JP2010504973A5 - - Google Patents
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- JP2010504973A5 JP2010504973A5 JP2009530406A JP2009530406A JP2010504973A5 JP 2010504973 A5 JP2010504973 A5 JP 2010504973A5 JP 2009530406 A JP2009530406 A JP 2009530406A JP 2009530406 A JP2009530406 A JP 2009530406A JP 2010504973 A5 JP2010504973 A5 JP 2010504973A5
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- 208000037265 diseases, disorders, signs and symptoms Diseases 0.000 claims 10
- 208000035475 disorder Diseases 0.000 claims 8
- 239000008194 pharmaceutical composition Substances 0.000 claims 3
- 201000010099 disease Diseases 0.000 claims 2
- 201000001320 Atherosclerosis Diseases 0.000 claims 1
- 208000029462 Immunodeficiency disease Diseases 0.000 claims 1
- 208000019693 Lung disease Diseases 0.000 claims 1
- 206010028980 Neoplasm Diseases 0.000 claims 1
- 208000030852 Parasitic disease Diseases 0.000 claims 1
- 108060008682 Tumor Necrosis Factor Proteins 0.000 claims 1
- 102000000852 Tumor Necrosis Factor-alpha Human genes 0.000 claims 1
- 230000002159 abnormal effect Effects 0.000 claims 1
- 239000013543 active substance Substances 0.000 claims 1
- 230000033115 angiogenesis Effects 0.000 claims 1
- 239000010425 asbestos Substances 0.000 claims 1
- 201000011510 cancer Diseases 0.000 claims 1
- 208000015114 central nervous system disease Diseases 0.000 claims 1
- 150000001875 compounds Chemical class 0.000 claims 1
- 230000006378 damage Effects 0.000 claims 1
- 208000002780 macular degeneration Diseases 0.000 claims 1
- 229910052895 riebeckite Inorganic materials 0.000 claims 1
- 150000003839 salts Chemical class 0.000 claims 1
- 208000017520 skin disease Diseases 0.000 claims 1
- 239000012453 solvate Substances 0.000 claims 1
- 208000011580 syndromic disease Diseases 0.000 claims 1
Applications Claiming Priority (3)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| US84747106P | 2006-09-26 | 2006-09-26 | |
| US60/847,471 | 2006-09-26 | ||
| PCT/US2007/020765 WO2008039489A2 (en) | 2006-09-26 | 2007-09-25 | 5-substituted quinazolinone derivatives as antitumor agents |
Related Child Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| JP2013210802A Division JP5901599B2 (ja) | 2006-09-26 | 2013-10-08 | ５−置換キナゾリノン誘導体、それを含む組成物、及びその使用方法 |
Publications (3)
| Publication Number | Publication Date |
|---|---|
| JP2010504973A JP2010504973A (ja) | 2010-02-18 |
| JP2010504973A5 true JP2010504973A5 (enExample) | 2010-11-18 |
| JP5388854B2 JP5388854B2 (ja) | 2014-01-15 |
Family
ID=39230813
Family Applications (4)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| JP2009530406A Expired - Fee Related JP5388854B2 (ja) | 2006-09-26 | 2007-09-25 | ５−置換キナゾリノン誘導体、それを含む組成物、及びその使用方法 |
| JP2013210802A Expired - Fee Related JP5901599B2 (ja) | 2006-09-26 | 2013-10-08 | ５−置換キナゾリノン誘導体、それを含む組成物、及びその使用方法 |
| JP2015218025A Expired - Fee Related JP6133383B2 (ja) | 2006-09-26 | 2015-11-06 | ５−置換キナゾリノン誘導体、それを含む組成物、及びその使用方法 |
| JP2017082496A Ceased JP2017165744A (ja) | 2006-09-26 | 2017-04-19 | ５−置換キナゾリノン誘導体、それを含む組成物、及びその使用方法 |
Family Applications After (3)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| JP2013210802A Expired - Fee Related JP5901599B2 (ja) | 2006-09-26 | 2013-10-08 | ５−置換キナゾリノン誘導体、それを含む組成物、及びその使用方法 |
| JP2015218025A Expired - Fee Related JP6133383B2 (ja) | 2006-09-26 | 2015-11-06 | ５−置換キナゾリノン誘導体、それを含む組成物、及びその使用方法 |
| JP2017082496A Ceased JP2017165744A (ja) | 2006-09-26 | 2017-04-19 | ５−置換キナゾリノン誘導体、それを含む組成物、及びその使用方法 |
Country Status (33)
Families Citing this family (80)
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| US8835506B2 (en) | 2008-06-05 | 2014-09-16 | Stc.Unm | Methods and related compositions for the treatment of cancer |
| US20100160368A1 (en) * | 2008-08-18 | 2010-06-24 | Gregory Jefferson J | Methods of Treating Dermatological Disorders and Inducing Interferon Biosynthesis With Shorter Durations of Imiquimod Therapy |
| EP2378876B1 (en) | 2008-12-19 | 2018-11-14 | Medicis Pharmaceutical Corporation | Lower dosage strength imiquimod formulations and short dosing regimens for treating actinic keratosis |
| DK2433124T3 (en) * | 2009-05-19 | 2017-06-19 | Vivia Biotech Sl | PROCEDURES FOR PROVIDING PERSONALIZED MEDICAL EX VIVO TESTS FOR HEMATOLOGICAL NEOPLASMS |
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| MX336923B (es) | 2009-07-13 | 2016-02-05 | Medicis Pharmaceutical Corp | Formulaciones de imiquimod de concentracion de dosificacion inferior y regimenes de dosificacion cortos para tratar verrugas genitales y perianales. |
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| AU2012236655B2 (en) | 2011-03-28 | 2016-09-22 | Deuterx, Llc, | 2',6'-dioxo-3'-deutero-piperdin-3-yl-isoindoline compounds |
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| CA2877736C (en) | 2012-06-29 | 2021-12-07 | Celgene Corporation | Methods for determining drug efficacy using cereblon-associated proteins |
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| CN104755472A (zh) * | 2012-09-04 | 2015-07-01 | 细胞基因公司 | 3-(5-氨基-2-甲基-4-氧代喹唑啉-3(4h)-基)哌啶-2,6-二酮的同位素体及其制备方法 |
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| CA2935495C (en) * | 2013-01-14 | 2021-04-20 | Deuterx, Llc | 3-(5-substituted-4-oxoquinazolin-3(4h)-yl)-3-deutero-piperidine-2,6-dione derivatives |
| US9290475B2 (en) | 2013-03-14 | 2016-03-22 | Deuterx, Llc | 3-(substituted-4-oxoquinazolin-3(4H)-yl)-3-deutero-piperidine-2,6-dione derivatives and compositions comprising and methods of using the same |
| MX368286B (es) | 2013-04-17 | 2019-09-27 | Signal Pharm Llc | Terapia de combinacion que comprende un inhibidor de tor cinasa y un compuesto de quinazolinona 5-sustituida para tratar cancer. |
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