HK1060567A1 - Crystalline monohydrate, method for producing the same and the use thereof in the production of a medicament. - Google Patents

Crystalline monohydrate, method for producing the same and the use thereof in the production of a medicament.

Info

Publication number
HK1060567A1
HK1060567A1 HK04103583A HK04103583A HK1060567A1 HK 1060567 A1 HK1060567 A1 HK 1060567A1 HK 04103583 A HK04103583 A HK 04103583A HK 04103583 A HK04103583 A HK 04103583A HK 1060567 A1 HK1060567 A1 HK 1060567A1
Authority
HK
Hong Kong
Prior art keywords
medicament
producing
production
same
crystalline monohydrate
Prior art date
Application number
HK04103583A
Other languages
English (en)
Inventor
Rolf Banholzer
Peter Sieger
Christian Kulinna
Michael Trunk
Manfred Ludwig August Graulich
Peter Specht
Helmut Meissner
Andreas Mathes
Original Assignee
Boehringer Ingelheim Pharma
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Family has litigation
First worldwide family litigation filed litigation Critical https://patents.darts-ip.com/?family=7659568&utm_source=google_patent&utm_medium=platform_link&utm_campaign=public_patent_search&patent=HK1060567(A1) "Global patent litigation dataset” by Darts-ip is licensed under a Creative Commons Attribution 4.0 International License.
Application filed by Boehringer Ingelheim Pharma filed Critical Boehringer Ingelheim Pharma
Publication of HK1060567A1 publication Critical patent/HK1060567A1/xx

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D451/00Heterocyclic compounds containing 8-azabicyclo [3.2.1] octane, 9-azabicyclo [3.3.1] nonane, or 3-oxa-9-azatricyclo [3.3.1.0<2,4>] nonane ring systems, e.g. tropane or granatane alkaloids, scopolamine; Cyclic acetals thereof
    • C07D451/02Heterocyclic compounds containing 8-azabicyclo [3.2.1] octane, 9-azabicyclo [3.3.1] nonane, or 3-oxa-9-azatricyclo [3.3.1.0<2,4>] nonane ring systems, e.g. tropane or granatane alkaloids, scopolamine; Cyclic acetals thereof containing not further condensed 8-azabicyclo [3.2.1] octane or 3-oxa-9-azatricyclo [3.3.1.0<2,4>] nonane ring systems, e.g. tropane; Cyclic acetals thereof
    • C07D451/04Heterocyclic compounds containing 8-azabicyclo [3.2.1] octane, 9-azabicyclo [3.3.1] nonane, or 3-oxa-9-azatricyclo [3.3.1.0<2,4>] nonane ring systems, e.g. tropane or granatane alkaloids, scopolamine; Cyclic acetals thereof containing not further condensed 8-azabicyclo [3.2.1] octane or 3-oxa-9-azatricyclo [3.3.1.0<2,4>] nonane ring systems, e.g. tropane; Cyclic acetals thereof with hetero atoms directly attached in position 3 of the 8-azabicyclo [3.2.1] octane or in position 7 of the 3-oxa-9-azatricyclo [3.3.1.0<2,4>] nonane ring system
    • C07D451/06Oxygen atoms
    • C07D451/10Oxygen atoms acylated by aliphatic or araliphatic carboxylic acids, e.g. atropine, scopolamine
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P11/00Drugs for disorders of the respiratory system
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P11/00Drugs for disorders of the respiratory system
    • A61P11/06Antiasthmatics
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P11/00Drugs for disorders of the respiratory system
    • A61P11/16Central respiratory analeptics
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00Drugs for disorders of the nervous system
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P43/00Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00

Landscapes

  • Health & Medical Sciences (AREA)
  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • General Health & Medical Sciences (AREA)
  • General Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Engineering & Computer Science (AREA)
  • Animal Behavior & Ethology (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • Pulmonology (AREA)
  • Biomedical Technology (AREA)
  • Neurology (AREA)
  • Neurosurgery (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Nitrogen Condensed Heterocyclic Rings (AREA)
  • Medicinal Preparation (AREA)
  • Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
HK04103583A 2000-10-12 2004-05-20 Crystalline monohydrate, method for producing the same and the use thereof in the production of a medicament. HK1060567A1 (en)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
DE10050621 2000-10-12
PCT/EP2001/011225 WO2002030928A1 (de) 2000-10-12 2001-09-28 Kristallines monohydrat, verfahren zu dessen herstellung und dessen verwendung zur herstellung eines arzneimittels

Publications (1)

Publication Number Publication Date
HK1060567A1 true HK1060567A1 (en) 2004-08-13

Family

ID=7659568

Family Applications (2)

Application Number Title Priority Date Filing Date
HK04103583A HK1060567A1 (en) 2000-10-12 2004-05-20 Crystalline monohydrate, method for producing the same and the use thereof in the production of a medicament.
HK06106478.2A HK1086557A1 (en) 2000-10-12 2006-06-07 Crystalline monohydrate, method for producing the same and the use thereof in the production of a medicament

Family Applications After (1)

Application Number Title Priority Date Filing Date
HK06106478.2A HK1086557A1 (en) 2000-10-12 2006-06-07 Crystalline monohydrate, method for producing the same and the use thereof in the production of a medicament

Country Status (47)

