AR034389A1 - Monohidrato cristalino de bromuro de tiotropio, procedimiento para su preparacion, su utilización para la preparacion de un medicamento, un medicamento que lo contiene, los hidratos cristalinos del bromuro de tiotropio y un procedimiento para preparacion de estos hidratos cristalinos - Google Patents

Monohidrato cristalino de bromuro de tiotropio, procedimiento para su preparacion, su utilización para la preparacion de un medicamento, un medicamento que lo contiene, los hidratos cristalinos del bromuro de tiotropio y un procedimiento para preparacion de estos hidratos cristalinos

Info

Publication number
AR034389A1
AR034389A1 ARP010104782A ARP010104782A AR034389A1 AR 034389 A1 AR034389 A1 AR 034389A1 AR P010104782 A ARP010104782 A AR P010104782A AR P010104782 A ARP010104782 A AR P010104782A AR 034389 A1 AR034389 A1 AR 034389A1
Authority
AR
Argentina
Prior art keywords
preparation
procedure
tiotropio
bromide
medicinal product
Prior art date
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
Pending
Application number
ARP010104782A
Other languages
English (en)
Inventor
Rolf Banholzer
Peter Sieger
Christian Kulinna
Michael Trunk
Manfred Ludwig August Graulich
Peter Specht
Helmut Meissner
Andreas Mathes
Current Assignee (The listed assignees may be inaccurate. Google has not performed a legal analysis and makes no representation or warranty as to the accuracy of the list.)
Boehringer Ingelheim Pharma GmbH Co KG
Original Assignee
Boehringer Ingelheim Pharma GmbH Co KG
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Family has litigation
First worldwide family litigation filed litigation Critical https://patents.darts-ip.com/?family=7659568&utm_source=google_patent&utm_medium=platform_link&utm_campaign=public_patent_search&patent=AR034389(A1) "Global patent litigation dataset” by Darts-ip is licensed under a Creative Commons Attribution 4.0 International License.
Application filed by Boehringer Ingelheim Pharma GmbH Co KG filed Critical Boehringer Ingelheim Pharma GmbH Co KG
Publication of AR034389A1 publication Critical patent/AR034389A1/es
Pending legal-status Critical Current

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D451/00—Heterocyclic compounds containing 8-azabicyclo [3.2.1] octane, 9-azabicyclo [3.3.1] nonane, or 3-oxa-9-azatricyclo [3.3.1.0<2,4>] nonane ring systems, e.g. tropane or granatane alkaloids, scopolamine; Cyclic acetals thereof
    • C07D451/02—Heterocyclic compounds containing 8-azabicyclo [3.2.1] octane, 9-azabicyclo [3.3.1] nonane, or 3-oxa-9-azatricyclo [3.3.1.0<2,4>] nonane ring systems, e.g. tropane or granatane alkaloids, scopolamine; Cyclic acetals thereof containing not further condensed 8-azabicyclo [3.2.1] octane or 3-oxa-9-azatricyclo [3.3.1.0<2,4>] nonane ring systems, e.g. tropane; Cyclic acetals thereof
    • C07D451/04—Heterocyclic compounds containing 8-azabicyclo [3.2.1] octane, 9-azabicyclo [3.3.1] nonane, or 3-oxa-9-azatricyclo [3.3.1.0<2,4>] nonane ring systems, e.g. tropane or granatane alkaloids, scopolamine; Cyclic acetals thereof containing not further condensed 8-azabicyclo [3.2.1] octane or 3-oxa-9-azatricyclo [3.3.1.0<2,4>] nonane ring systems, e.g. tropane; Cyclic acetals thereof with hetero atoms directly attached in position 3 of the 8-azabicyclo [3.2.1] octane or in position 7 of the 3-oxa-9-azatricyclo [3.3.1.0<2,4>] nonane ring system
    • C07D451/06—Oxygen atoms
    • C07D451/10—Oxygen atoms acylated by aliphatic or araliphatic carboxylic acids, e.g. atropine, scopolamine
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P11/00—Drugs for disorders of the respiratory system
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P11/00—Drugs for disorders of the respiratory system
    • A61P11/06—Antiasthmatics
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P11/00—Drugs for disorders of the respiratory system
    • A61P11/16—Central respiratory analeptics
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00—Drugs for disorders of the nervous system
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P43/00—Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00

Landscapes

  • Health & Medical Sciences (AREA)
  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • General Health & Medical Sciences (AREA)
  • General Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Engineering & Computer Science (AREA)
  • Animal Behavior & Ethology (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • Pulmonology (AREA)
  • Biomedical Technology (AREA)
  • Neurology (AREA)
  • Neurosurgery (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Nitrogen Condensed Heterocyclic Rings (AREA)
  • Medicinal Preparation (AREA)
  • Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)

Abstract

El presente se refiere a un monohidrato cristalino de bromuro de (1alfa, 2beta, 4beta, 5alfa, 7beta)-7-[(hidroxi-di-2-tienil-acetil)oxi]-9,9-dimetil-3-oxa-9-azonia-triciclo[3.3.1.02,4]nonano, a un procedimiento para su preparación, así como a su utilización para la preparación de un medicamento, particularmente para la preparación de un medicamento con efecto anticolinérgico.
ARP010104782A 2000-10-12 2001-10-12 Monohidrato cristalino de bromuro de tiotropio, procedimiento para su preparacion, su utilización para la preparacion de un medicamento, un medicamento que lo contiene, los hidratos cristalinos del bromuro de tiotropio y un procedimiento para preparacion de estos hidratos cristalinos Pending AR034389A1 (es)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
DE10050621 2000-10-12

