AU2012236834B2 - (alpha- substituted aralkylamino and heteroarylalkylamino) pyrimidinyl and 1,3,5 -triazinyl benzimidazoles, pharmaceutical compositions containing them, and these compounds for use in treating proliferative diseases - Google Patents

(alpha- substituted aralkylamino and heteroarylalkylamino) pyrimidinyl and 1,3,5 -triazinyl benzimidazoles, pharmaceutical compositions containing them, and these compounds for use in treating proliferative diseases Download PDF

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AU2012236834B2
AU2012236834B2 AU2012236834A AU2012236834A AU2012236834B2 AU 2012236834 B2 AU2012236834 B2 AU 2012236834B2 AU 2012236834 A AU2012236834 A AU 2012236834A AU 2012236834 A AU2012236834 A AU 2012236834A AU 2012236834 B2 AU2012236834 B2 AU 2012236834B2
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hydrogen
substituents
optionally substituted
certain embodiments
alkyl
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AU2012236834A1 (en
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S. David Brown
David J. Matthews
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Lite Strategy Inc
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Mei Pharma Inc
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    • A61K31/535—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with at least one nitrogen and one oxygen as the ring hetero atoms, e.g. 1,2-oxazines
    • A61K31/5375—1,4-Oxazines, e.g. morpholine
    • A61K31/5377—1,4-Oxazines, e.g. morpholine not condensed and containing further heterocyclic rings, e.g. timolol
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AU2012236834A 2011-03-28 2012-03-27 (alpha- substituted aralkylamino and heteroarylalkylamino) pyrimidinyl and 1,3,5 -triazinyl benzimidazoles, pharmaceutical compositions containing them, and these compounds for use in treating proliferative diseases Active AU2012236834B2 (en)

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AU2016201558A AU2016201558B2 (en) 2011-03-28 2016-03-10 (alpha- substituted aralkylamino and heteroarylalkylamino) pyrimidinyl and 1,3,5 -triazinyl benzimidazoles, pharmaceutical compositions containing them, and these compounds for use in treating proliferative diseases

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Application Number Priority Date Filing Date Title
US201161468502P 2011-03-28 2011-03-28
US61/468,502 2011-03-28
US201161530859P 2011-09-02 2011-09-02
US61/530,859 2011-09-02
US201161560699P 2011-11-16 2011-11-16
US61/560,699 2011-11-16
PCT/US2012/030640 WO2012135160A1 (en) 2011-03-28 2012-03-27 (alpha- substituted aralkylamino and heteroarylalkylamino) pyrimidinyl and 1,3,5 -triazinyl benzimidazoles, pharmaceutical compositions containing them, and these compounds for use in treating proliferative diseases

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AU2012236834B2 true AU2012236834B2 (en) 2015-12-10

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AU2016201558A Active AU2016201558B2 (en) 2011-03-28 2016-03-10 (alpha- substituted aralkylamino and heteroarylalkylamino) pyrimidinyl and 1,3,5 -triazinyl benzimidazoles, pharmaceutical compositions containing them, and these compounds for use in treating proliferative diseases

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