EE200300171A - Kristalliline monohüdraat, meetodid selle valmistamiseks ja selle kasutamine farmatseutilise kompositsiooni valmistamiseks - Google Patents

Kristalliline monohüdraat, meetodid selle valmistamiseks ja selle kasutamine farmatseutilise kompositsiooni valmistamiseks

Info

Publication number
EE200300171A
EE200300171A EEP200300171A EEP200300171A EE200300171A EE 200300171 A EE200300171 A EE 200300171A EE P200300171 A EEP200300171 A EE P200300171A EE P200300171 A EEP200300171 A EE P200300171A EE 200300171 A EE200300171 A EE 200300171A
Authority
EE
Estonia
Prior art keywords
preparation
methods
pharmaceutical composition
crystalline monohydrate
monohydrate
Prior art date
Application number
EEP200300171A
Other languages
English (en)
Inventor
Banholzer Rolf
Sieger Peter
Kulinna Christian
Trunk Michael
Ludwig August Graulich Manfred
Specht Peter
Meissner Helmut
Mathes Andreas
Original Assignee
Boehringer Ingelheim Pharma Gmbh & Co. Kg
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Family has litigation
First worldwide family litigation filed litigation Critical https://patents.darts-ip.com/?family=7659568&utm_source=google_patent&utm_medium=platform_link&utm_campaign=public_patent_search&patent=EE200300171(A) "Global patent litigation dataset” by Darts-ip is licensed under a Creative Commons Attribution 4.0 International License.
Application filed by Boehringer Ingelheim Pharma Gmbh & Co. Kg filed Critical Boehringer Ingelheim Pharma Gmbh & Co. Kg
Publication of EE200300171A publication Critical patent/EE200300171A/et
Publication of EE04567B1 publication Critical patent/EE04567B1/et

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D451/00—Heterocyclic compounds containing 8-azabicyclo [3.2.1] octane, 9-azabicyclo [3.3.1] nonane, or 3-oxa-9-azatricyclo [3.3.1.0<2,4>] nonane ring systems, e.g. tropane or granatane alkaloids, scopolamine; Cyclic acetals thereof
    • C07D451/02—Heterocyclic compounds containing 8-azabicyclo [3.2.1] octane, 9-azabicyclo [3.3.1] nonane, or 3-oxa-9-azatricyclo [3.3.1.0<2,4>] nonane ring systems, e.g. tropane or granatane alkaloids, scopolamine; Cyclic acetals thereof containing not further condensed 8-azabicyclo [3.2.1] octane or 3-oxa-9-azatricyclo [3.3.1.0<2,4>] nonane ring systems, e.g. tropane; Cyclic acetals thereof
    • C07D451/04—Heterocyclic compounds containing 8-azabicyclo [3.2.1] octane, 9-azabicyclo [3.3.1] nonane, or 3-oxa-9-azatricyclo [3.3.1.0<2,4>] nonane ring systems, e.g. tropane or granatane alkaloids, scopolamine; Cyclic acetals thereof containing not further condensed 8-azabicyclo [3.2.1] octane or 3-oxa-9-azatricyclo [3.3.1.0<2,4>] nonane ring systems, e.g. tropane; Cyclic acetals thereof with hetero atoms directly attached in position 3 of the 8-azabicyclo [3.2.1] octane or in position 7 of the 3-oxa-9-azatricyclo [3.3.1.0<2,4>] nonane ring system
    • C07D451/06—Oxygen atoms
    • C07D451/10—Oxygen atoms acylated by aliphatic or araliphatic carboxylic acids, e.g. atropine, scopolamine
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P11/00—Drugs for disorders of the respiratory system
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P11/00—Drugs for disorders of the respiratory system
    • A61P11/06—Antiasthmatics
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P11/00—Drugs for disorders of the respiratory system
    • A61P11/16—Central respiratory analeptics
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00—Drugs for disorders of the nervous system
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P43/00—Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00
EEP200300171A 2000-10-12 2001-09-28 Kristalliline monohdraat, meetod selle valmistamiseks ja selle kasutamine ravimi valmistamiseks EE04567B1 (et)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
DE10050621 2000-10-12
PCT/EP2001/011225 WO2002030928A1 (de) 2000-10-12 2001-09-28 Kristallines monohydrat, verfahren zu dessen herstellung und dessen verwendung zur herstellung eines arzneimittels

Publications (2)

Publication Number Publication Date
EE200300171A true EE200300171A (et) 2003-06-16
EE04567B1 EE04567B1 (et) 2005-12-15

Family

ID=7659568

Family Applications (1)

Application Number Title Priority Date Filing Date
EEP200300171A EE04567B1 (et) 2000-10-12 2001-09-28 Kristalliline monohdraat, meetod selle valmistamiseks ja selle kasutamine ravimi valmistamiseks

Country Status (47)

