HK1163661A1 - Heteroaryl derivatives as cftr modulators cftr - Google Patents
Heteroaryl derivatives as cftr modulators cftrInfo
- Publication number
- HK1163661A1 HK1163661A1 HK12103803.7A HK12103803A HK1163661A1 HK 1163661 A1 HK1163661 A1 HK 1163661A1 HK 12103803 A HK12103803 A HK 12103803A HK 1163661 A1 HK1163661 A1 HK 1163661A1
- Authority
- HK
- Hong Kong
- Prior art keywords
- cftr
- modulators
- heteroaryl derivatives
- heteroaryl
- derivatives
- Prior art date
Links
Classifications
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- C07D491/02—Heterocyclic compounds containing in the condensed ring system both one or more rings having oxygen atoms as the only ring hetero atoms and one or more rings having nitrogen atoms as the only ring hetero atoms, not provided for by groups C07D451/00 - C07D459/00, C07D463/00, C07D477/00 or C07D489/00 in which the condensed system contains two hetero rings
- C07D491/04—Ortho-condensed systems
- C07D491/044—Ortho-condensed systems with only one oxygen atom as ring hetero atom in the oxygen-containing ring
- C07D491/048—Ortho-condensed systems with only one oxygen atom as ring hetero atom in the oxygen-containing ring the oxygen-containing ring being five-membered
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- A61K31/435—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom
- A61K31/44—Non condensed pyridines; Hydrogenated derivatives thereof
- A61K31/4427—Non condensed pyridines; Hydrogenated derivatives thereof containing further heterocyclic ring systems
- A61K31/443—Non condensed pyridines; Hydrogenated derivatives thereof containing further heterocyclic ring systems containing a five-membered ring with oxygen as a ring hetero atom
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US3215908P | 2008-02-28 | 2008-02-28 | |
PCT/US2009/035064 WO2009108657A2 (en) | 2008-02-28 | 2009-02-25 | Heteroaryl derivatives as cftr modulators |
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EP (1) | EP2271622B1 (de) |
JP (3) | JP5523352B2 (de) |
CN (3) | CN103382201B (de) |
AU (1) | AU2009219363B2 (de) |
CA (3) | CA2716109C (de) |
ES (1) | ES2647531T3 (de) |
HK (1) | HK1163661A1 (de) |
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