JP2014509647A5 - - Google Patents

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JP2014509647A5
JP2014509647A5 JP2014502668A JP2014502668A JP2014509647A5 JP 2014509647 A5 JP2014509647 A5 JP 2014509647A5 JP 2014502668 A JP2014502668 A JP 2014502668A JP 2014502668 A JP2014502668 A JP 2014502668A JP 2014509647 A5 JP2014509647 A5 JP 2014509647A5
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Japan
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heterocyclyl
aryl
alkyl
compound
heteroaryl
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JP2014502668A
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Japanese (ja)
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JP6042406B2 (ja
JP2014509647A (ja
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Priority claimed from PCT/US2012/030640 external-priority patent/WO2012135160A1/en
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JP2014502668A 2011-03-28 2012-03-27 （α−置換アラルキルアミノ及びヘテロアリールアルキルアミノ）ピリミジニル及び１，３，５−トリアジニルベンズイミダゾール、それらを含む医薬組成物、並びに増殖性疾患の治療で使用するためのこれらの化合物 Active JP6042406B2 (ja)

Applications Claiming Priority (7)

Application Number Priority Date Filing Date Title
US201161468502P 2011-03-28 2011-03-28
US61/468,502 2011-03-28
US201161530859P 2011-09-02 2011-09-02
US61/530,859 2011-09-02
US201161560699P 2011-11-16 2011-11-16
US61/560,699 2011-11-16
PCT/US2012/030640 WO2012135160A1 (en) 2011-03-28 2012-03-27 (alpha- substituted aralkylamino and heteroarylalkylamino) pyrimidinyl and 1,3,5 -triazinyl benzimidazoles, pharmaceutical compositions containing them, and these compounds for use in treating proliferative diseases

Publications (3)

Publication Number Publication Date
JP2014509647A JP2014509647A (ja) 2014-04-21
JP2014509647A5 true JP2014509647A5 (enExample) 2015-05-14
JP6042406B2 JP6042406B2 (ja) 2016-12-14

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JP2014502668A Active JP6042406B2 (ja) 2011-03-28 2012-03-27 （α−置換アラルキルアミノ及びヘテロアリールアルキルアミノ）ピリミジニル及び１，３，５−トリアジニルベンズイミダゾール、それらを含む医薬組成物、並びに増殖性疾患の治療で使用するためのこれらの化合物

Country Status (17)

Country Link
US (6) US9056852B2 (enExample)
EP (1) EP2691384B1 (enExample)
JP (1) JP6042406B2 (enExample)
KR (1) KR101940831B1 (enExample)
CN (2) CN107501241B (enExample)
AU (2) AU2012236834B2 (enExample)
BR (1) BR112013024907A2 (enExample)
CA (1) CA2831582C (enExample)
DK (1) DK2691384T3 (enExample)
ES (1) ES2608967T3 (enExample)
IL (1) IL228600B (enExample)
MX (1) MX345238B (enExample)
RU (1) RU2608742C2 (enExample)
SG (1) SG193982A1 (enExample)
TW (1) TWI572599B (enExample)
WO (1) WO2012135160A1 (enExample)
ZA (1) ZA201307224B (enExample)

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US11236079B2 (en) * 2018-04-10 2022-02-01 Neuropore Therapies, Inc. Morpholine derivates as inhibitors of Vps34
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JP2021534116A (ja) * 2018-08-14 2021-12-09 エムイーアイ ファーマ，インク． 再発性の濾胞性リンパ腫の処置
WO2020036995A1 (en) * 2018-08-14 2020-02-20 Mei Pharma, Inc. Combination therapy
WO2020036999A1 (en) * 2018-08-14 2020-02-20 Mei Pharma, Inc. Treatment of b cell malignancies
BR112021007830A2 (pt) * 2018-11-20 2021-08-03 Bayer Aktiengesellschaft antagonistas do adrenoceptor-alfa2 do subtipo c (al-fa-2c) para o tratamento da apneia do sono
TW202038945A (zh) * 2018-12-21 2020-11-01 美商梅製藥公司 組合療法
MX2022012339A (es) * 2020-04-07 2022-10-27 Mei Pharma Inc Preparacion de un 1,3,5-triazinil benzimidazol.
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