Country Link
EP (2) EP1326862B1 (et)
JP (1) JP3764422B2 (et)
KR (1) KR100823860B1 (et)
CN (2) CN100519558C (et)
AP (1) AP1572A (et)
AR (2) AR034389A1 (et)
AT (1) ATE276253T1 (et)
AU (2) AU1499602A (et)
BG (1) BG66161B1 (et)
BR (1) BR0114584A (et)
CA (1) CA2425539C (et)
CR (1) CR6938A (et)
CZ (1) CZ301841B6 (et)
DE (1) DE50103666D1 (et)
DK (1) DK1326862T3 (et)
DZ (1) DZ3478A1 (et)
EA (1) EA004381B1 (et)
EC (1) ECSP034540A (et)
EE (1) EE04567B1 (et)
EG (1) EG24142A (et)
ES (1) ES2228965T3 (et)
GE (1) GEP20063905B (et)
HK (2) HK1060567A1 (et)
HR (1) HRP20030276B1 (et)
HU (1) HU226830B1 (et)
IL (2) IL155335A0 (et)
IS (1) IS2339B (et)
MA (1) MA25842A1 (et)
ME (2) ME00243B (et)
MX (1) MXPA03003221A (et)
MY (1) MY126931A (et)
NO (1) NO328465B1 (et)
NZ (1) NZ525733A (et)
OA (1) OA12403A (et)
PE (1) PE20020422A1 (et)
PL (1) PL207870B1 (et)
PT (1) PT1326862E (et)
RS (1) RS50218B (et)
SA (1) SA01220412B1 (et)
SI (1) SI1326862T1 (et)
SK (1) SK287009B6 (et)
TR (1) TR200402579T4 (et)
TW (1) TW589313B (et)
UA (1) UA74215C2 (et)
UY (2) UY26962A1 (et)
WO (1) WO2002030928A1 (et)
ZA (1) ZA200302500B (et)

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Also Published As

Publication number Publication date
SI1326862T1 (en) 2005-02-28
KR20030042008A (ko) 2003-05-27
CZ301841B6 (cs) 2010-07-07
IS2339B (is) 2008-02-15
ME00243B (me) 2011-05-10
HRP20030276B1 (en) 2006-02-28
SK4362003A3 (en) 2003-08-05
UY34901A (es) 2015-02-27
AU1499602A (en) 2002-04-22
HK1060567A1 (en) 2004-08-13
PT1326862E (pt) 2004-11-30
EG24142A (en) 2008-08-06
YU27303A (sh) 2006-05-25
DZ3478A1 (fr) 2002-04-18
SK287009B6 (sk) 2009-09-07
HK1086557A1 (en) 2006-09-22
CN1221549C (zh) 2005-10-05
SA01220412B1 (ar) 2006-11-05
WO2002030928A1 (de) 2002-04-18
TR200402579T4 (tr) 2004-12-21
BG66161B1 (bg) 2011-09-30
ZA200302500B (en) 2004-04-22
PL207870B1 (pl) 2011-02-28
EE04567B1 (et) 2005-12-15
GEP20063905B (en) 2006-08-25
AP1572A (en) 2006-02-13
NO328465B1 (no) 2010-02-22
MEP40008A (en) 2011-02-10
HU226830B1 (en) 2009-11-30
RS50218B (sr) 2009-07-15
IS6772A (is) 2003-04-09
EP1326862A1 (de) 2003-07-16
PL366041A1 (en) 2005-01-24
HUP0301022A3 (en) 2005-12-28
JP2004526668A (ja) 2004-09-02
CN1733761A (zh) 2006-02-15
ECSP034540A (es) 2003-07-25
NO20031694L (no) 2003-04-11
MY126931A (en) 2006-10-31
CN1469877A (zh) 2004-01-21
CA2425539C (en) 2007-04-03
AR068527A2 (es) 2009-11-18
AU2002214996B2 (en) 2007-03-15
EP1326862B1 (de) 2004-09-15
UA74215C2 (uk) 2005-11-15
HUP0301022A2 (hu) 2003-10-28
ES2228965T3 (es) 2005-04-16
DE50103666D1 (de) 2004-10-21
OA12403A (en) 2006-04-18
CA2425539A1 (en) 2003-04-11
TW589313B (en) 2004-06-01
IL155335A0 (en) 2003-11-23
NZ525733A (en) 2005-01-28
EP1468998A1 (de) 2004-10-20
AR034389A1 (es) 2004-02-25
IL155335A (en) 2009-02-11
DK1326862T3 (da) 2004-11-22
MA25842A1 (fr) 2003-07-01
BG107687A (bg) 2003-09-30
EA004381B1 (ru) 2004-04-29
NO20031694D0 (no) 2003-04-11
AP2003002775A0 (en) 2003-03-31
HRP20030276A2 (en) 2005-02-28
MXPA03003221A (es) 2004-12-03
ATE276253T1 (de) 2004-10-15
KR100823860B1 (ko) 2008-04-21
PE20020422A1 (es) 2002-06-28
CN100519558C (zh) 2009-07-29
CR6938A (es) 2004-10-28
JP3764422B2 (ja) 2006-04-05
UY26962A1 (es) 2002-06-20
BR0114584A (pt) 2003-08-26
EA200300457A1 (ru) 2003-10-30

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