Country Link
EP (2) EP1326862B1 (sr)
JP (1) JP3764422B2 (sr)
KR (1) KR100823860B1 (sr)
CN (2) CN100519558C (sr)
AP (1) AP1572A (sr)
AR (2) AR034389A1 (sr)
AT (1) ATE276253T1 (sr)
AU (2) AU2002214996B2 (sr)
BG (1) BG66161B1 (sr)
BR (1) BR0114584A (sr)
CA (1) CA2425539C (sr)
CR (1) CR6938A (sr)
CZ (1) CZ301841B6 (sr)
DE (1) DE50103666D1 (sr)
DK (1) DK1326862T3 (sr)
DZ (1) DZ3478A1 (sr)
EA (1) EA004381B1 (sr)
EC (1) ECSP034540A (sr)
EE (1) EE04567B1 (sr)
EG (1) EG24142A (sr)
ES (1) ES2228965T3 (sr)
GE (1) GEP20063905B (sr)
HK (2) HK1060567A1 (sr)
HR (1) HRP20030276B1 (sr)
HU (1) HU226830B1 (sr)
IL (2) IL155335A0 (sr)
IS (1) IS2339B (sr)
MA (1) MA25842A1 (sr)
ME (2) ME00243B (sr)
MX (1) MXPA03003221A (sr)
MY (1) MY126931A (sr)
NO (1) NO328465B1 (sr)
NZ (1) NZ525733A (sr)
OA (1) OA12403A (sr)
PE (1) PE20020422A1 (sr)
PL (1) PL207870B1 (sr)
PT (1) PT1326862E (sr)
RS (1) RS50218B (sr)
SA (1) SA01220412B1 (sr)
SI (1) SI1326862T1 (sr)
SK (1) SK287009B6 (sr)
TR (1) TR200402579T4 (sr)
TW (1) TW589313B (sr)
UA (1) UA74215C2 (sr)
UY (2) UY26962A1 (sr)
WO (1) WO2002030928A1 (sr)
ZA (1) ZA200302500B (sr)

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Also Published As

Publication number Publication date
TR200402579T4 (tr) 2004-12-21
GEP20063905B (en) 2006-08-25
AR034389A1 (es) 2004-02-25
WO2002030928A1 (de) 2002-04-18
EP1468998A1 (de) 2004-10-20
YU27303A (sh) 2006-05-25
PT1326862E (pt) 2004-11-30
DE50103666D1 (de) 2004-10-21
SK287009B6 (sk) 2009-09-07
MA25842A1 (fr) 2003-07-01
CN100519558C (zh) 2009-07-29
PL366041A1 (en) 2005-01-24
SI1326862T1 (en) 2005-02-28
IL155335A (en) 2009-02-11
ATE276253T1 (de) 2004-10-15
EA004381B1 (ru) 2004-04-29
NO20031694D0 (no) 2003-04-11
HU226830B1 (en) 2009-11-30
ZA200302500B (en) 2004-04-22
CN1221549C (zh) 2005-10-05
EE200300171A (et) 2003-06-16
AP2003002775A0 (en) 2003-03-31
DZ3478A1 (fr) 2002-04-18
ECSP034540A (es) 2003-07-25
HRP20030276A2 (en) 2005-02-28
NO328465B1 (no) 2010-02-22
BG107687A (bg) 2003-09-30
SA01220412B1 (ar) 2006-11-05
IS2339B (is) 2008-02-15
RS50218B (sr) 2009-07-15
EP1326862B1 (de) 2004-09-15
HUP0301022A3 (en) 2005-12-28
HRP20030276B1 (en) 2006-02-28
KR20030042008A (ko) 2003-05-27
TW589313B (en) 2004-06-01
CA2425539C (en) 2007-04-03
BR0114584A (pt) 2003-08-26
AP1572A (en) 2006-02-13
CR6938A (es) 2004-10-28
MY126931A (en) 2006-10-31
AU2002214996B2 (en) 2007-03-15
MXPA03003221A (es) 2004-12-03
EP1326862A1 (de) 2003-07-16
OA12403A (en) 2006-04-18
EA200300457A1 (ru) 2003-10-30
HK1086557A1 (en) 2006-09-22
JP2004526668A (ja) 2004-09-02
UY34901A (es) 2015-02-27
DK1326862T3 (da) 2004-11-22
BG66161B1 (bg) 2011-09-30
EG24142A (en) 2008-08-06
UA74215C2 (uk) 2005-11-15
CZ301841B6 (cs) 2010-07-07
CA2425539A1 (en) 2003-04-11
AR068527A2 (es) 2009-11-18
HUP0301022A2 (hu) 2003-10-28
CN1469877A (zh) 2004-01-21
MEP40008A (en) 2011-02-10
JP3764422B2 (ja) 2006-04-05
NO20031694L (no) 2003-04-11
NZ525733A (en) 2005-01-28
SK4362003A3 (en) 2003-08-05
AU1499602A (en) 2002-04-22
PE20020422A1 (es) 2002-06-28
PL207870B1 (pl) 2011-02-28
IS6772A (is) 2003-04-09
ME00243B (me) 2011-05-10
EE04567B1 (et) 2005-12-15
KR100823860B1 (ko) 2008-04-21
UY26962A1 (es) 2002-06-20
CN1733761A (zh) 2006-02-15
IL155335A0 (en) 2003-11-23
ES2228965T3 (es) 2005-04-16

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