JP2011523628A - 有効なコンジュゲートおよび親水性リンカー - Google Patents

有効なコンジュゲートおよび親水性リンカー Download PDF

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JP2011523628A
JP2011523628A JP2011507633A JP2011507633A JP2011523628A JP 2011523628 A JP2011523628 A JP 2011523628A JP 2011507633 A JP2011507633 A JP 2011507633A JP 2011507633 A JP2011507633 A JP 2011507633A JP 2011523628 A JP2011523628 A JP 2011523628A
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bond
antibody
cell
conjugate
binding agent
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JP2011523628A5 (enExample
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シン,ラジーヴァ
コヴトゥン,エレーナ
ウィルヘルム,シャロン・ディー
チャリ,ラビ・ヴイ・ジェイ
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イミュノジェン・インコーポレーテッド
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    • A61K31/395Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/535Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with at least one nitrogen and one oxygen as the ring hetero atoms, e.g. 1,2-oxazines
    • A61K31/53751,4-Oxazines, e.g. morpholine
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