JP2007504174A5 - - Google Patents

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Publication number
JP2007504174A5
JP2007504174A5 JP2006525016A JP2006525016A JP2007504174A5 JP 2007504174 A5 JP2007504174 A5 JP 2007504174A5 JP 2006525016 A JP2006525016 A JP 2006525016A JP 2006525016 A JP2006525016 A JP 2006525016A JP 2007504174 A5 JP2007504174 A5 JP 2007504174A5
Authority
JP
Japan
Prior art keywords
disorders
epilepsy
pharmaceutical composition
pain
depression
Prior art date
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
Pending
Application number
JP2006525016A
Other languages
English (en)
Japanese (ja)
Other versions
JP2007504174A (ja
Filing date
Publication date
Priority claimed from US10/655,393 external-priority patent/US7186726B2/en
Application filed filed Critical
Publication of JP2007504174A publication Critical patent/JP2007504174A/ja
Publication of JP2007504174A5 publication Critical patent/JP2007504174A5/ja
Pending legal-status Critical Current

Links

JP2006525016A 2003-09-03 2004-09-03 カルシウムチャネル遮断薬として使用されるピペラジン置換化合物 Pending JP2007504174A (ja)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
US10/655,393 US7186726B2 (en) 1998-06-30 2003-09-03 Preferentially substituted calcium channel blockers
PCT/CA2004/001629 WO2005021523A1 (en) 2003-09-03 2004-09-03 Piperazine substituted compounds used as calcium channel blockers

Publications (2)

Publication Number Publication Date
JP2007504174A JP2007504174A (ja) 2007-03-01
JP2007504174A5 true JP2007504174A5 (enExample) 2007-10-18

Family

ID=34273458

Family Applications (1)

Application Number Title Priority Date Filing Date
JP2006525016A Pending JP2007504174A (ja) 2003-09-03 2004-09-03 カルシウムチャネル遮断薬として使用されるピペラジン置換化合物

Country Status (12)

Country Link
US (2) US7186726B2 (enExample)
EP (1) EP1670775A4 (enExample)
JP (1) JP2007504174A (enExample)
CN (1) CN1871225A (enExample)
AU (1) AU2004268711A1 (enExample)
BR (1) BRPI0414094A (enExample)
CA (1) CA2537487A1 (enExample)
IL (1) IL174025A0 (enExample)
MX (1) MXPA06002467A (enExample)
NZ (1) NZ546254A (enExample)
WO (1) WO2005021523A1 (enExample)
ZA (1) ZA200602684B (enExample)

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US7511077B2 (en) * 2005-02-09 2009-03-31 Neuromed Pharmaceuticals Ltd. Diamine calcium channel blockers
JP2008534630A (ja) * 2005-04-08 2008-08-28 ニューロメッド ファーマシューティカルズ リミテッド 疼痛の軽減のためのｎ型カルシウムチャネルブロッカーを含む組み合わせ治療の方法
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CA2633457A1 (en) * 2005-12-19 2007-06-28 Neuromed Pharmaceuticals Ltd. Heterocyclic amide derivatives as calcium channel blockers
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WO2007133481A2 (en) * 2006-05-11 2007-11-22 Neuromed Pharmaceuticals Ltd. Method for increasing the bioavailability of benzhydryl piperazine containing compounds
US20100029681A1 (en) * 2006-05-26 2010-02-04 Hassan Pajouhesh Heterocyclic compounds as calcium channel blockers
CA2663280A1 (en) * 2006-09-14 2008-03-20 Neuromed Pharmaceuticals Ltd. Diaryl piperidine compounds as calcium channel blockers
EP2074105A4 (en) * 2006-10-13 2010-10-06 Neuromed Pharmaceuticals Ltd CYCLOPROPYL-PIPERAZINE COMPOUNDS AS CALCIUM INHIBITORS
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WO2008050200A1 (en) * 2006-10-24 2008-05-02 Pfizer Products Inc. Oxadiazole compounds as calcium channel antagonists
US20080139578A1 (en) * 2006-11-30 2008-06-12 Catherine Abbadie Substituted piperizines for the treatment of pain
GB0700893D0 (en) 2007-01-17 2007-02-21 King S College London Male contraceptive
US8263607B2 (en) 2007-05-22 2012-09-11 Astellas Pharma Inc. 1-substituted tetrahydroisoquinoline compound
MX2010004028A (es) * 2007-10-17 2010-04-30 Kudos Pharm Ltd 4-[3-(4-ciclopropancarbonil-piperacin-1-carbonil)-4-fluoro-bencil ]-2h-ftalacin-1-ona.
WO2009132454A1 (en) * 2008-04-28 2009-11-05 Neuromed Pharmaceuticals Ltd. Di-t-butylphenyl piperazines as calcium channel blockers
US20090270338A1 (en) * 2008-04-28 2009-10-29 Galemmo Jr Robert Diaryl-cyclylalkyl derivatives as calcium channel blockers
EP2346495B2 (en) 2008-10-07 2023-05-24 Kudos Pharmaceuticals Limited Pharmaceutical formulation 514
EP2558087A4 (en) 2010-03-11 2013-09-11 Univ New York AMID COMPOUNDS AS RORYT MODULATORS AND ITS USES
US8409560B2 (en) 2011-03-08 2013-04-02 Zalicus Pharmaceuticals Ltd. Solid dispersion formulations and methods of use thereof
WO2012122279A1 (en) 2011-03-08 2012-09-13 Zalicus Pharmaceuticals Ltd. Solid dispersion formulations and methods of use thereof
SG11201400456RA (en) 2011-09-09 2014-04-28 Univ New York Amido compounds as ror?tmodulators and uses thereof
CN103130745B (zh) * 2011-11-28 2017-03-15 中国人民解放军军事医学科学院毒物药物研究所 二芳基哌嗪类化合物及其医药用途
CN105218501A (zh) * 2014-07-03 2016-01-06 南京大学 含哌嗪环的香豆素类衍生物及其制备与在抗菌药物中的应用

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US6492375B2 (en) * 1998-06-30 2002-12-10 Neuromed Technologies, Inc. Partially saturated calcium channel blockers
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