EE05104B1 - Asetidiini derivaadid, nende valmistamise meetodid ja farmatseutiline kompositsioon - Google Patents

Asetidiini derivaadid, nende valmistamise meetodid ja farmatseutiline kompositsioon

Info

Publication number
EE05104B1
EE05104B1 EEP200200487A EEP200200487A EE05104B1 EE 05104 B1 EE05104 B1 EE 05104B1 EE P200200487 A EEP200200487 A EE P200200487A EE P200200487 A EEP200200487 A EE P200200487A EE 05104 B1 EE05104 B1 EE 05104B1
Authority
EE
Estonia
Prior art keywords
preparation
methods
pharmaceutical composition
azetidine derivatives
azetidine
Prior art date
Application number
EEP200200487A
Other languages
English (en)
Inventor
Achard Daniel
Bouchard Herv
Bouquerel Jean
Filoche Bruno
Grisoni Serge
Hittinger Augustin
Myers Michael
Original Assignee
Aventis Pharma S.A.
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Aventis Pharma S.A. filed Critical Aventis Pharma S.A.
Publication of EE200200487A publication Critical patent/EE200200487A/et
Publication of EE05104B1 publication Critical patent/EE05104B1/et

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    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D401/00—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom
    • C07D401/02—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings
    • C07D401/06—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings linked by a carbon chain containing only aliphatic carbon atoms
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    • A61P1/08—Drugs for disorders of the alimentary tract or the digestive system for nausea, cinetosis or vertigo; Antiemetics
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    • C07D205/04—Heterocyclic compounds containing four-membered rings with one nitrogen atom as the only ring hetero atom not condensed with other rings having no double bonds between ring members or between ring members and non-ring members
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    • C07D403/10—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, not provided for by group C07D401/00 containing two hetero rings linked by a carbon chain containing aromatic rings
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    • C07D403/12—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, not provided for by group C07D401/00 containing two hetero rings linked by a chain containing hetero atoms as chain links
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    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D403/00—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, not provided for by group C07D401/00
    • C07D403/14—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, not provided for by group C07D401/00 containing three or more hetero rings
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    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D409/00—Heterocyclic compounds containing two or more hetero rings, at least one ring having sulfur atoms as the only ring hetero atoms
    • C07D409/02—Heterocyclic compounds containing two or more hetero rings, at least one ring having sulfur atoms as the only ring hetero atoms containing two hetero rings
    • C07D409/06—Heterocyclic compounds containing two or more hetero rings, at least one ring having sulfur atoms as the only ring hetero atoms containing two hetero rings linked by a carbon chain containing only aliphatic carbon atoms
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D409/00—Heterocyclic compounds containing two or more hetero rings, at least one ring having sulfur atoms as the only ring hetero atoms
    • C07D409/02—Heterocyclic compounds containing two or more hetero rings, at least one ring having sulfur atoms as the only ring hetero atoms containing two hetero rings
    • C07D409/12—Heterocyclic compounds containing two or more hetero rings, at least one ring having sulfur atoms as the only ring hetero atoms containing two hetero rings linked by a chain containing hetero atoms as chain links
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D409/00—Heterocyclic compounds containing two or more hetero rings, at least one ring having sulfur atoms as the only ring hetero atoms
    • C07D409/14—Heterocyclic compounds containing two or more hetero rings, at least one ring having sulfur atoms as the only ring hetero atoms containing three or more hetero rings

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  • Health & Medical Sciences (AREA)
  • Organic Chemistry (AREA)
  • Chemical & Material Sciences (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Engineering & Computer Science (AREA)
  • Veterinary Medicine (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • General Health & Medical Sciences (AREA)
  • Public Health (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Medicinal Chemistry (AREA)
  • General Chemical & Material Sciences (AREA)
  • Neurosurgery (AREA)
  • Biomedical Technology (AREA)
  • Neurology (AREA)
  • Pain & Pain Management (AREA)
  • Psychiatry (AREA)
  • Addiction (AREA)
  • Heart & Thoracic Surgery (AREA)
  • Cardiology (AREA)
  • Ophthalmology & Optometry (AREA)
  • Pulmonology (AREA)
  • Diabetes (AREA)
  • Anesthesiology (AREA)
  • Hematology (AREA)
  • Endocrinology (AREA)
  • Psychology (AREA)
  • Reproductive Health (AREA)
  • Hospice & Palliative Care (AREA)
  • Pregnancy & Childbirth (AREA)
  • Child & Adolescent Psychology (AREA)
  • Gynecology & Obstetrics (AREA)
  • Immunology (AREA)
  • Rheumatology (AREA)
  • Obesity (AREA)
  • Otolaryngology (AREA)
  • Nutrition Science (AREA)
EEP200200487A 2000-03-03 2001-03-01 Asetidiini derivaadid, nende valmistamise meetodid ja farmatseutiline kompositsioon EE05104B1 (et)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
FR0002775A FR2805818B1 (fr) 2000-03-03 2000-03-03 Derives d'azetidine, leur preparation et les compositions pharmaceutiques les contenant
PCT/FR2001/000600 WO2001064632A1 (fr) 2000-03-03 2001-03-01 Derives d'azetidine, leur preparation et les compositions pharmaceutiques les contenant

