JP2013502424A5 - - Google Patents
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- JP2013502424A5 JP2013502424A5 JP2012525652A JP2012525652A JP2013502424A5 JP 2013502424 A5 JP2013502424 A5 JP 2013502424A5 JP 2012525652 A JP2012525652 A JP 2012525652A JP 2012525652 A JP2012525652 A JP 2012525652A JP 2013502424 A5 JP2013502424 A5 JP 2013502424A5
- Authority
- JP
- Japan
- Prior art keywords
- alkyl
- alkenyl
- alkynyl
- group
- saturated
- Prior art date
- Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
- Ceased
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- 0 C*CCC(*c1cnc(*)cc1)*I Chemical compound C*CCC(*c1cnc(*)cc1)*I 0.000 description 2
Applications Claiming Priority (3)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| US27210109P | 2009-08-17 | 2009-08-17 | |
| US61/272,101 | 2009-08-17 | ||
| PCT/US2010/045817 WO2011022440A2 (en) | 2009-08-17 | 2010-08-17 | Heat shock protein binding compounds, compositions, and methods for making and using same |
Related Child Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| JP2015160345A Division JP6465774B2 (ja) | 2009-08-17 | 2015-08-17 | 熱ショックタンパク質結合化合物、組成物、およびそれらを製造するための方法 |
Publications (2)
| Publication Number | Publication Date |
|---|---|
| JP2013502424A JP2013502424A (ja) | 2013-01-24 |
| JP2013502424A5 true JP2013502424A5 (https=) | 2013-10-03 |
Family
ID=43607564
Family Applications (3)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| JP2012525652A Ceased JP2013502424A (ja) | 2009-08-17 | 2010-08-17 | 熱ショックタンパク質結合化合物、組成物、およびそれらを製造するための方法 |
| JP2015160345A Expired - Fee Related JP6465774B2 (ja) | 2009-08-17 | 2015-08-17 | 熱ショックタンパク質結合化合物、組成物、およびそれらを製造するための方法 |
| JP2018158360A Withdrawn JP2018188476A (ja) | 2009-08-17 | 2018-08-27 | 熱ショックタンパク質結合化合物、組成物、ならびにそれらを製造および使用するための方法 |
Family Applications After (2)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| JP2015160345A Expired - Fee Related JP6465774B2 (ja) | 2009-08-17 | 2015-08-17 | 熱ショックタンパク質結合化合物、組成物、およびそれらを製造するための方法 |
| JP2018158360A Withdrawn JP2018188476A (ja) | 2009-08-17 | 2018-08-27 | 熱ショックタンパク質結合化合物、組成物、ならびにそれらを製造および使用するための方法 |
Country Status (13)
| Country | Link |
|---|---|
| US (3) | US9567318B2 (https=) |
| EP (2) | EP3205647B1 (https=) |
| JP (3) | JP2013502424A (https=) |
| KR (1) | KR101906146B1 (https=) |
| CN (2) | CN108752280A (https=) |
| AU (1) | AU2010284255B2 (https=) |
| BR (1) | BR112012003637A2 (https=) |
| CA (1) | CA2771190C (https=) |
| EA (1) | EA201290062A1 (https=) |
| ES (2) | ES2608670T3 (https=) |
| MX (1) | MX353747B (https=) |
| NZ (3) | NZ713361A (https=) |
| WO (1) | WO2011022440A2 (https=) |
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| US20050070712A1 (en) * | 2003-09-26 | 2005-03-31 | Christi Kosogof | Pyrimidine derivatives as ghrelin receptor modulators |
| CA2557372C (en) | 2004-03-05 | 2013-01-08 | F. Hoffmann-La Roche Ag | Diaminopyrimidines as p2x3 and p2x2/3 antagonists |
| JP4906715B2 (ja) * | 2004-05-08 | 2012-03-28 | ニューロジェン・コーポレーション | ４，５−ジ置換−２−アリールピリミジン類 |
| JP2008533166A (ja) * | 2005-03-16 | 2008-08-21 | ターゲジェン インコーポレーティッド | ピリミジン化合物および使用法 |
| ES2562056T3 (es) | 2005-09-01 | 2016-03-02 | F. Hoffmann-La Roche Ag | Diaminopirimidinas como moduladores P2X3 y P2X2/3 |
