JP2005524660A5 - - Google Patents

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Publication number
JP2005524660A5
JP2005524660A5 JP2003571259A JP2003571259A JP2005524660A5 JP 2005524660 A5 JP2005524660 A5 JP 2005524660A5 JP 2003571259 A JP2003571259 A JP 2003571259A JP 2003571259 A JP2003571259 A JP 2003571259A JP 2005524660 A5 JP2005524660 A5 JP 2005524660A5
Authority
JP
Japan
Prior art keywords
oxo
oxazolidinecarboxamide
methyl
dihydro
phenyl
Prior art date
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
Pending
Application number
JP2003571259A
Other languages
English (en)
Japanese (ja)
Other versions
JP2005524660A (ja
Filing date
Publication date
Application filed filed Critical
Priority claimed from PCT/US2003/003125 external-priority patent/WO2003072553A1/en
Publication of JP2005524660A publication Critical patent/JP2005524660A/ja
Publication of JP2005524660A5 publication Critical patent/JP2005524660A5/ja
Pending legal-status Critical Current

Links

JP2003571259A 2002-02-25 2003-02-24 Ｎ−アリール−２−オキサゾリジノン−５−カルボキサミドおよびその誘導体ならびに抗細菌剤としてのそれらの使用 Pending JP2005524660A (ja)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
US35949502P 2002-02-25 2002-02-25
PCT/US2003/003125 WO2003072553A1 (en) 2002-02-25 2003-02-24 N-aryl-2-oxazolidinone-5-carboxamides and their derivates and their use as antibacterials

Publications (2)

Publication Number Publication Date
JP2005524660A JP2005524660A (ja) 2005-08-18
JP2005524660A5 true JP2005524660A5 (https=) 2006-04-13

Family

ID=27766097

Family Applications (1)

Application Number Title Priority Date Filing Date
JP2003571259A Pending JP2005524660A (ja) 2002-02-25 2003-02-24 Ｎ−アリール−２−オキサゾリジノン−５−カルボキサミドおよびその誘導体ならびに抗細菌剤としてのそれらの使用

Country Status (36)

Country Link
US (1) US6919329B2 (https=)
EP (1) EP1478629B1 (https=)
JP (1) JP2005524660A (https=)
KR (1) KR100613532B1 (https=)
CN (1) CN1639135A (https=)
AP (1) AP1902A (https=)
AR (1) AR038536A1 (https=)
AT (1) ATE342258T1 (https=)
AU (1) AU2003210807A1 (https=)
BR (1) BR0307924A (https=)
CA (1) CA2476038A1 (https=)
CO (1) CO5611128A2 (https=)
CY (1) CY1105797T1 (https=)
DE (1) DE60308998T2 (https=)
DK (1) DK1478629T3 (https=)
EA (1) EA007490B1 (https=)
EC (1) ECSP045245A (https=)
ES (1) ES2271615T3 (https=)
GE (1) GEP20074198B (https=)
HR (1) HRP20040717A2 (https=)
IS (1) IS7376A (https=)
MA (1) MA27180A1 (https=)
MX (1) MXPA04008205A (https=)
MY (1) MY135233A (https=)
NO (1) NO20044062L (https=)
NZ (1) NZ534521A (https=)
OA (1) OA12779A (https=)
PL (1) PL372461A1 (https=)
PT (1) PT1478629E (https=)
SI (1) SI1478629T1 (https=)
TN (1) TNSN04163A1 (https=)
TW (1) TW200305568A (https=)
UA (1) UA80112C2 (https=)
WO (1) WO2003072553A1 (https=)
YU (1) YU72804A (https=)
ZA (1) ZA200406362B (https=)

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JP5534497B2 (ja) 2005-06-08 2014-07-02 メリンタ セラピューティクス，インコーポレイテッド トリアゾール類の合成方法
DE602006010702D1 (de) 2005-06-29 2010-01-07 Pharmacia & Upjohn Co Llc Homomorpholinoxazolidinone als antibakterielle mittel
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WO2007004032A1 (en) * 2005-07-06 2007-01-11 Pharmacia & Upjohn Company Llc Oxazolidiones containing cyclobutane as antibacterial agents
BRPI0620196A2 (pt) * 2005-12-23 2013-01-15 Astrazeneca Ab composto, processo para a preparaÇço do mesmo, composiÇço farmacÊutica, uso de um composto, e, mÉtodos para a produÇço de um efeito antibacteriano em um animal de sangue quente, para a inibiÇço de dna girase e/ou topoisomerase iv bacteriana em um animal de sangue quente e para o tratamento de uma infecÇço bacteriana em um animal de sangue quente
WO2007088478A1 (en) * 2006-02-01 2007-08-09 Pfizer Products Inc. Indazole oxazolidinones as antibacterial agents
KR20080110877A (ko) * 2006-03-31 2008-12-19 재단법인 이쯔우 연구소 헤테로환을 갖는 신규 화합물
WO2008026563A1 (en) * 2006-08-30 2008-03-06 Shionogi & Co., Ltd. Hydrazine amide derivative
US8088777B2 (en) * 2006-08-30 2012-01-03 Shionogi & Co., Ltd. Urea derivative
JP5455906B2 (ja) * 2007-08-06 2014-03-26 ミクウルク ファーマシューティカルズ，インコーポレイテッド 細菌感染症治療のための抗微生物性オルト−フルオロフェニルオキサゾリジノン
CN101883768A (zh) 2007-10-02 2010-11-10 财团法人乙卯研究所 具有7元杂环的噁唑烷酮衍生物
US20120040974A1 (en) * 2008-08-18 2012-02-16 Yale University Mif modulators
US9643922B2 (en) 2008-08-18 2017-05-09 Yale University MIF modulators
US9540322B2 (en) 2008-08-18 2017-01-10 Yale University MIF modulators
CN102224151A (zh) 2008-11-20 2011-10-19 万能药生物有限公司 新的抗微生物剂
MY156354A (en) * 2009-02-03 2016-02-15 Merck Sharp & Dohme Crystalline form of r)-3-(4-(2-(2-methyltetrazol-5-yl)pyridin-5-yl)-3-fluorophenyl)-5-hydroxymethyl oxazolidin-2-one dihydrogen phosphate
KR20120106697A (ko) 2009-06-26 2012-09-26 파나세아 바이오테크 리미티드 신규 아자비시클로헥산
JP5996532B2 (ja) 2010-07-15 2016-09-21 バイエル・インテレクチュアル・プロパティ・ゲゼルシャフト・ミット・ベシュレンクテル・ハフツングＢａｙｅｒ Ｉｎｔｅｌｌｅｃｔｕａｌ Ｐｒｏｐｅｒｔｙ ＧｍｂＨ 有害生物防除剤としての新規複素環式化合物
UA112897C2 (uk) 2012-05-09 2016-11-10 Байєр Фарма Акцієнгезелльшафт Біциклічно заміщені урацили та їх застосування для лікування і/або профілактики захворювань
US9382276B2 (en) 2014-02-21 2016-07-05 Micurx Pharmaceuticals, Inc. Water-soluble O-carbonyl phosphoramidate prodrugs for therapeutic administration
JP7205529B2 (ja) * 2018-02-26 2023-01-17 住友化学株式会社 オキサゾリジノン化合物の製造方法

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