Publications (2)

Publication Number Publication Date
EE200200487A EE200200487A (et) 2004-02-16
EE05104B1 true EE05104B1 (et) 2008-12-15

Family

ID=8847705

Family Applications (1)

Application Number Title Priority Date Filing Date
EEP200200487A EE05104B1 (et) 2000-03-03 2001-03-01 Asetidiini derivaadid, nende valmistamise meetodid ja farmatseutiline kompositsioon

Country Status (37)

Country Link
EP (1) EP1263720B1 (et)
JP (1) JP2003525268A (et)
KR (1) KR100786411B1 (et)
CN (1) CN1185213C (et)
AR (1) AR027608A1 (et)
AT (1) ATE432919T1 (et)
AU (2) AU3752501A (et)
BG (1) BG107056A (et)
BR (1) BR0108871A (et)
CA (1) CA2400116A1 (et)
CY (1) CY1109343T1 (et)
CZ (1) CZ20022931A3 (et)
DE (1) DE60138872D1 (et)
DK (1) DK1263720T3 (et)
DZ (1) DZ3313A1 (et)
EA (1) EA006583B1 (et)
EE (1) EE05104B1 (et)
ES (1) ES2328104T3 (et)
FR (1) FR2805818B1 (et)
HR (1) HRP20020711A2 (et)
HU (1) HUP0301404A3 (et)
IL (2) IL151428A0 (et)
MA (1) MA26877A1 (et)
ME (1) MEP24608A (et)
MX (1) MXPA02008360A (et)
NO (1) NO324505B1 (et)
NZ (1) NZ521075A (et)
OA (1) OA12220A (et)
PL (1) PL357534A1 (et)
PT (1) PT1263720E (et)
RS (1) RS50417B (et)
SI (1) SI1263720T1 (et)
SK (1) SK12452002A3 (et)
TW (1) TWI230153B (et)
UA (1) UA72593C2 (et)
WO (1) WO2001064632A1 (et)
ZA (1) ZA200206905B (et)

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AU2002319627A1 (en) 2001-07-20 2003-03-03 Merck And Co., Inc. Substituted imidazoles as cannabinoid receptor modulators
FR2833842B1 (fr) * 2001-12-21 2004-02-13 Aventis Pharma Sa Compositions pharmaceutiques a base de derives d'azetidine
CA2478183C (en) 2002-03-12 2010-02-16 Merck & Co. Inc. Substituted amides
US7105526B2 (en) 2002-06-28 2006-09-12 Banyu Pharmaceuticals Co., Ltd. Benzimidazole derivatives
AU2003250117B2 (en) 2002-07-29 2007-05-10 F. Hoffmann-La Roche Ag Novel benzodioxoles
DE60322114D1 (de) 2003-01-02 2008-08-21 Hoffmann La Roche Pyrrolyl-thiazole und ihre verwendung als inverse agonisten des cb 1 rezeptors
EP1583742B1 (en) 2003-01-02 2009-12-02 F. Hoffmann-La Roche Ag Cb 1 receptour inverse agonists
US7772188B2 (en) 2003-01-28 2010-08-10 Ironwood Pharmaceuticals, Inc. Methods and compositions for the treatment of gastrointestinal disorders
WO2004089927A1 (en) * 2003-04-07 2004-10-21 Cortical Pty Ltd Novel methods for the treatment of inflammatory diseases
FR2854633B1 (fr) * 2003-05-07 2005-06-24 Sanofi Synthelabo Derives de piperidinyl-et piperazinyl-alkylcarbamates, leur preparation et leur application en therapeutique
NZ543451A (en) * 2003-06-11 2008-08-29 Merck & Co Inc Substituted 3-alkyl and 3-alkenyl azetidine derivitives
RU2344132C2 (ru) 2003-06-20 2009-01-20 Ф.Хоффманн-Ля Рош Аг 2-аминобензотиазолы в качестве обратных агонистов рецепторов cb1
GB0320983D0 (en) * 2003-09-08 2003-10-08 Biofocus Plc Compound libraries
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