1989-03-27
EG18001A (en) 1991-11-30
ZW9086A1 (en) 1986-12-03
ES554215A0 (es) 1987-10-16
CA1273629A (en) 1990-09-04
GR861065B (en) 1986-09-01

Similar Documents

Publication Publication Date Title
US4614614A (en) Process for the manufacture of optically active azetidinones
KR860008189A (ko) 7-아미노-3- 프로페닐 세팔로스포란산 및 그 에스텔
KR840007876A (ko) 아크릴산 아미드의 제조방법
KR830001947A (ko) 화합물의 제조방법
HUT35649A (en) Process for preparing substituted 2-mercapto-imidazoles
ATE126230T1 (de) Cephalosporinderivate und verfahren zur herstellung von cephem-verbindungen.
KR840005463A (ko) Omt의 c-23-변형유도체의 제조방법
DK95280A (da) Brom-substituerede deacetoxycephalosporiner og fremgangsmaade til fremstilling heraf
MY130320A (en) 1-bromoethyl ethyl carbonate and its use in the preparation of 1''- ethoxycarbonyloxyethyl esters of penicillins and novel intermediates, methods for its preparation and 1-bromoethylchloroformate and 1-bromoethylbromoformate obtained as intermediates
EP0140437A3 (en) Substituted azetidine derivatives, process for their preparation, and their use as intermediates
US4176231A (en) Process for preparing 3-exomethylenecepham sulfoxides
KR840006663A (ko) 1-옥사-β-락탐의 제조방법
EP0117872A1 (en) Process for preparing cephalosporin compounds
CA2037688A1 (en) Organo cuprate process for cefprozil
GB1479802A (en) Process for preparing cephalosporins
KR850002105A (ko) 3-아지도세팔포스포린의 제조방법
CA1252466A (en) METHOD FOR THE PREPARATION OF 1,2,5,6-TETRAHYDRO-4H-PYRROLO[3,2,1-1J]-QUINOLIN-4-ONE; 5-HALOGENO-1,2,3-(1,2-DIHYDROPYRROLO)-4-QUINOLONES, INTERMEDIATE PRODUCTS FOR THIS PREPARATION
RU93029051A (ru) Способ получения n-/циклогексилтио/фталимида
KR870000526B1 (ko) 아제티디논 설핀산의 제조방법
JPH043400B2 (enrdf_load_stackoverflow)
EP0122002A1 (en) Process for preparing azetidinone derivatives
KR830007677A (ko) 1,3-티아졸리딘-4-일-카복실산 유도체의 제조방법
KR850007599A (ko) 3-아지노메틸 리파마이신의 제조방법
GB1312030A (en) Penicillin compounds and a method of synthesising same
KR900011777A (ko) 신규한 아미노 카르복실산 유도체

Legal Events

Date Code Title Description
PA0109 Patent application

Patent event code: PA01091R01D

Comment text: Patent Application

Patent event date: 19860422

PG1501 Laying open of application
A201 Request for examination
PA0201 Request for examination

Patent event code: PA02012R01D

Patent event date: 19870825

Comment text: Request for Examination of Application

Patent event code: PA02011R01I

Patent event date: 19860422

Comment text: Patent Application

E902 Notification of reason for refusal
PE0902 Notice of grounds for rejection

Comment text: Notification of reason for refusal

Patent event date: 19890617

Patent event code: PE09021S01D

E601 Decision to refuse application
PE0601 Decision on rejection of patent

Patent event date: 19900119

Comment text: Decision to Refuse Application

Patent event code: PE06012S01D

Patent event date: 19890617

Comment text: Notification of reason for refusal

Patent event code: PE06011S01I

J2X1 Appeal (before the patent court)

Free format text: APPEAL AGAINST DECISION TO DECLINE REFUSAL

PJ2001 Appeal

Appeal kind category: Appeal against decision to decline refusal

Decision date: 19910430

Appeal identifier: 1990201000194

Request date: 19900221