Publications (1)

Publication Number Publication Date
AR034389A1 true AR034389A1 (es) 2004-02-25

Family

ID=7659568

Family Applications (2)

Application Number Title Priority Date Filing Date
ARP010104782A Pending AR034389A1 (es) 2000-10-12 2001-10-12 Monohidrato cristalino de bromuro de tiotropio, procedimiento para su preparacion, su utilización para la preparacion de un medicamento, un medicamento que lo contiene, los hidratos cristalinos del bromuro de tiotropio y un procedimiento para preparacion de estos hidratos cristalinos
ARP080104109A AR068527A2 (es) 2000-10-12 2008-09-19 Un procedimiento para preparar monohidrato de bromuro de tiotropio cristalino

Family Applications After (1)

Application Number Title Priority Date Filing Date
ARP080104109A AR068527A2 (es) 2000-10-12 2008-09-19 Un procedimiento para preparar monohidrato de bromuro de tiotropio cristalino

Country Status (47)

Country Link
EP (2) EP1468998A1 (es)
JP (1) JP3764422B2 (es)
KR (1) KR100823860B1 (es)
CN (2) CN1221549C (es)
AP (1) AP1572A (es)
AR (2) AR034389A1 (es)
AT (1) ATE276253T1 (es)
AU (2) AU2002214996B2 (es)
BG (1) BG66161B1 (es)
BR (1) BR0114584A (es)
CA (1) CA2425539C (es)
CR (1) CR6938A (es)
CZ (1) CZ301841B6 (es)
DE (1) DE50103666D1 (es)
DK (1) DK1326862T3 (es)
DZ (1) DZ3478A1 (es)
EA (1) EA004381B1 (es)
EC (1) ECSP034540A (es)
EE (1) EE04567B1 (es)
EG (1) EG24142A (es)
ES (1) ES2228965T3 (es)
GE (1) GEP20063905B (es)
HK (2) HK1060567A1 (es)
HR (1) HRP20030276B1 (es)
HU (1) HU226830B1 (es)
IL (2) IL155335A0 (es)
IS (1) IS2339B (es)
MA (1) MA25842A1 (es)
ME (2) ME00243B (es)
MX (1) MXPA03003221A (es)
MY (1) MY126931A (es)
NO (1) NO328465B1 (es)
NZ (1) NZ525733A (es)
OA (1) OA12403A (es)
PE (1) PE20020422A1 (es)
PL (1) PL207870B1 (es)
PT (1) PT1326862E (es)
RS (1) RS50218B (es)
SA (1) SA01220412B1 (es)
SI (1) SI1326862T1 (es)
SK (1) SK287009B6 (es)
TR (1) TR200402579T4 (es)
TW (1) TW589313B (es)
UA (1) UA74215C2 (es)
UY (2) UY26962A1 (es)
WO (1) WO2002030928A1 (es)
ZA (1) ZA200302500B (es)

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Publication number Publication date
NZ525733A (en) 2005-01-28
HRP20030276B1 (en) 2006-02-28
JP2004526668A (ja) 2004-09-02
KR100823860B1 (ko) 2008-04-21
NO328465B1 (no) 2010-02-22
CZ301841B6 (cs) 2010-07-07
MXPA03003221A (es) 2004-12-03
NO20031694D0 (no) 2003-04-11
MA25842A1 (fr) 2003-07-01
BG107687A (bg) 2003-09-30
ES2228965T3 (es) 2005-04-16
SK4362003A3 (en) 2003-08-05
KR20030042008A (ko) 2003-05-27
BG66161B1 (bg) 2011-09-30
JP3764422B2 (ja) 2006-04-05
HK1086557A1 (en) 2006-09-22
AP1572A (en) 2006-02-13
HK1060567A1 (en) 2004-08-13
UA74215C2 (uk) 2005-11-15
CN1733761A (zh) 2006-02-15
EP1326862A1 (de) 2003-07-16
IL155335A (en) 2009-02-11
DK1326862T3 (da) 2004-11-22
PE20020422A1 (es) 2002-06-28
YU27303A (sh) 2006-05-25
CR6938A (es) 2004-10-28
AR068527A2 (es) 2009-11-18
DZ3478A1 (fr) 2002-04-18
IS2339B (is) 2008-02-15
SI1326862T1 (en) 2005-02-28
ZA200302500B (en) 2004-04-22
DE50103666D1 (de) 2004-10-21
SK287009B6 (sk) 2009-09-07
CA2425539A1 (en) 2003-04-11
AU1499602A (en) 2002-04-22
EA200300457A1 (ru) 2003-10-30
HUP0301022A2 (hu) 2003-10-28
BR0114584A (pt) 2003-08-26
WO2002030928A1 (de) 2002-04-18
TW589313B (en) 2004-06-01
EA004381B1 (ru) 2004-04-29
AU2002214996B2 (en) 2007-03-15
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RS50218B (sr) 2009-07-15
UY34901A (es) 2015-02-27
CN1469877A (zh) 2004-01-21
CN100519558C (zh) 2009-07-29
TR200402579T4 (tr) 2004-12-21
OA12403A (en) 2006-04-18
MY126931A (en) 2006-10-31
EP1468998A1 (de) 2004-10-20
ME00243B (me) 2011-05-10
GEP20063905B (en) 2006-08-25
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IL155335A0 (en) 2003-11-23
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AP2003002775A0 (en) 2003-03-31
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IS6772A (is) 2003-04-09
HRP20030276A2 (en) 2005-02-28
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