JP2007504174A5 - - Google Patents

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Publication number
JP2007504174A5
JP2007504174A5 JP2006525016A JP2006525016A JP2007504174A5 JP 2007504174 A5 JP2007504174 A5 JP 2007504174A5 JP 2006525016 A JP2006525016 A JP 2006525016A JP 2006525016 A JP2006525016 A JP 2006525016A JP 2007504174 A5 JP2007504174 A5 JP 2007504174A5
Authority
JP
Japan
Prior art keywords
disorders
epilepsy
pharmaceutical composition
pain
depression
Prior art date
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
Pending
Application number
JP2006525016A
Other languages
English (en)
Japanese (ja)
Other versions
JP2007504174A (ja
Filing date
Publication date
Priority claimed from US10/655,393 external-priority patent/US7186726B2/en
Application filed filed Critical
Publication of JP2007504174A publication Critical patent/JP2007504174A/ja
Publication of JP2007504174A5 publication Critical patent/JP2007504174A5/ja
Pending legal-status Critical Current

Links

JP2006525016A 2003-09-03 2004-09-03 カルシウムチャネル遮断薬として使用されるピペラジン置換化合物 Pending JP2007504174A (ja)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
US10/655,393 US7186726B2 (en) 1998-06-30 2003-09-03 Preferentially substituted calcium channel blockers
PCT/CA2004/001629 WO2005021523A1 (en) 2003-09-03 2004-09-03 Piperazine substituted compounds used as calcium channel blockers

Publications (2)

Publication Number Publication Date
JP2007504174A JP2007504174A (ja) 2007-03-01
JP2007504174A5 true JP2007504174A5 (enExample) 2007-10-18

Family

ID=34273458

Family Applications (1)

Application Number Title Priority Date Filing Date
JP2006525016A Pending JP2007504174A (ja) 2003-09-03 2004-09-03 カルシウムチャネル遮断薬として使用されるピペラジン置換化合物

Country Status (12)

Country Link
US (2) US7186726B2 (enExample)
EP (1) EP1670775A4 (enExample)
JP (1) JP2007504174A (enExample)
CN (1) CN1871225A (enExample)
AU (1) AU2004268711A1 (enExample)
BR (1) BRPI0414094A (enExample)
CA (1) CA2537487A1 (enExample)
IL (1) IL174025A0 (enExample)
MX (1) MXPA06002467A (enExample)
NZ (1) NZ546254A (enExample)
WO (1) WO2005021523A1 (enExample)
ZA (1) ZA200602684B (enExample)

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GB0419072D0 (en) 2004-08-26 2004-09-29 Kudos Pharm Ltd Phthalazinone derivatives
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US7511077B2 (en) * 2005-02-09 2009-03-31 Neuromed Pharmaceuticals Ltd. Diamine calcium channel blockers
EP1871372A4 (en) * 2005-04-08 2010-06-02 Neuromed Pharmaceuticals Ltd COMBINATION THERAPY WHICH INCLUDES AN AGENT BLOCKING CALCIUM CHANNELS OF TYPE N FOR THE RELIEF OF PAIN
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WO2008043183A1 (en) * 2006-10-13 2008-04-17 Neuromed Pharmaceuticals Ltd. Cyclopropyl-piperazine compounds as calcium channel blockers
TWI404716B (zh) * 2006-10-17 2013-08-11 Kudos Pharm Ltd 酞嗪酮（ｐｈｔｈａｌａｚｉｎｏｎｅ）衍生物
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US20080139578A1 (en) * 2006-11-30 2008-06-12 Catherine Abbadie Substituted piperizines for the treatment of pain
GB0700893D0 (en) * 2007-01-17 2007-02-21 King S College London Male contraceptive
AU2008254061B2 (en) 2007-05-22 2012-06-14 Astellas Pharma Inc. 1-substituted tetrahydroisoquinoline compound
RU2487868C2 (ru) * 2007-10-17 2013-07-20 Кудос Фармасеутикалс Лимитед 4-[3-(4-циклопропанкарбонил-пиперазин-1-карбонил)-4-фтор-бензил]-2н-фталазин-1-он
CA2722706A1 (en) * 2008-04-28 2009-11-05 Zalicus Pharmaceuticals Ltd. Di-t-butylphenyl piperazines as calcium channel blockers
US20090270338A1 (en) * 2008-04-28 2009-10-29 Galemmo Jr Robert Diaryl-cyclylalkyl derivatives as calcium channel blockers
NZ592719A (en) 2008-10-07 2012-09-28 Astrazeneca Uk Ltd PHARMACEUTICAL FORMULATION 514 comprising 4-[3-( 4-cyclopropanecarbonyl-piperazine-1-carbonyl)-4-fluoro-benzyl]-2H-phthalazin-1-one
US9492439B2 (en) 2010-03-11 2016-11-15 New York University Amido compounds as RORγt modulators and uses thereof
US8409560B2 (en) 2011-03-08 2013-04-02 Zalicus Pharmaceuticals Ltd. Solid dispersion formulations and methods of use thereof
US8591944B2 (en) 2011-03-08 2013-11-26 Zalicus Pharmaceuticals Ltd. Solid dispersion formulations and methods of use thereof
MX2014002810A (es) * 2011-09-09 2014-09-08 Univ New York Compuestos amido como moduladores del receptor nuclear huérfanoyt y usos de los mismos.
CN103130745B (zh) * 2011-11-28 2017-03-15 中国人民解放军军事医学科学院毒物药物研究所 二芳基哌嗪类化合物及其医药用途
CN105218501A (zh) * 2014-07-03 2016-01-06 南京大学 含哌嗪环的香豆素类衍生物及其制备与在抗菌药物中的应用

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US6943168B2 (en) * 1998-06-30 2005-09-13 Neuromed Technologies Inc. Calcium channel inhibitors comprising benzhydril spaced from piperazine
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