JP2010528027A - Ｐｉ３キナーゼ阻害物質としてのキノリン誘導体 - Google Patents

Ｐｉ３キナーゼ阻害物質としてのキノリン誘導体 Download PDF

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JP2010528027A
JP2010528027A JP2010509463A JP2010509463A JP2010528027A JP 2010528027 A JP2010528027 A JP 2010528027A JP 2010509463 A JP2010509463 A JP 2010509463A JP 2010509463 A JP2010509463 A JP 2010509463A JP 2010528027 A JP2010528027 A JP 2010528027A
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pyridinyl
substituted
quinolinyl
cancer
group
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Japanese (ja)
Inventor
ニコラス・ディ・アダムス
アミタ・エム・チョーダリ
カーラ・エイ・ドナテリ
スティーブン・デイビッド・ナイト
ケネス・アレン・ニューランダー
シンシア・エイ・パリッシュ
ランス・リジャース
マーサ・エイ・サーポング
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GlaxoSmithKline LLC
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GlaxoSmithKline LLC
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    • A61K31/435—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom
    • A61K31/47—Quinolines; Isoquinolines
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JP2010509463A 2007-05-18 2008-05-16 Ｐｉ３キナーゼ阻害物質としてのキノリン誘導体 Pending JP2010528027A (ja)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
US93876107P 2007-05-18 2007-05-18
PCT/US2008/063821 WO2008144464A1 (en) 2007-05-18 2008-05-16 Quinoline derivatives as p13 kinase inhibitors

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