JP4284071B2 - イソインドール−イミド化合物、組成物、およびそれらの使用 - Google Patents

イソインドール−イミド化合物、組成物、およびそれらの使用 Download PDF

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JP4284071B2
JP4284071B2 JP2002559408A JP2002559408A JP4284071B2 JP 4284071 B2 JP4284071 B2 JP 4284071B2 JP 2002559408 A JP2002559408 A JP 2002559408A JP 2002559408 A JP2002559408 A JP 2002559408A JP 4284071 B2 JP4284071 B2 JP 4284071B2
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Prior art keywords
alkyl
dioxo
mmol
piperidyl
methyl
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JP2004525889A (ja
JP2004525889A5 (US20030045552A1-20030306-C00110.png
Inventor
ロバージ,マイケル,ジェイ.
チェン,ロジャー,シェン−チュウ
ミュラー,ジョージ,ダブリュー.
マン,ホン−ワー
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Celgene Corp
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Celgene Corp
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    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D401/00Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom
    • C07D401/02Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings
    • C07D401/04Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings directly linked by a ring-member-to-ring-member bond
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/33Heterocyclic compounds
    • A61K31/395Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/435Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom
    • A61K31/44Non condensed pyridines; Hydrogenated derivatives thereof
    • AHUMAN NECESSITIES
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    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
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    • A61P1/00Drugs for disorders of the alimentary tract or the digestive system
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    • YGENERAL TAGGING OF NEW TECHNOLOGICAL DEVELOPMENTS; GENERAL TAGGING OF CROSS-SECTIONAL TECHNOLOGIES SPANNING OVER SEVERAL SECTIONS OF THE IPC; TECHNICAL SUBJECTS COVERED BY FORMER USPC CROSS-REFERENCE ART COLLECTIONS [XRACs] AND DIGESTS
    • Y02TECHNOLOGIES OR APPLICATIONS FOR MITIGATION OR ADAPTATION AGAINST CLIMATE CHANGE
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    • Y02A50/30Against vector-borne diseases, e.g. mosquito-borne, fly-borne, tick-borne or waterborne diseases whose impact is exacerbated by climate change
JP2002559408A 2000-12-27 2001-12-21 イソインドール−イミド化合物、組成物、およびそれらの使用 Expired - Fee Related JP4284071B2 (ja)

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
US25837200P 2000-12-27 2000-12-27
US09/972,487 US20030045552A1 (en) 2000-12-27 2001-10-05 Isoindole-imide compounds, compositions, and uses thereof
PCT/US2001/050401 WO2002059106A1 (en) 2000-12-27 2001-12-21 Isoindole-imide compounds, compositions, and uses thereof

Related Child Applications (1)

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JP2005321049A Division JP4648822B2 (ja) 2000-12-27 2005-11-04 イソインドール−イミド化合物、組成物、およびそれらの使用

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JP2004525889A JP2004525889A (ja) 2004-08-26
JP2004525889A5 JP2004525889A5 (US20030045552A1-20030306-C00110.png) 2006-01-05
JP4284071B2 true JP4284071B2 (ja) 2009-06-24

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JP2002559408A Expired - Fee Related JP4284071B2 (ja) 2000-12-27 2001-12-21 イソインドール−イミド化合物、組成物、およびそれらの使用
JP2005321049A Expired - Fee Related JP4648822B2 (ja) 2000-12-27 2005-11-04 イソインドール−イミド化合物、組成物、およびそれらの使用
JP2010110388A Pending JP2010195824A (ja) 2000-12-27 2010-05-12 イソインドール−イミド化合物、組成物、およびそれらの使用

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JP2010110388A Pending JP2010195824A (ja) 2000-12-27 2010-05-12 イソインドール−イミド化合物、組成物、およびそれらの使用

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US (1) US20030045552A1 (US20030045552A1-20030306-C00110.png)
EP (3) EP1767533A1 (US20030045552A1-20030306-C00110.png)
JP (3) JP4284071B2 (US20030045552A1-20030306-C00110.png)
KR (4) KR20070026879A (US20030045552A1-20030306-C00110.png)
AT (1) ATE352548T1 (US20030045552A1-20030306-C00110.png)
AU (3) AU2002248252B2 (US20030045552A1-20030306-C00110.png)
CA (1) CA2433021C (US20030045552A1-20030306-C00110.png)
CY (1) CY1106423T1 (US20030045552A1-20030306-C00110.png)
CZ (1) CZ20032041A3 (US20030045552A1-20030306-C00110.png)
DE (1) DE60126344T2 (US20030045552A1-20030306-C00110.png)
DK (1) DK1363900T3 (US20030045552A1-20030306-C00110.png)
ES (1) ES2275758T3 (US20030045552A1-20030306-C00110.png)
HK (1) HK1061396A1 (US20030045552A1-20030306-C00110.png)
HU (1) HU229003B1 (US20030045552A1-20030306-C00110.png)
IL (2) IL156646A0 (US20030045552A1-20030306-C00110.png)
MX (1) MXPA03005786A (US20030045552A1-20030306-C00110.png)
NZ (1) NZ526893A (US20030045552A1-20030306-C00110.png)
PT (1) PT1363900E (US20030045552A1-20030306-C00110.png)
WO (1) WO2002059106A1 (US20030045552A1-20030306-C00110.png)
ZA (1) ZA200305759B (US20030045552A1-20030306-C00110.png)

Cited By (1)

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