| WO2007131034A1 (en) | 2006-05-03 | 2007-11-15 | The Regents Of The University Of Michigan | Pyrimidone derivatives which are modulators of heat shock protein (hsp) 70 |
| JP2008081492A (ja) * | 2006-08-31 | 2008-04-10 | Banyu Pharmaceut Co Ltd | オーロラａ選択的阻害作用を有する新規アミノピリジン誘導体 |
| US20080124407A1 (en) | 2006-10-10 | 2008-05-29 | University Of Washington | Inhibiting cyp3a4 induction |
| EA017405B9 (ru) | 2006-12-08 | 2014-05-30 | АйАрЭм ЭлЭлСи | Соединения и композиции в качестве ингибиторов протеинкиназы |
| PT2114900T (pt) * | 2007-01-31 | 2019-01-17 | Ym Biosciences Australia Pty | Compostos à base de tiopirimidina e as suas utilizações |
| TW200911240A (en) | 2007-06-11 | 2009-03-16 | Kyowa Hakko Kogyo Kk | Anti-tumor agent |
| WO2009023846A2 (en) * | 2007-08-15 | 2009-02-19 | The Research Foundation Of State University Of New York | Methods for heat shock protein dependent cancer treatment |
| WO2009061345A2 (en) | 2007-11-07 | 2009-05-14 | Cornell Research Foundation, Inc. | Targeting cdk4 and cdk6 in cancer therapy |
| PE20091236A1 (es) * | 2007-11-22 | 2009-09-16 | Astrazeneca Ab | Derivados de pirimidina como immunomoduladores de tlr7 |
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| NZ713361A (en) | 2009-08-17 | 2017-06-30 | Memorial Sloan Kettering Cancer Center | Heat shock protein binding compounds, compositions, and methods for making and using same |
| WO2014078294A1 (en) | 2012-11-13 | 2014-05-22 | Memorial Sloan-Kettering Cancer Center | Indole compounds and their use as antimicrobials |
| JP6607870B2 (ja) | 2014-05-13 | 2019-11-20 | メモリアル スローン ケタリング キャンサー センター | Ｈｓｐ７０モジュレーターならびにその作製および使用方法 |
| WO2016203405A1 (en) | 2015-06-19 | 2016-12-22 | Novartis Ag | Compounds and compositions for inhibiting the activity of shp2 |
| CA2998753A1 (en) | 2015-09-18 | 2017-03-23 | St. Jude Children's Research Hospital | Methods and compositions of inhibiting dcn1-ubc12 interaction |
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2010
- 2010-08-17 NZ NZ713361A patent/NZ713361A/en not_active IP Right Cessation
- 2010-08-17 NZ NZ623069A patent/NZ623069A/en not_active IP Right Cessation
- 2010-08-17 AU AU2010284255A patent/AU2010284255B2/en not_active Ceased
- 2010-08-17 NZ NZ59826210A patent/NZ598262A/en not_active IP Right Cessation
- 2010-08-17 CN CN201810695781.9A patent/CN108752280A/zh active Pending
- 2010-08-17 ES ES10810519.8T patent/ES2608670T3/es active Active
- 2010-08-17 MX MX2012001993A patent/MX353747B/es active IP Right Grant
- 2010-08-17 BR BR112012003637A patent/BR112012003637A2/pt not_active IP Right Cessation
- 2010-08-17 CN CN2010800368189A patent/CN102753177A/zh active Pending
- 2010-08-17 CA CA2771190A patent/CA2771190C/en not_active Expired - Fee Related
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- 2010-08-17 KR KR1020127006838A patent/KR101906146B1/ko not_active Expired - Fee Related
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- 2010-08-17 EA EA201290062A patent/EA201290062A1/ru unknown
- 2010-08-17 JP JP2012525652A patent/JP2013502424A/ja not_active Ceased
- 2010-08-17 WO PCT/US2010/045817 patent/WO2011022440A2/en not_active Ceased
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